NO20041279L - Metylen-4-azasteroider. - Google Patents

Metylen-4-azasteroider.

Info

Publication number: NO20041279L
Authority: NO; Norway
Prior art keywords: sup; methylene; denote; hydrogen atom; denotes
Prior art date: 2001-08-28

Application number

NONO/SPC/2A

Other languages

English (en)

Other versions

NO326564B1 (no

Inventor

Klaus Schollkopf

Walter Elger

Alexander Hillisch

Peter Droscher

Bernd Menzenbach

Hans-Udo Schweikert

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-08-28

Filing date

2004-03-26

Publication date

2004-03-26

2004-03-26 Application filed by Schering Ag filed Critical Schering Ag

2004-03-26 Publication of NO20041279L publication Critical patent/NO20041279L/no

2009-01-12 Publication of NO326564B1 publication Critical patent/NO326564B1/no

Links

125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 3
208000002874 Acne Vulgaris Diseases 0.000 abstract 1
201000004384 Alopecia Diseases 0.000 abstract 1
206010020112 Hirsutism Diseases 0.000 abstract 1
206010000496 acne Diseases 0.000 abstract 1
231100000360 alopecia Toxicity 0.000 abstract 1
239000003098 androgen Substances 0.000 abstract 1
125000001246 bromo group Chemical group Br* 0.000 abstract 1
125000001309 chloro group Chemical group Cl* 0.000 abstract 1
201000010099 disease Diseases 0.000 abstract 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
125000001153 fluoro group Chemical group F* 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
208000017497 prostate disease Diseases 0.000 abstract 1
230000002194 synthesizing effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
- C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/06—Antiabortive agents; Labour repressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO20041279A 2001-08-28 2004-03-26 Metylen-4-azasteroider, fremgangsmater for fremstilling av forbindelsene, farmasoytiske preparater som omfatter dem, og anvendelse av forbindelsene til fremstilling av farmasoytiske produkter NO326564B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10141984A DE10141984A1 (de)	2001-08-28	2001-08-28	Neue 17-Methylen-4-azasteroide
PCT/EP2002/009587 WO2003020744A1 (de)	2001-08-28	2002-08-28	Methylen-4-azasteroide

Publications (2)

Publication Number	Publication Date
NO20041279L true NO20041279L (no)	2004-03-26
NO326564B1 NO326564B1 (no)	2009-01-12

Family

ID=7696782

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20041279A NO326564B1 (no)	2001-08-28	2004-03-26	Metylen-4-azasteroider, fremgangsmater for fremstilling av forbindelsene, farmasoytiske preparater som omfatter dem, og anvendelse av forbindelsene til fremstilling av farmasoytiske produkter

Country Status (21)

Country	Link
US (1)	US7186728B2 (no)
EP (1)	EP1409513B1 (no)
JP (1)	JP3927174B2 (no)
KR (1)	KR100550514B1 (no)
CN (1)	CN1322002C (no)
AT (1)	ATE323100T1 (no)
AU (1)	AU2002342625B8 (no)
BR (1)	BR0212104A (no)
CA (1)	CA2458932C (no)
CY (1)	CY1105083T1 (no)
DE (2)	DE10141984A1 (no)
DK (1)	DK1409513T3 (no)
ES (1)	ES2262856T3 (no)
HU (1)	HUP0401597A3 (no)
IL (2)	IL160540A0 (no)
NO (1)	NO326564B1 (no)
PL (1)	PL367460A1 (no)
PT (1)	PT1409513E (no)
RU (1)	RU2293740C2 (no)
WO (1)	WO2003020744A1 (no)
ZA (1)	ZA200402368B (no)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN110643557B (zh) *	2019-04-23	2021-12-31	天津科技大学	一种基因工程菌的构建及其在高效催化5α-雄烯二酮生产中的应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5264427A (en) *	1992-01-29	1993-11-23	Research Corporation Technologies, Inc.	20-substituted pregnene derivatives and their use as androgen synthesis inhibitors
JPH11513711A (ja) *	1995-10-23	1999-11-24	メルクエンドカンパニーインコーポレーテッド	１７−アルキル−７−置換−４−アザステロイド誘導体
US5763361A (en) *	1995-10-23	1998-06-09	Merck & Co., Inc.	17-alkyl-7-substituted-4-aza steroid derivatives as 5-α-reductase inhibitors
US5994334A (en)	1997-02-05	1999-11-30	University Of Maryland	Androgen synthesis inhibitors
AU2001268661A1 (en) *	2000-06-27	2002-01-08	Aventis Pharma S.A.	20-fluoro-17(20)-vinyl steroids as inhibitors of c17-20-lyase and 5-alpha reductase
DE10043846A1 (de) *	2000-09-04	2002-04-04	Jenapharm Gmbh	17-Methylensteroide, Verfahren zu deren Herstellung und diese Verbindung enthaltende pharmazeutische Zusammensetzungen

2001
- 2001-08-28 DE DE10141984A patent/DE10141984A1/de not_active Withdrawn
2002
- 2002-08-28 DE DE50206397T patent/DE50206397D1/de not_active Expired - Lifetime
- 2002-08-28 IL IL16054002A patent/IL160540A0/xx unknown
- 2002-08-28 JP JP2003525014A patent/JP3927174B2/ja not_active Expired - Fee Related
- 2002-08-28 PT PT02779279T patent/PT1409513E/pt unknown
- 2002-08-28 BR BR0212104-2A patent/BR0212104A/pt not_active IP Right Cessation
- 2002-08-28 CN CNB028170814A patent/CN1322002C/zh not_active Expired - Fee Related
- 2002-08-28 CA CA002458932A patent/CA2458932C/en not_active Expired - Fee Related
- 2002-08-28 HU HU0401597A patent/HUP0401597A3/hu unknown
- 2002-08-28 WO PCT/EP2002/009587 patent/WO2003020744A1/de not_active Ceased
- 2002-08-28 AU AU2002342625A patent/AU2002342625B8/en not_active Ceased
- 2002-08-28 KR KR1020047002922A patent/KR100550514B1/ko not_active Expired - Fee Related
- 2002-08-28 ES ES02779279T patent/ES2262856T3/es not_active Expired - Lifetime
- 2002-08-28 DK DK02779279T patent/DK1409513T3/da active
- 2002-08-28 EP EP02779279A patent/EP1409513B1/de not_active Expired - Lifetime
- 2002-08-28 US US10/487,862 patent/US7186728B2/en not_active Expired - Fee Related
- 2002-08-28 PL PL02367460A patent/PL367460A1/xx unknown
- 2002-08-28 RU RU2004109166/04A patent/RU2293740C2/ru not_active IP Right Cessation
- 2002-08-28 AT AT02779279T patent/ATE323100T1/de not_active IP Right Cessation
2004
- 2004-02-24 IL IL160540A patent/IL160540A/en not_active IP Right Cessation
- 2004-03-25 ZA ZA200402368A patent/ZA200402368B/en unknown
- 2004-03-26 NO NO20041279A patent/NO326564B1/no not_active IP Right Cessation
2006
- 2006-07-10 CY CY20061100960T patent/CY1105083T1/el unknown

Also Published As

Publication number	Publication date
WO2003020744A1 (de)	2003-03-13
AU2002342625B8 (en)	2009-01-08
CA2458932C (en)	2008-07-22
JP3927174B2 (ja)	2007-06-06
KR20040032978A (ko)	2004-04-17
ATE323100T1 (de)	2006-04-15
DE50206397D1 (de)	2006-05-24
HUP0401597A2 (hu)	2004-12-28
EP1409513B1 (de)	2006-04-12
CY1105083T1 (el)	2009-11-04
AU2002342625B2 (en)	2008-12-04
CA2458932A1 (en)	2003-03-13
ES2262856T3 (es)	2006-12-01
JP2005504786A (ja)	2005-02-17
HUP0401597A3 (en)	2011-02-28
DE10141984A1 (de)	2003-03-20
HK1071376A1 (en)	2005-07-15
CN1549822A (zh)	2004-11-24
KR100550514B1 (ko)	2006-02-13
EP1409513A1 (de)	2004-04-21
DK1409513T3 (da)	2006-08-14
US7186728B2 (en)	2007-03-06
IL160540A0 (en)	2004-07-25
RU2004109166A (ru)	2005-10-10
NO326564B1 (no)	2009-01-12
RU2293740C2 (ru)	2007-02-20
BR0212104A (pt)	2004-08-24
PL367460A1 (en)	2005-02-21
CN1322002C (zh)	2007-06-20
IL160540A (en)	2009-11-18
US20040248921A1 (en)	2004-12-09
PT1409513E (pt)	2006-08-31
ZA200402368B (en)	2005-05-20

Legal Events

Date	Code	Title	Description
2011-04-04	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
DE60236600D1 (de)	2010-07-15	Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
MXPA03011006A (es)	2004-02-27	Compuestos de cicloalquil urea benzo-fusionados 1,4-disustituidos.
ATE253545T1 (de)	2003-11-15	Biarylessigsäure-derivate und ihre verwendung als cox-2 inhibitoren
MXPA04001323A (es)	2004-05-20	Dihidro-3-halo-1h-pirazol-5-carboxilatos sustituidos, su preparacion y uso.
BRPI0413305A (pt)	2006-10-10	compostos azabicìclicos fundidos que inibem o receptor de subtipo de receptor de vanilóide 1 (vr1)
BR0114045A (pt)	2003-07-01	Poliarilcarboxamidas úteis como agentes redutores de lipìdeos
ATE357434T1 (de)	2007-04-15	Disubstituierte thiazolylcarboxanilide und ihre verwendung als mikrobizide
DK1485359T3 (da)	2008-04-14	Natriumkanalblokkere
MXPA02011370A (es)	2003-06-06	Iminoazinas substituidas.
WO2001017963A3 (en)	2001-11-15	Aminoalkoxy carbazoles and their use as 5-ht ligands
ATE244699T1 (de)	2003-07-15	Substituierte anilinverbindungen
DE602004009200D1 (de)	2007-11-08	Tetrahydrochinazolinderivate als cfr-antagonisten
IL179607A0 (en)	2007-05-15	Indoles useful in the treatment of inflammation
ATE359786T1 (de)	2007-05-15	Camptothecin derivate
DE50208918D1 (de)	2007-01-18	6-aminomorphinanderivate, herstellungsverfahren dafür und deren verwendung
EA200300804A1 (ru)	2003-12-25	Усовершенствованный способ получения карбапенема
TR200302288T2 (tr)	2004-12-21	Terapi için yeni bileşikler ve metotlar.
EA200100040A1 (ru)	2001-06-25	Химический синтез морфолиновых производных
ATE353884T1 (de)	2007-03-15	Multifunktionelle kationische photoinitiatoren, deren herstellung und verwendung
PT1204659E (pt)	2004-04-30	Benzofuranos serotoninergicos
DK1409513T3 (da)	2006-08-14	Methylen-4-azasteroider
EA200500032A1 (ru)	2005-08-25	Производные ацилоксипирролидина и их применение в качестве лигандов v1b или v1b и v1a рецепторов
SE0302035D0 (sv)	2003-07-09	New compound
NO20033049L (no)	2003-08-18	Fremgangsmåte for fremstilling av (+/-) trans-4-p-fluorfenyl- 3-hydroksymetyl-1-metylpiperidin
ATE319708T1 (de)	2006-03-15	Azol- oder triazol-derivate, verfahren zu deren herstellung und ihre verwendung als fungizide