NO20012099L - Fremgangsmåte for fremstilling av 4-arylpiperidin-3- karbinoler og beslektede forbindelser - Google Patents

Fremgangsmåte for fremstilling av 4-arylpiperidin-3- karbinoler og beslektede forbindelser

Info

Publication number
NO20012099L
NO20012099L NO20012099A NO20012099A NO20012099L NO 20012099 L NO20012099 L NO 20012099L NO 20012099 A NO20012099 A NO 20012099A NO 20012099 A NO20012099 A NO 20012099A NO 20012099 L NO20012099 L NO 20012099L
Authority
NO
Norway
Prior art keywords
arylpiperidine
carbinols
preparation
related compounds
compounds
Prior art date
Application number
NO20012099A
Other languages
English (en)
Norwegian (no)
Other versions
NO20012099D0 (no
Inventor
Theodorus Hendricus Ant Peters
Franciscus Bernardus Benneker
Hans Jan Hoorn
Frantisek Picha
Original Assignee
Synthon Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthon Bv filed Critical Synthon Bv
Publication of NO20012099D0 publication Critical patent/NO20012099D0/no
Publication of NO20012099L publication Critical patent/NO20012099L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74Oxygen atoms
    • C07D211/76Oxygen atoms attached in position 2 or 6
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20012099A 1998-11-02 2001-04-27 Fremgangsmåte for fremstilling av 4-arylpiperidin-3- karbinoler og beslektede forbindelser NO20012099L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10667398P 1998-11-02 1998-11-02
PCT/IB1999/001762 WO2000026187A1 (fr) 1998-11-02 1999-11-01 Procede de production de 4-arylpiperidine-3-carbinols et composes correspondants

Publications (2)

Publication Number Publication Date
NO20012099D0 NO20012099D0 (no) 2001-04-27
NO20012099L true NO20012099L (no) 2001-07-02

Family

ID=22312658

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20012099A NO20012099L (no) 1998-11-02 2001-04-27 Fremgangsmåte for fremstilling av 4-arylpiperidin-3- karbinoler og beslektede forbindelser

Country Status (5)

Country Link
EP (1) EP1124802A1 (fr)
AU (1) AU6360999A (fr)
CZ (1) CZ20011465A3 (fr)
NO (1) NO20012099L (fr)
WO (1) WO2000026187A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0986389B1 (fr) 1997-05-29 2004-10-13 Smithkline Beecham Corporation Nouveau procede
US20010053862A1 (en) * 1998-12-22 2001-12-20 Bruce Ronsen Process for preparing arylpiperidine carbinol intermediates and derivatives
WO2000037443A1 (fr) * 1998-12-22 2000-06-29 Pentech Pharmaceuticals, Inc. Procede de preparation d'intermediaires et de derives de arylpiperidine carbinol
CZ20023694A3 (cs) * 2000-05-12 2003-05-14 Synthon B. V. Tosylátové soli 4-(p-fluorfenyl)-piperidin-3-methanolů
EP1347960B1 (fr) * 2001-01-04 2004-11-17 Ferrer Internacional, S.A. Procede de preparation de (+)-trans-4-p-fluorophenyl-3-hydroxymethyl-1-methylpiperidine
NZ532432A (en) 2001-10-22 2005-02-25 Synthon Bv N-formyl paroxetine compounds and their use in a synthetic route for obtaining paroxetine
WO2007089193A1 (fr) * 2006-02-02 2007-08-09 Astrazeneca Ab Procédé de synthèse du 2-hydroxy-3-[5-(morpholin-4-ylméthyl)pyridin-2-yl]1h-indole-5-carbonitrile sous forme de base libre ou de ses sels

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI792076A7 (fi) * 1978-07-05 1981-01-01 Ciba Geigy Ag Menetelmä uusien fenyylipiperidiinijohdannaisten valmistamiseksi.
EP0223334B1 (fr) * 1985-08-10 1991-07-10 Beecham Group Plc Procédé de préparation d'aryl-pipéridine-carbinols
US5258517A (en) * 1992-08-06 1993-11-02 Sepracor, Inc. Method of preparing optically pure precursors of paroxetine
GB9526645D0 (en) * 1995-12-28 1996-02-28 Chiroscience Ltd Stereoselective synthesis
JP3446468B2 (ja) * 1996-04-15 2003-09-16 旭硝子株式会社 ピペリジンカルビノール類の製造方法
EP0986389B1 (fr) * 1997-05-29 2004-10-13 Smithkline Beecham Corporation Nouveau procede

Also Published As

Publication number Publication date
CZ20011465A3 (cs) 2001-08-15
WO2000026187A1 (fr) 2000-05-11
NO20012099D0 (no) 2001-04-27
AU6360999A (en) 2000-05-22
EP1124802A1 (fr) 2001-08-22

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