NO20014672L - Fremgangsmåte ved fremstilling av trisykliske aminoalkoholderivater - Google Patents

Fremgangsmåte ved fremstilling av trisykliske aminoalkoholderivater

Info

Publication number
NO20014672L
NO20014672L NO20014672A NO20014672A NO20014672L NO 20014672 L NO20014672 L NO 20014672L NO 20014672 A NO20014672 A NO 20014672A NO 20014672 A NO20014672 A NO 20014672A NO 20014672 L NO20014672 L NO 20014672L
Authority
NO
Norway
Prior art keywords
group
hydrogen atom
preparation
amino alcohol
alcohol derivatives
Prior art date
Application number
NO20014672A
Other languages
English (en)
Other versions
NO20014672D0 (no
Inventor
Koki Matsubara
Hitoshi Kida
Original Assignee
Asahi Chemical Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asahi Chemical Ind filed Critical Asahi Chemical Ind
Publication of NO20014672D0 publication Critical patent/NO20014672D0/no
Publication of NO20014672L publication Critical patent/NO20014672L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/12—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
    • C07C311/13—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings the carbon skeleton containing six-membered aromatic rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Foreliggende oppfinnelse er rettet på fremgangsmåter ved fremstilling av en forbindelse som er nyttig for behandling og forhindring av diabetes, obesitas, hyper- lipidemi og lignende, hvilken forbindelse er representert ved formel (1): OH H (1) NHSO2R1 hvori R1 representerer en lavere alkylgruppe eller en benzylgruppe; *l representerer et asymmetrisk karbon- atom; R2 representerer et hydrogenatom, et halogenatorr eller en hydroksylgruppe; og A representerer en av de følgende grupper: hvori X representerer NH, O eller S; R6 representerer et hydrogenatom, en hydroksylgruppe, en aminogruppe eller en acetylaminogruppe; og *2 representerer et asymmetrisk karbonatom når R6 ikke er et hydrogenatom, og på mellomprodukter som er nyttige for nevnte proses- ser. Fremgangsmåtene ifølge foreliggende oppfinnelse er lettvinte, praktiske fremgangsmåter med lave omkost- ninger, og de har få prosesstrinn med god industriell virkningsgrad.
NO20014672A 1999-03-26 2001-09-26 Fremgangsmåte ved fremstilling av trisykliske aminoalkoholderivater NO20014672L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8319799 1999-03-26
PCT/JP2000/001696 WO2000058287A1 (en) 1999-03-26 2000-03-21 Novel method for manufacturing tricyclic amino alcohol derivatives

Publications (2)

Publication Number Publication Date
NO20014672D0 NO20014672D0 (no) 2001-09-26
NO20014672L true NO20014672L (no) 2001-11-01

Family

ID=13795612

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20014672A NO20014672L (no) 1999-03-26 2001-09-26 Fremgangsmåte ved fremstilling av trisykliske aminoalkoholderivater

Country Status (11)

Country Link
US (1) US6495701B1 (no)
EP (1) EP1174425A1 (no)
KR (1) KR20020005630A (no)
CN (1) CN1349501A (no)
AU (1) AU3195800A (no)
BR (1) BR0009315A (no)
CA (1) CA2368448A1 (no)
MX (1) MXPA01009633A (no)
NO (1) NO20014672L (no)
TW (1) TW519537B (no)
WO (1) WO2000058287A1 (no)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA02002283A (es) * 1999-09-03 2002-07-30 Asahi Chemical Ind Proceso para preparar derivados triciclicos de amino alcoholes.
BR0014469A (pt) * 1999-10-04 2002-06-11 Asahi Chemical Ind Processo para melhorar a solubilidade de um derivado de amino álcool tricìclico, composição farmacêutica, processo para preparar a mesma, e, derivado de amino álcool tricìclico
AU2001252575A1 (en) * 2000-04-28 2001-11-12 Asahi Kasei Kabushiki Kaisha Novel tricyclic compounds
AU2001252573A1 (en) * 2000-04-28 2001-11-12 Asahi Kasei Kabushiki Kaisha Novel substituted tricyclic compounds
AU5257401A (en) 2000-04-28 2001-11-12 Asahi Chemical Ind Novel bicyclic compounds
JPWO2002074306A1 (ja) * 2001-03-19 2004-07-08 旭化成ファーマ株式会社 脂肪肝治療薬
DE60239170D1 (de) * 2001-10-25 2011-03-24 Asahi Kasei Pharma Corp Bicyclische Verbindungen
US7847111B2 (en) * 2006-06-19 2010-12-07 Canada Inc. Semi-synthetic route for the preparation of paclitaxel, docetaxel, and 10-deacetylbaccatin III from 9-dihydro-13-acetylbaccatin III
KR100821567B1 (ko) * 2006-11-01 2008-04-15 한국화학연구원 광학 활성 2-설포닐옥시-1-페닐에탄올 유도체의 제조방법
KR20110050733A (ko) * 2008-10-09 2011-05-16 아사히 가세이 파마 가부시키가이샤 인다졸 유도체
US8008506B2 (en) 2008-10-09 2011-08-30 Asahi Kasei Pharma Corporation Indazole compounds
US20100222404A1 (en) * 2008-11-04 2010-09-02 Asahi Kasei Pharma Corporation Indazole derivative dihydrochloride

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04187685A (ja) 1990-11-21 1992-07-06 Eisai Co Ltd 光学活性ナフチルエタノール誘導体の製造方法
CA2164685C (en) 1994-12-07 2005-03-08 Takeshi Ohkuma Method for producing an alcohol
EP1300381B1 (en) 1995-12-06 2006-03-08 Japan Science and Technology Agency Process for preparing optically active alcohols
CA2242351C (en) 1996-01-10 2003-03-11 Asahi Kasei Kogyo Kabushiki Kaisha Novel tricyclic compounds and drug compositions containing the same
US6172099B1 (en) * 1997-07-03 2001-01-09 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds having saturated rings and medicinal compositions containing the same
DE19846183A1 (de) 1998-10-07 2000-04-27 Bosch Gmbh Robert Zweigang-Getriebe, insbesondere Vorsatzgetriebe für Nebenaggregate in Kraftfahrzeugen
KR20020005648A (ko) 1999-04-01 2002-01-17 야마모토 카즈모토 삼환성 아미노알콜 유도체의 아지드를 경유하는 제조법

Also Published As

Publication number Publication date
KR20020005630A (ko) 2002-01-17
TW519537B (en) 2003-02-01
MXPA01009633A (es) 2003-07-21
AU3195800A (en) 2000-10-16
WO2000058287A1 (en) 2000-10-05
US6495701B1 (en) 2002-12-17
CN1349501A (zh) 2002-05-15
CA2368448A1 (en) 2000-10-05
NO20014672D0 (no) 2001-09-26
BR0009315A (pt) 2001-12-18
EP1174425A1 (en) 2002-01-23

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