NO20005769L - cyclosporin derivatives - Google Patents

cyclosporin derivatives

Info

Publication number: NO20005769L
Authority: NO; Norway
Prior art keywords: cyclosporin derivatives; cyclosporin; derivatives
Prior art date: 1998-05-15

Application number

NO20005769A

Other languages

Norwegian (no)

Other versions

NO20005769D0 (en

Inventor

Robert Heger

Helmut Auweter

Peter Pflueger

Joerg Breitenbach

Rudolf Binder

Juergen Zeidler

Gunther Berndl

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-05-15

Filing date

2000-11-14

Publication date

2000-11-14

2000-11-14 Application filed by Basf Ag filed Critical Basf Ag

2000-11-14 Publication of NO20005769L publication Critical patent/NO20005769L/en

2000-11-14 Publication of NO20005769D0 publication Critical patent/NO20005769D0/en

Links

PMATZTZNYRCHOR-CGLBZJNRSA-N Cyclosporin A Chemical class CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O PMATZTZNYRCHOR-CGLBZJNRSA-N 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/51—Nanocapsules; Nanoparticles
- A61K9/5107—Excipients; Inactive ingredients
- A61K9/5123—Organic compounds, e.g. fats, sugars
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1658—Proteins, e.g. albumin, gelatin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/51—Nanocapsules; Nanoparticles
- A61K9/5107—Excipients; Inactive ingredients
- A61K9/513—Organic macromolecular compounds; Dendrimers
- A61K9/5169—Proteins, e.g. albumin, gelatin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches

Landscapes

Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Immunology (AREA)
Optics & Photonics (AREA)
Biomedical Technology (AREA)
Nanotechnology (AREA)
Physics & Mathematics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
Gastroenterology & Hepatology (AREA)
Transplantation (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicinal Preparation (AREA)

NO20005769A 1998-05-15 2000-11-14 cyclosporin derivatives NO20005769D0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19821951A DE19821951A1 (en)	1998-05-15	1998-05-15	Orally administered solid or liquid cyclosporin compositions
PCT/EP1999/003002 WO1999059541A2 (en)	1998-05-15	1999-05-04	Cyclosporin preparations

Publications (2)

Publication Number	Publication Date
NO20005769L true NO20005769L (en)	2000-11-14
NO20005769D0 NO20005769D0 (en)	2000-11-14

Family

ID=7867961

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20005769A NO20005769D0 (en)	1998-05-15	2000-11-14	cyclosporin derivatives

Country Status (8)

Country	Link
EP (1)	EP1077676A2 (en)
JP (1)	JP2002515415A (en)
CN (1)	CN1301171A (en)
AU (1)	AU3930399A (en)
CA (1)	CA2332270A1 (en)
DE (1)	DE19821951A1 (en)
NO (1)	NO20005769D0 (en)
WO (1)	WO1999059541A2 (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9920558D0 (en) *	1999-08-31	1999-11-03	Bradford Particle Design Ltd	Methods for particle formation and their products
GB2381453A (en) *	1999-08-31	2003-05-07	Bradford Particle Design Ltd	Active/polymer coformulations
US20020034525A1 (en) *	2000-06-30	2002-03-21	Kao Corporation	Skin cosmetic composition
EP2061440A2 (en) *	2007-04-04	2009-05-27	Sigmoid Pharma Limited	A pharmaceutical composition of tacrolimus
JP6627380B2 (en) *	2015-09-30	2020-01-08	ユーハ味覚糖株式会社	Nanoparticle dispersion liquid with improved permeability of ascorbic acid or ascorbic acid derivative
CN106173799B (en) *	2016-07-08	2019-08-16	武汉轻工大学	Natamycin microemulsion and preparation method thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MX9201782A (en) *	1991-04-19	1992-10-01	Sandoz Ag	PARTICLES OF BIOLOGICALLY ACTIVE SUBSTANCES, SUBSTANTIALLY INSOLUBLE IN WATER, PROCESS FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITION THAT CONTAINS THEM.
ES2108258T3 (en) *	1992-01-17	1997-12-16	Alfatec Pharma Gmbh	GRANULES CONTAINING PEPTIDIC DRUG SUBSTANCES AND THEIR PREPARATION AS WELL AS THEIR USE.
ES2177652T3 (en) *	1994-11-03	2002-12-16	Novartis Ag	NEW FORMS OF PREPARATION OF CYCLOSPORINE FOR ORAL APPLICATION WITH SIMPLE COMPOSITION AND HIGH BIODISPONIBILITY, AND PROCEDURE FOR OBTAINING IT.
KR100239799B1 (en) *	1995-01-21	2000-02-01	손경식	Cyclosporin a solid micelle dispersion for oral administration, the preparation method thereof and its solid dosage form
IE75744B1 (en) *	1995-04-03	1997-09-24	Elan Corp Plc	Controlled release biodegradable micro- and nanospheres containing cyclosporin
US5827822A (en) *	1996-03-25	1998-10-27	Sangstat Medical Corporation	Cyclosporin a formulations as nanoparticles
DE19819273A1 (en) *	1998-04-30	1999-11-11	Pharmatec International S Giul	Pharmaceutical ciclosporin formulation with improved biopharmaceutical properties, increased physical quality and stability as well as processes for its manufacture

1998
- 1998-05-15 DE DE19821951A patent/DE19821951A1/en not_active Withdrawn
1999
- 1999-05-04 AU AU39303/99A patent/AU3930399A/en not_active Abandoned
- 1999-05-04 CA CA002332270A patent/CA2332270A1/en not_active Abandoned
- 1999-05-04 EP EP99922158A patent/EP1077676A2/en not_active Withdrawn
- 1999-05-04 WO PCT/EP1999/003002 patent/WO1999059541A2/en not_active Ceased
- 1999-05-04 CN CN99806202A patent/CN1301171A/en active Pending
- 1999-05-04 JP JP2000549206A patent/JP2002515415A/en not_active Withdrawn
2000
- 2000-11-14 NO NO20005769A patent/NO20005769D0/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO1999059541A3 (en)	2000-01-20
EP1077676A2 (en)	2001-02-28
JP2002515415A (en)	2002-05-28
NO20005769D0 (en)	2000-11-14
CA2332270A1 (en)	1999-11-25
AU3930399A (en)	1999-12-06
WO1999059541A2 (en)	1999-11-25
CN1301171A (en)	2001-06-27
DE19821951A1 (en)	1999-11-18

Legal Events

Date	Code	Title	Description
2004-01-19	FC2A	Withdrawal, rejection or dismissal of laid open patent application

Publication	Publication Date	Title
NO20010193L (en)	2001-01-12	Tiobenzimidazol derivatives
DK0930302T3 (en)	2003-07-21	Benzosulfone derivatives
ATE341990T1 (en)	2006-11-15	SIGMIDOSCOPE
DE59902874D1 (en)	2002-10-31	BUCHSENKONTAKT
DE59901560D1 (en)	2002-07-04	RETROGRADER TIBIANAGEL
NO20010514D0 (en)	2001-01-30	Aminometylkarboksylsyre derivatives
DE69934788D1 (en)	2007-02-22	BIOZIDE BENZYLBIPHENYL DERIVATIVE
ATE259810T1 (en)	2004-03-15	PHENYL-XANTHINE DERIVATIVES
PT928790E (en)	2003-07-31	TIAZOLO DERIVATIVES
DE69902762D1 (en)	2002-10-10	RISER-SPAN ARRANGEMENT
ID27735A (en)	2001-04-26	ARILALKANOILPIRIDAZIN-ARILALKANOILPIRIDAZIN
ATE262513T1 (en)	2004-04-15	BENZOYLPYRIDAZINE
DK1115716T3 (en)	2003-02-24	2-phenylpyran-4-one derivatives
PT1056716E (en)	2003-04-30	CYCLOHEXANODIOL DERIVATIVES
ATE233253T1 (en)	2003-03-15	CHROMEDER DERIVATIVES
DK1134219T3 (en)	2005-10-17	Cucloalkyl-substituted aminomethylpyrrolidine derivatives
DE59901046D1 (en)	2002-05-02	Methylcyclotetradec-5-en-1-one
DK1060183T3 (en)	2003-08-11	5-deoxycytidine derivatives
DE59808995D1 (en)	2003-08-14	endomicroscope
DE59807217D1 (en)	2003-03-20	NADELLAGER
PT1123283E (en)	2004-09-30	TIAZOLE DERIVATIVES
NO20005769D0 (en)	2000-11-14	cyclosporin derivatives
DE59900612D1 (en)	2002-02-21	Dispersionsazofarbstoffmischungen
DE59902088D1 (en)	2002-08-29	Achrathermer Reimager
PT928793E (en)	2002-10-31	TIAZOL DERIVATIVES