NO20031319D0 - Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser - Google Patents

Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser

Info

Publication number
NO20031319D0
NO20031319D0 NO20031319A NO20031319A NO20031319D0 NO 20031319 D0 NO20031319 D0 NO 20031319D0 NO 20031319 A NO20031319 A NO 20031319A NO 20031319 A NO20031319 A NO 20031319A NO 20031319 D0 NO20031319 D0 NO 20031319D0
Authority
NO
Norway
Prior art keywords
alkyl
sulfonyl
heteroaryl
aryl
hydroxy
Prior art date
Application number
NO20031319A
Other languages
English (en)
Inventor
Bang-Chi Chen
Joseph E Sundeen
Rulin Zhao
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20031319D0 publication Critical patent/NO20031319D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Epoxy Compounds (AREA)
NO20031319A 2000-09-21 2003-03-21 Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser NO20031319D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23412100P 2000-09-21 2000-09-21
PCT/US2001/042171 WO2002024638A1 (en) 2000-09-21 2001-09-17 Process for the preparation of n-(substituted phenyl)-3-alkyl-, aryl- and heteroarylsulfonyl-2-hydroxy-2-alkyl- and haloalkylpropanamide compounds

Publications (1)

Publication Number Publication Date
NO20031319D0 true NO20031319D0 (no) 2003-03-21

Family

ID=22880013

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20031319A NO20031319D0 (no) 2000-09-21 2003-03-21 Fremgangsmåte for fremstilling av N-(substituert fenyl)-3- alkyl-, aryl- ogheteroaryl-sulfonyl-2-hydroksy-2-alkyl- oghalogenalkylpropanamidforbindelser

Country Status (15)

Country Link
US (1) US6562994B2 (no)
EP (1) EP1322603A1 (no)
JP (1) JP2004509164A (no)
KR (1) KR20030048408A (no)
CN (1) CN1501912A (no)
AU (1) AU2001295044A1 (no)
BR (1) BR0114277A (no)
CA (1) CA2423158A1 (no)
CZ (1) CZ2003836A3 (no)
HU (1) HUP0302930A3 (no)
IL (1) IL155041A0 (no)
MX (1) MXPA03002495A (no)
NO (1) NO20031319D0 (no)
PL (1) PL361705A1 (no)
WO (1) WO2002024638A1 (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7102026B2 (en) 2001-06-13 2006-09-05 Teva Gyógyszergyár Zártkörüen Müködö Részvénytársaság Process for preparing and isolating rac-bicalutamide and its intermediates
JP4255381B2 (ja) * 2001-12-13 2009-04-15 住友化学株式会社 ビカルタミドの結晶およびその製造方法
AU2003209667A1 (en) * 2003-02-21 2004-09-09 Hetero Drugs Limited Bicalutamide polymorphs
WO2005009946A1 (en) * 2003-06-25 2005-02-03 TEVA Gyógyszergyár Részvénytársaság Process for purifying and isolating rac-bicalutamide
JP2005060302A (ja) * 2003-08-12 2005-03-10 Sumitomo Chemical Co Ltd N−メタクリロイル−4−シアノ−3−トリフルオロメチルアニリンの製造方法および安定化方法
JP4322621B2 (ja) 2003-10-16 2009-09-02 住友化学株式会社 4’−シアノ−3−[(4−フルオロフェニル)スルホニル]−2−ヒドロキシ−2−メチル−3’−トリフルオロメチルプロピオンアニリドの製造方法
WO2006103689A1 (en) * 2005-03-29 2006-10-05 Usv Limited Process for preparation of bicalutamide
CA2513356A1 (en) * 2005-07-26 2007-01-26 Apotex Pharmachem Inc. Process for production of bicalutamide
EP1777216A1 (en) * 2005-09-26 2007-04-25 SOLMAG S.p.A. A process for the preparation and purification of bicalutamide
AU2006329551A1 (en) 2005-12-27 2007-07-05 Dabur Pharma Limited An improved process for preparation of Bicalutamide
KR20170001736A (ko) * 2007-09-11 2017-01-04 지티엑스, 인코포레이티드 고형의 선택적인 안드로겐 수용체 모듈레이터
US7968603B2 (en) 2007-09-11 2011-06-28 University Of Tennessee Research Foundation Solid forms of selective androgen receptor modulators
WO2009087666A2 (en) * 2008-01-04 2009-07-16 Kekule Pharma An improved process for production of bicalutamide useful in the treatment of prostate cancer
JP2013544768A (ja) 2010-09-29 2013-12-19 シルパ メディケア リミテッド ビカルタミドの調製方法
SG11202011135WA (en) 2018-05-14 2020-12-30 Nuvation Bio Inc Anti-cancer nuclear hormone receptor-targeting compounds
CN109336798B (zh) * 2018-11-19 2021-11-16 常州新星联生物科技有限公司 一种比卡鲁胺硫醚中间体的制备方法
CN109320442B (zh) * 2018-11-19 2021-01-15 启东华拓药业有限公司 一种比卡鲁胺的合成方法
US11826430B2 (en) * 2019-05-14 2023-11-28 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB543631A (no) *
GB2092136B (en) 1981-01-17 1985-06-05 Mitsui Toatsu Chemicals Production of n-substituted amide compounds
ATE28864T1 (de) 1982-07-23 1987-08-15 Ici Plc Amide-derivate.

Also Published As

Publication number Publication date
HUP0302930A2 (hu) 2003-12-29
MXPA03002495A (es) 2004-05-05
WO2002024638A1 (en) 2002-03-28
IL155041A0 (en) 2003-10-31
AU2001295044A1 (en) 2002-04-02
CA2423158A1 (en) 2002-03-28
BR0114277A (pt) 2004-12-21
CN1501912A (zh) 2004-06-02
KR20030048408A (ko) 2003-06-19
CZ2003836A3 (cs) 2003-08-13
HUP0302930A3 (en) 2006-02-28
JP2004509164A (ja) 2004-03-25
US20020086902A1 (en) 2002-07-04
EP1322603A1 (en) 2003-07-02
PL361705A1 (en) 2004-10-04
US6562994B2 (en) 2003-05-13

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