NO180780C - Pyridonkarboksylsyrederivat - Google Patents

Pyridonkarboksylsyrederivat

Info

Publication number: NO180780C
Authority: NO; Norway
Prior art keywords: represent; various; derivatives; carboxylic acid; acid derivative
Prior art date: 1991-05-28

Application number

NO934279A

Other languages

English (en)

Norwegian (no)

Other versions

NO934279L (no

NO180780B (no

NO934279D0 (no

Inventor

Isao Hayakawa

Youichi Kimura

Hisashi Takahashi

Original Assignee

Daiichi Seiyaku Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-05-28

Filing date

1993-11-26

Publication date

1997-06-18

1993-11-26 Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co

1993-11-26 Publication of NO934279D0 publication Critical patent/NO934279D0/no

1994-01-28 Publication of NO934279L publication Critical patent/NO934279L/no

1997-03-10 Publication of NO180780B publication Critical patent/NO180780B/no

1997-06-18 Publication of NO180780C publication Critical patent/NO180780C/no

Links

YSLIPUSJNFIFAB-UHFFFAOYSA-N 2-oxopyridine-1-carboxylic acid Chemical class OC(=O)N1C=CC=CC1=O YSLIPUSJNFIFAB-UHFFFAOYSA-N 0.000 title abstract 2
IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
230000000844 anti-bacterial effect Effects 0.000 abstract 2
150000007660 quinolones Chemical class 0.000 abstract 2
229940088710 antibiotic agent Drugs 0.000 abstract 1
125000001028 difluoromethyl group Chemical group [H]C(F)(F)* 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
125000000623 heterocyclic group Chemical group 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyridine Compounds (AREA)
Cephalosporin Compounds (AREA)
Quinoline Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Stringed Musical Instruments (AREA)
Table Devices Or Equipment (AREA)

NO934279A 1991-05-28 1993-11-26 Pyridonkarboksylsyrederivat NO180780C (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP22542591		1991-05-28
PCT/JP1992/000687 WO1992021659A1 (fr)	1991-05-28	1992-05-27	Derive d'acide pyridonecarboxylique

Publications (4)

Publication Number	Publication Date
NO934279D0 NO934279D0 (no)	1993-11-26
NO934279L NO934279L (no)	1994-01-28
NO180780B NO180780B (no)	1997-03-10
NO180780C true NO180780C (no)	1997-06-18

Family

ID=16829173

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO934279A NO180780C (no)	1991-05-28	1993-11-26	Pyridonkarboksylsyrederivat

Country Status (16)

Country	Link
US (1)	US5696132A (de)
EP (1)	EP0593766B1 (de)
JP (1)	JP3215500B2 (de)
KR (1)	KR100232937B1 (de)
AT (1)	ATE196135T1 (de)
AU (1)	AU661999B2 (de)
CA (1)	CA2110260C (de)
DE (1)	DE69231422T2 (de)
DK (1)	DK0593766T3 (de)
ES (1)	ES2151488T3 (de)
FI (1)	FI109201B (de)
GR (1)	GR3034966T3 (de)
NO (1)	NO180780C (de)
RU (1)	RU2100351C1 (de)
TW (1)	TW212179B (de)
WO (1)	WO1992021659A1 (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP3165742B2 (ja) *	1991-07-16	2001-05-14	中外製薬株式会社	キノロンカルボン酸誘導体の製造方法
NO304832B1 (no) *	1992-05-27	1999-02-22	Ube Industries	Aminokinolonderivater samt middel mot HIV
CA2112165C (en) *	1992-12-25	2003-04-08	Makoto Takemura	Bicyclic amine derivatives
DE4339134A1 (de) *	1993-11-16	1995-05-18	Bayer Ag	1-(2-Fluorcyclopropyl)-chinolon- und -naphthyridoncarbonsäure-Derivate
DE4408212A1 (de) *	1994-03-11	1995-09-14	Bayer Ag	5-Vinyl- und 5-Ethinyl-chinolon- und -naphthyridon-carbonsäuren
WO1996023782A1 (en) *	1995-02-02	1996-08-08	Daiichi Pharmaceutical Co., Ltd.	Heterocyclic compounds
WO1996024593A1 (en)	1995-02-07	1996-08-15	Daiichi Pharmaceutical Co., Ltd.	Heterocyclic spiro derivatives
KR19990071558A (ko) *	1995-11-22	1999-09-27	스즈키 다다시	치환된 아미노시클로알킬피롤리딘 유도체
US6121285A (en)	1995-11-22	2000-09-19	Daiichi Pharmaceutical Co., Ltd.	Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
AU1040597A (en) *	1996-12-04	1998-06-29	Daiichi Pharmaceutical Co., Ltd.	Substituted aminomethylpyrrolidine derivatives
JPH1149698A (ja)	1997-07-31	1999-02-23	Santen Pharmaceut Co Ltd	安定性を向上させたラクトフェリンの水性製剤
WO2005111015A1 (ja) *	2004-05-13	2005-11-24	Daiichi Pharmaceutical Co., Ltd.	置換ピロリジン誘導体
JP3995705B2 (ja) *	2004-11-17	2007-10-24	湧永製薬株式会社	新規ピリドンカルボン酸誘導体又はその塩
US7563805B2 (en) *	2005-05-19	2009-07-21	Daiichi Pharmaceutical Co., Ltd.	Tri-, tetra-substituted-3-aminopyrrolidine derivative
US7977346B2 (en)	2006-01-17	2011-07-12	Guoqing Paul Chen	Spiro compounds and methods of use
CN105330590B (zh) *	2015-10-15	2018-09-25	广州市朗启医药科技有限责任公司	西他沙星五元环侧链中间体的制备方法
CN109942488A (zh) *	2019-04-04	2019-06-28	山东省联合农药工业有限公司	一种喹啉羧酸酯类化合物及其制备方法与用途

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS6028978A (ja) *	1983-07-27	1985-02-14	Dainippon Pharmaceut Co Ltd	１，８−ナフチリジン誘導体
JPS6212760A (ja) *	1984-12-14	1987-01-21	Dai Ichi Seiyaku Co Ltd	１−（２−ハロゲノシクロプロピル）キノリンカルボン酸誘導体
DE3509546A1 (de) *	1985-03-16	1986-09-25	Bayer Ag, 5090 Leverkusen	7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3705621C2 (de) *	1986-02-25	1997-01-09	Otsuka Pharma Co Ltd	Heterocyclisch substituierte Chinoloncarbonsäurederivate
DE3702393A1 (de) *	1987-01-28	1988-08-11	Bayer Ag	8-cyano-1-cyclopropyl-1,4-dihydro-4-oxo- 3-chinolincarbonsaeuren, verfahren zu ihrer herstellung und diese enthaltende antibakterielle mittel
US5563138A (en) *	1987-04-16	1996-10-08	Otsuka Pharmaceutical Company, Limited	Benzoheterocyclic compounds
US4851418A (en) *	1987-08-21	1989-07-25	Warner-Lambert Company	Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
IL90062A (en) *	1988-04-27	1994-10-07	Daiichi Seiyaku Co	Pyridonecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
DE3906365A1 (de) *	1988-07-15	1990-01-18	Bayer Ag	7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
US5057520A (en) *	1989-03-24	1991-10-15	Abbott Laboratories	7-(peptidylpyrolidinyl)naphthyridine antibacterial compounds
DE69019859T2 (de) *	1989-03-30	1995-10-05	Wakunaga Seiyaku Kk	Chinolon-Derivate und deren Salze, Verfahren zu deren Herstellung und diese enthaltende antibakterielle Wirkstoffe.
US5140033A (en) *	1989-04-03	1992-08-18	Bayer Aktiengesellschaft	Antibacterial 5-alkylquinolonecarboxylic acids
US5252734A (en) *	1989-04-03	1993-10-12	Bayer Aktiengesellschaft	Antibacterial 5-alkylquinolonecarboxylic acids
DE3910663A1 (de) *	1989-04-03	1990-10-04	Bayer Ag	5-alkylchinoloncarbonsaeuren
DE3918544A1 (de) *	1989-06-07	1990-12-13	Bayer Ag	Verfahren zur herstellung von 7-(3-amino- sowie 3-amino-methyl-1-pyrrolidinyl)-3-chinolon- carbonsaeuren sowie -naphthyridoncarbonsaeuren
MY109714A (en) *	1990-10-18	1997-04-30	Daiichi Seiyaku Co	Process for preparing 8-chloroquinolone derivatives
US5072001A (en) *	1990-11-30	1991-12-10	Warner-Lambert Company	Certain optically active substituted 3-pyrraidine acetic acid derivatives useful as intermediates
US5137892A (en) *	1990-12-12	1992-08-11	Abbott Laboratories	Quinoline, naphthyridine and pyridobenzoxazine derivatives

1992
- 1992-05-27 DE DE69231422T patent/DE69231422T2/de not_active Expired - Fee Related
- 1992-05-27 KR KR1019930703606A patent/KR100232937B1/ko not_active Expired - Fee Related
- 1992-05-27 AT AT92910698T patent/ATE196135T1/de not_active IP Right Cessation
- 1992-05-27 DK DK92910698T patent/DK0593766T3/da active
- 1992-05-27 US US08/142,444 patent/US5696132A/en not_active Expired - Fee Related
- 1992-05-27 CA CA002110260A patent/CA2110260C/en not_active Expired - Fee Related
- 1992-05-27 ES ES92910698T patent/ES2151488T3/es not_active Expired - Lifetime
- 1992-05-27 EP EP92910698A patent/EP0593766B1/de not_active Expired - Lifetime
- 1992-05-27 RU RU93058417/04A patent/RU2100351C1/ru not_active IP Right Cessation
- 1992-05-27 AU AU18872/92A patent/AU661999B2/en not_active Ceased
- 1992-05-27 WO PCT/JP1992/000687 patent/WO1992021659A1/ja not_active Ceased
- 1992-05-28 JP JP13650492A patent/JP3215500B2/ja not_active Expired - Fee Related
- 1992-05-29 TW TW081104208A patent/TW212179B/zh active
1993
- 1993-11-25 FI FI935243A patent/FI109201B/fi not_active IP Right Cessation
- 1993-11-26 NO NO934279A patent/NO180780C/no not_active IP Right Cessation
2000
- 2000-11-30 GR GR20000402669T patent/GR3034966T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
NO934279L (no)	1994-01-28
GR3034966T3 (en)	2001-02-28
FI935243L (fi)	1994-01-11
NO180780B (no)	1997-03-10
DE69231422D1 (de)	2000-10-12
AU1887292A (en)	1993-01-08
CA2110260A1 (en)	1992-12-10
DE69231422T2 (de)	2001-03-29
ES2151488T3 (es)	2001-01-01
CA2110260C (en)	2001-12-04
EP0593766A4 (de)	1994-12-07
US5696132A (en)	1997-12-09
NO934279D0 (no)	1993-11-26
AU661999B2 (en)	1995-08-17
ATE196135T1 (de)	2000-09-15
JP3215500B2 (ja)	2001-10-09
EP0593766A1 (de)	1994-04-27
RU2100351C1 (ru)	1997-12-27
JPH05163244A (ja)	1993-06-29
WO1992021659A1 (fr)	1992-12-10
FI935243A0 (fi)	1993-11-25
KR100232937B1 (ko)	1999-12-01
FI109201B (fi)	2002-06-14
EP0593766B1 (de)	2000-09-06
TW212179B (de)	1993-09-01
DK0593766T3 (da)	2000-10-09

Legal Events

Date	Code	Title	Description
2005-01-03	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
ATE196135T1 (de)	2000-09-15	Pyridoncarbonsäurederivate
ATE194835T1 (de)	2000-08-15	Pyridazinonderivat
DK0655996T3 (da)	2001-12-27	Substituerede benzylamino-nitrogenholdige, ikke-aromatiske, heterocykliske forbindelser
CA2109613A1 (en)	1993-01-07	Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
DK0937048T3 (da)	2004-04-19	Heterocykliske derivater, der inhiberer faktor Xa
NZ228893A (en)	1990-06-26	Substituted quinoline and naphthyridine derivatives and pharmaceutical compositions
HUT62893A (en)	1993-06-28	Process for producing substituted pyrimidine derivatives and pharmaceutical compositions comprising such compounds as active ingredient
ATE227293T1 (de)	2002-11-15	2,3-disubstituierte-(5,6)-heteroarylkondensiert - pyrimidin-4-one
DE69426773D1 (de)	2001-04-05	Pyrazol-derivate
HUT61004A (en)	1992-11-30	Process for producing quinoxaline derivatives and pharmaceutical compositions comprising such compounds as active ingredient
EE03215B1 (et)	1999-08-16	3-kinoloonkarboksüülhappe derivaatide ühereaktoriline saamismeetod
NO306992B1 (no)	2000-01-24	Quinolinderivater, farmasoeytiske preparater inneholdende forbindelsene og anvendelsen av forbindelsene
ATE411309T1 (de)	2008-10-15	Pyridonkarbonsaüre derivate und deren verwendung als antibakterielle wirkstoffe
BG50163A3 (bg)	1992-05-15	Метод за получаване на ацилови производни
RU93058417A (ru)	1996-12-27	Производные пиридон-карбоновой кислоты, антимикробный агент
DE69128630D1 (de)	1998-02-12	Benzopyran derivat, seine darstellung und pharmazeutische zusammensetzung, welche dieses enthält
ATE202555T1 (de)	2001-07-15	Cyclohexandiharnstoff-derivate und verfahren zu deren herstellung
ZA937085B (en)	1994-08-11	e derivatives active on the cardiovascular system 17-Aryl and 17-heterocyclyl-5Beta-14Beta androstanprocesses for their preparation and pharmaceutical compositions containing same
AU1659192A (en)	1992-12-30	Novel 2h-benzo(b)pyrane derivatives substituted in the 4 position by aryl or n-heteroaryl, process for producing them and preparations containing the compounds
ITMI920082A1 (it)	1993-07-17	Derivati solforati di acidi biliari
AP9400608A0 (en)	1995-07-12	"New nicotinic acid derivative".
MX9803557A (es)	1998-09-30	Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producir tales compuestos.
MX9803556A (es)	1998-09-30	Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producirlos.