NO20031319D0 - Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser - Google Patents
Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelserInfo
- Publication number
- NO20031319D0 NO20031319D0 NO20031319A NO20031319A NO20031319D0 NO 20031319 D0 NO20031319 D0 NO 20031319D0 NO 20031319 A NO20031319 A NO 20031319A NO 20031319 A NO20031319 A NO 20031319A NO 20031319 D0 NO20031319 D0 NO 20031319D0
- Authority
- NO
- Norway
- Prior art keywords
- alkyl
- sulfonyl
- heteroaryl
- aryl
- hydroxy
- Prior art date
Links
- 125000003118 aryl group Chemical group 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C253/00—Preparation of carboxylic acid nitriles
- C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23412100P | 2000-09-21 | 2000-09-21 | |
| PCT/US2001/042171 WO2002024638A1 (en) | 2000-09-21 | 2001-09-17 | Process for the preparation of n-(substituted phenyl)-3-alkyl-, aryl- and heteroarylsulfonyl-2-hydroxy-2-alkyl- and haloalkylpropanamide compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20031319D0 true NO20031319D0 (no) | 2003-03-21 |
Family
ID=22880013
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20031319A NO20031319D0 (no) | 2000-09-21 | 2003-03-21 | Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6562994B2 (no) |
| EP (1) | EP1322603A1 (no) |
| JP (1) | JP2004509164A (no) |
| KR (1) | KR20030048408A (no) |
| CN (1) | CN1501912A (no) |
| AU (1) | AU2001295044A1 (no) |
| BR (1) | BR0114277A (no) |
| CA (1) | CA2423158A1 (no) |
| CZ (1) | CZ2003836A3 (no) |
| HU (1) | HUP0302930A3 (no) |
| IL (1) | IL155041A0 (no) |
| MX (1) | MXPA03002495A (no) |
| NO (1) | NO20031319D0 (no) |
| PL (1) | PL361705A1 (no) |
| WO (1) | WO2002024638A1 (no) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7102026B2 (en) | 2001-06-13 | 2006-09-05 | Teva Gyógyszergyár Zártkörüen Müködö Részvénytársaság | Process for preparing and isolating rac-bicalutamide and its intermediates |
| JP4255381B2 (ja) * | 2001-12-13 | 2009-04-15 | 住友化学株式会社 | ビカルタミドの結晶およびその製造方法 |
| AU2003209667A1 (en) * | 2003-02-21 | 2004-09-09 | Hetero Drugs Limited | Bicalutamide polymorphs |
| WO2005009946A1 (en) * | 2003-06-25 | 2005-02-03 | TEVA Gyógyszergyár Részvénytársaság | Process for purifying and isolating rac-bicalutamide |
| JP2005060302A (ja) * | 2003-08-12 | 2005-03-10 | Sumitomo Chemical Co Ltd | N−メタクリロイル−4−シアノ−3−トリフルオロメチルアニリンの製造方法および安定化方法 |
| JP4322621B2 (ja) | 2003-10-16 | 2009-09-02 | 住友化学株式会社 | 4’−シアノ−3−[(4−フルオロフェニル)スルホニル]−2−ヒドロキシ−2−メチル−3’−トリフルオロメチルプロピオンアニリドの製造方法 |
| WO2006103689A1 (en) * | 2005-03-29 | 2006-10-05 | Usv Limited | Process for preparation of bicalutamide |
| CA2513356A1 (en) * | 2005-07-26 | 2007-01-26 | Apotex Pharmachem Inc. | Process for production of bicalutamide |
| EP1777216A1 (en) * | 2005-09-26 | 2007-04-25 | SOLMAG S.p.A. | A process for the preparation and purification of bicalutamide |
| AU2006329551A1 (en) | 2005-12-27 | 2007-07-05 | Dabur Pharma Limited | An improved process for preparation of Bicalutamide |
| KR20170001736A (ko) * | 2007-09-11 | 2017-01-04 | 지티엑스, 인코포레이티드 | 고형의 선택적인 안드로겐 수용체 모듈레이터 |
| US7968603B2 (en) | 2007-09-11 | 2011-06-28 | University Of Tennessee Research Foundation | Solid forms of selective androgen receptor modulators |
| WO2009087666A2 (en) * | 2008-01-04 | 2009-07-16 | Kekule Pharma | An improved process for production of bicalutamide useful in the treatment of prostate cancer |
| JP2013544768A (ja) | 2010-09-29 | 2013-12-19 | シルパ メディケア リミテッド | ビカルタミドの調製方法 |
| SG11202011135WA (en) | 2018-05-14 | 2020-12-30 | Nuvation Bio Inc | Anti-cancer nuclear hormone receptor-targeting compounds |
| CN109336798B (zh) * | 2018-11-19 | 2021-11-16 | 常州新星联生物科技有限公司 | 一种比卡鲁胺硫醚中间体的制备方法 |
| CN109320442B (zh) * | 2018-11-19 | 2021-01-15 | 启东华拓药业有限公司 | 一种比卡鲁胺的合成方法 |
| US11826430B2 (en) * | 2019-05-14 | 2023-11-28 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB543631A (no) * | ||||
| GB2092136B (en) | 1981-01-17 | 1985-06-05 | Mitsui Toatsu Chemicals | Production of n-substituted amide compounds |
| ATE28864T1 (de) | 1982-07-23 | 1987-08-15 | Ici Plc | Amide-derivate. |
-
2001
- 2001-09-17 HU HU0302930A patent/HUP0302930A3/hu unknown
- 2001-09-17 CA CA002423158A patent/CA2423158A1/en not_active Abandoned
- 2001-09-17 BR BR0114277-1A patent/BR0114277A/pt not_active IP Right Cessation
- 2001-09-17 MX MXPA03002495A patent/MXPA03002495A/es active IP Right Grant
- 2001-09-17 AU AU2001295044A patent/AU2001295044A1/en not_active Abandoned
- 2001-09-17 IL IL15504101A patent/IL155041A0/xx unknown
- 2001-09-17 CN CNA018189334A patent/CN1501912A/zh active Pending
- 2001-09-17 KR KR10-2003-7004173A patent/KR20030048408A/ko not_active Ceased
- 2001-09-17 EP EP01975752A patent/EP1322603A1/en not_active Withdrawn
- 2001-09-17 US US09/953,759 patent/US6562994B2/en not_active Expired - Fee Related
- 2001-09-17 CZ CZ2003836A patent/CZ2003836A3/cs unknown
- 2001-09-17 PL PL36170501A patent/PL361705A1/xx not_active Application Discontinuation
- 2001-09-17 WO PCT/US2001/042171 patent/WO2002024638A1/en not_active Ceased
- 2001-09-17 JP JP2002529051A patent/JP2004509164A/ja active Pending
-
2003
- 2003-03-21 NO NO20031319A patent/NO20031319D0/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HUP0302930A2 (hu) | 2003-12-29 |
| MXPA03002495A (es) | 2004-05-05 |
| WO2002024638A1 (en) | 2002-03-28 |
| IL155041A0 (en) | 2003-10-31 |
| AU2001295044A1 (en) | 2002-04-02 |
| CA2423158A1 (en) | 2002-03-28 |
| BR0114277A (pt) | 2004-12-21 |
| CN1501912A (zh) | 2004-06-02 |
| KR20030048408A (ko) | 2003-06-19 |
| CZ2003836A3 (cs) | 2003-08-13 |
| HUP0302930A3 (en) | 2006-02-28 |
| JP2004509164A (ja) | 2004-03-25 |
| US20020086902A1 (en) | 2002-07-04 |
| EP1322603A1 (en) | 2003-07-02 |
| PL361705A1 (en) | 2004-10-04 |
| US6562994B2 (en) | 2003-05-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20030012L (no) | Fremgangsmåte for fremstilling av substituerte oktanoylamider | |
| NO20042680L (no) | Fremgangsmater for fremstilling av O-demetylvenflaxine | |
| NO20021474L (no) | Forbindelser for behandling av ischemi | |
| ATE275145T1 (de) | Chinazolinderivate zur behandlung von tumoren | |
| DK1232152T3 (da) | Forbedret fremgangsmåde til fremstilling af nitrogensubstituerede aminotetraliner | |
| DE60217126D1 (de) | Herstellung von aminopyrimidinverbindungen | |
| ATE410430T1 (de) | 2,3-dihydro-6-nitroimidazoä2,1- büoxazolverbindungen zur behandlung von tuberkulose | |
| FI20011622A0 (fi) | Menetelmä sitalopraamin valmistamiseksi | |
| NO20031229L (no) | Fremgangsmåte for fremstilling av börstevarer | |
| DE60132600D1 (de) | Medikamente zur chemotherapeutischen behandlung von erkrankungen | |
| NO20040027L (no) | Fremgangsmate for fremstillingen av escitalopram | |
| NO20040253L (no) | Fremgangsmater for behandling av leverfibroser | |
| NO20040278L (no) | Fremgangsmate for fremstilling av perindopril | |
| ATE355067T1 (de) | 15-keto-prostaglandine zur behandlung arzneimittelinduzierter obstipation | |
| IL155041A0 (en) | Process for the preparation of n-(substituted phenyl)-3-alkyl-, aryl-and heteroarylsulfonyl-2-hydroxy-2-alkyl-and haloalkylpropanamide compounds | |
| NO20033433D0 (no) | Fremgangsmåte for fremstilling av 2-(2-pyridylmetyl)sulfinyl- 1H-benzimidasol | |
| NO20044814L (no) | Fremgangsmate for fremstilling av combretastaniner | |
| ATE273276T1 (de) | Cyclobutendion-derivate zur behandlung von artherosclerose | |
| NO20031413D0 (no) | Ny fremgangsmåte for fremstilling av oksabispidiner | |
| NO20030515D0 (no) | Fremgangsmåte for fremstilling av dinapsolin | |
| NO20035586L (no) | Fremgangsmate for fremstilling av cykloheksanol-derivater | |
| NO20035136D0 (no) | Fremgangsmåte til fremstilling av imipenem | |
| NO20000965L (no) | FremgangsmÕte for fremstilling av veksthormon-utskillende forbindelser | |
| DK1373232T3 (da) | Fremgangsmåde til fremstilling af N-substituerede 2,6-dialkylmorpholiner | |
| NO20043105L (no) | Fremgangsmate for fremstilling av 2-(substituert fenyl)-2-hydroksy-etyl-karbamater |