NO20051966L - Nye pyrimidinamidderivater og anvendelse derav - Google Patents

Nye pyrimidinamidderivater og anvendelse derav

Info

Publication number: NO20051966L
Authority: NO; Norway
Prior art keywords: derivatives; pyrimidinamide; disease; new; benzoylaminophenyl
Prior art date: 2002-09-27

Application number

NO20051966A

Other languages

English (en)

Norwegian (no)

Inventor

Pascal Furet

Werner Breitenstein

Paul William Manley

Sandra Jacob

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-09-27

Filing date

2005-04-22

Publication date

2005-04-22

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9944917&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20051966(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2005-04-22 Application filed by Novartis Ag filed Critical Novartis Ag

2005-04-22 Publication of NO20051966L publication Critical patent/NO20051966L/no

Links

FUXJMHXHGDAHPD-UHFFFAOYSA-N pyrimidine-2-carboxamide Chemical class NC(=O)C1=NC=CC=N1 FUXJMHXHGDAHPD-UHFFFAOYSA-N 0.000 title 1
201000010099 disease Diseases 0.000 abstract 3
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 3
238000000034 method Methods 0.000 abstract 2
102000001253 Protein Kinase Human genes 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000000694 effects Effects 0.000 abstract 1
230000005764 inhibitory process Effects 0.000 abstract 1
NGNJTDQLHYCUGI-UHFFFAOYSA-N n-[3-[(4-pyridin-4-ylpyrimidin-2-yl)amino]phenyl]benzamide Chemical class C=1C=CC=CC=1C(=O)NC(C=1)=CC=CC=1NC(N=1)=NC=CC=1C1=CC=NC=C1 NGNJTDQLHYCUGI-UHFFFAOYSA-N 0.000 abstract 1
230000001613 neoplastic effect Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
108060006633 protein kinase Proteins 0.000 abstract 1
238000002560 therapeutic procedure Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Hematology (AREA)
Urology & Nephrology (AREA)
Cardiology (AREA)
Pulmonology (AREA)
Heart & Thoracic Surgery (AREA)
Emergency Medicine (AREA)
Vascular Medicine (AREA)
Endocrinology (AREA)
Obesity (AREA)
Ophthalmology & Optometry (AREA)
Oncology (AREA)
Dermatology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyridine Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Hydrogenated Pyridines (AREA)

NO20051966A 2002-09-27 2005-04-22 Nye pyrimidinamidderivater og anvendelse derav NO20051966L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0222514.2A GB0222514D0 (en)	2002-09-27	2002-09-27	Organic compounds
PCT/EP2003/010724 WO2004029038A1 (en)	2002-09-27	2003-09-26	Novel pyrimidineamide derivatives and the use thereof

Publications (1)

Publication Number	Publication Date
NO20051966L true NO20051966L (no)	2005-04-22

Family

ID=9944917

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20051966A NO20051966L (no)	2002-09-27	2005-04-22	Nye pyrimidinamidderivater og anvendelse derav

Country Status (23)

Country	Link
US (1)	US7655669B2 (es)
EP (1)	EP1546127B1 (es)
JP (2)	JP4463685B2 (es)
KR (2)	KR100876055B1 (es)
CN (1)	CN100404528C (es)
AT (1)	ATE369355T1 (es)
AU (1)	AU2003270277B2 (es)
BR (1)	BR0314797A (es)
CA (1)	CA2499822C (es)
DE (1)	DE60315479T2 (es)
DK (1)	DK1546127T3 (es)
EC (1)	ECSP055701A (es)
ES (1)	ES2288615T3 (es)
GB (1)	GB0222514D0 (es)
MX (1)	MXPA05003253A (es)
NO (1)	NO20051966L (es)
NZ (1)	NZ538930A (es)
PL (1)	PL374443A1 (es)
PT (1)	PT1546127E (es)
RU (1)	RU2378267C2 (es)
SI (1)	SI1546127T1 (es)
WO (1)	WO2004029038A1 (es)
ZA (1)	ZA200502304B (es)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0222514D0 (en) *	2002-09-27	2002-11-06	Novartis Ag	Organic compounds
US7232825B2 (en) *	2003-05-02	2007-06-19	Guoqing P Chen	Phenylaminopyrimidine derivatives and methods of use
GB0325031D0 (en)	2003-10-27	2003-12-03	Novartis Ag	Organic compounds
DE10352979A1 (de) *	2003-11-13	2005-06-09	Merck Patent Gmbh	Pyridopyrimidinone
TW200616974A (en) *	2004-07-01	2006-06-01	Astrazeneca Ab	Chemical compounds
EP1789399A1 (en)	2004-08-31	2007-05-30	AstraZeneca AB	Quinazolinone derivatives and their use as b-raf inhibitors
ES2390227T3 (es)	2004-09-09	2012-11-07	Natco Pharma Limited	Nuevos derivados de fenilaminopirimidina como inhibidores de la BCR-ABL kinasa
US8735415B2 (en)	2004-09-09	2014-05-27	Natco Pharma Limited	Acid addition salts of (3,5-Bis trifluoromethyl)-N-[4-methyl-3-(4-pyridin-3yl-pyrimidin-2ylamino)-phenyl]-benzamide
US7939541B2 (en)	2004-09-09	2011-05-10	Natco Pharma Limited	Intermediates and a process employing the intermediates for the preparation of (3-trifluoromethylsulfonyl)-N-[4-methyl-3-(4-pyridin-3yl-pyrimidin-2ylamino)-phenyl]-benzamide
CN1939910A (zh)	2004-12-31	2007-04-04	孙飘扬	氨基嘧啶类化合物及其盐和其制备方法与药物用途
CN1972917B (zh) *	2004-12-31	2010-08-25	孙飘扬	氨基嘧啶类化合物及其盐和其制备方法与药物用途
CN101203224B (zh) *	2005-01-28	2010-11-03	诺瓦提斯公司	嘧啶基氨基苯甲酰胺在制备治疗对Tie-2激酶活性的调节有响应的疾病的药物中的用途
MY146795A (en) *	2005-06-09	2012-09-28	Novartis Ag	Process for the synthesis of organic compounds
WO2008020203A1 (en) *	2006-08-17	2008-02-21	Astrazeneca Ab	Pyridinylquinaz0linamine derivatives and their use as b-raf inhibitors
EP2068938B1 (en)	2006-09-22	2011-01-19	Novartis AG	Optimization of the treatment of philadelphia-positive leukemia with abl tyrosine kinase inhibitor imatinib
CA2668190A1 (en) *	2006-11-03	2008-05-15	Irm Llc	Compounds and compositions as protein kinase inhibitors
US7550591B2 (en) *	2007-05-02	2009-06-23	Chemagis Ltd.	Imatinib production process
EA019524B1 (ru)	2007-05-04	2014-04-30	Айрм Ллк	СОЕДИНЕНИЯ И КОМПОЗИЦИИ КАК ИНГИБИТОРЫ КИНАЗЫ с-kit И PDGFR
ATE544761T1 (de) *	2007-05-04	2012-02-15	Irm Llc	Pyrimidinderivate und zusammensetzungen als c-kit-und pdgfr-kinasehemmer
EP2152079A4 (en)	2007-06-04	2011-03-09	Avila Therapeutics Inc	HETEROCYCLIC COMPOUNDS AND USES THEREOF
AU2008289037B2 (en)	2007-08-22	2012-03-01	Novartis Ag	5- (4- (haloalkoxy) phenyl) pyrimidine-2-amine compounds and compositions as kinase inhibitors
JP5303557B2 (ja)	2007-08-22	2013-10-02	アイアールエム・リミテッド・ライアビリティ・カンパニー	キナーゼ阻害剤である２−ヘテロアリールアミノ−ピリミジン誘導体
US8067422B2 (en)	2008-03-04	2011-11-29	Natco Pharma Limited	Crystal form of phenylamino pyrimidine derivatives
BR112012028231A2 (pt) *	2010-05-11	2017-08-15	Krisani Biosciences P Ltd	Composto, síntese, composição e utilização em questão
CA2856291C (en)	2011-11-17	2020-08-11	Dana-Farber Cancer Institute, Inc.	Inhibitors of c-jun-n-terminal kinase (jnk)
AU2020232755A1 (en) *	2019-03-05	2021-11-04	Hongyi & Associates LLC.	Compounds for treating neurodegenerative diseases and cancers

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0233461B2 (en)	1986-01-13	2002-05-29	American Cyanamid Company	4,5,6-Substituted-2-pyrimidinamines
US5215989A (en)	1989-12-08	1993-06-01	Merck & Co., Inc.	Nitrogen-containing heterocyclic compounds as class III antiarrhythmic agents
US5521184A (en) *	1992-04-03	1996-05-28	Ciba-Geigy Corporation	Pyrimidine derivatives and processes for the preparation thereof
TW225528B (es)	1992-04-03	1994-06-21	Ciba Geigy Ag
US5516775A (en)	1992-08-31	1996-05-14	Ciba-Geigy Corporation	Further use of pyrimidine derivatives
EP0672035A1 (en)	1993-10-01	1995-09-20	Novartis AG	Pyrimidineamine derivatives and processes for the preparation thereof
US5543520A (en)	1993-10-01	1996-08-06	Ciba-Geigy Corporation	Pyrimidine derivatives
ITMI992711A1 (it)	1999-12-27	2001-06-27	Novartis Ag	Composti organici
US7087608B2 (en)	2000-03-03	2006-08-08	Robert Charles Atkins	Use of PDGF receptor tyrosine kinase inhibitors for the treatment of diabetic nephropathy
GB0022438D0 (en)	2000-09-13	2000-11-01	Novartis Ag	Organic Compounds
GB0025820D0 (en)	2000-10-20	2000-12-06	Novartis Ag	Organic compounds
DE60212836T2 (de)	2001-05-16	2007-01-25	Gpc Biotech Ag	Pyridylpyrimidin-derivate als wirksame verbindungen gegen prionen-krankheiten
GB0222514D0 (en) *	2002-09-27	2002-11-06	Novartis Ag	Organic compounds
EP1700164B1 (en)	2003-12-23	2010-08-04	Koninklijke Philips Electronics N.V.	Irradiation method

2002
- 2002-09-27 GB GBGB0222514.2A patent/GB0222514D0/en not_active Ceased
2003
- 2003-09-26 CN CNB038232138A patent/CN100404528C/zh not_active Expired - Fee Related
- 2003-09-26 KR KR1020057005204A patent/KR100876055B1/ko not_active Expired - Fee Related
- 2003-09-26 WO PCT/EP2003/010724 patent/WO2004029038A1/en not_active Ceased
- 2003-09-26 AT AT03750639T patent/ATE369355T1/de not_active IP Right Cessation
- 2003-09-26 RU RU2005113153/04A patent/RU2378267C2/ru not_active IP Right Cessation
- 2003-09-26 AU AU2003270277A patent/AU2003270277B2/en not_active Ceased
- 2003-09-26 KR KR1020077019251A patent/KR20070098940A/ko not_active Ceased
- 2003-09-26 MX MXPA05003253A patent/MXPA05003253A/es active IP Right Grant
- 2003-09-26 PT PT03750639T patent/PT1546127E/pt unknown
- 2003-09-26 SI SI200331014T patent/SI1546127T1/sl unknown
- 2003-09-26 BR BR0314797-5A patent/BR0314797A/pt not_active IP Right Cessation
- 2003-09-26 EP EP03750639A patent/EP1546127B1/en not_active Expired - Lifetime
- 2003-09-26 US US10/528,913 patent/US7655669B2/en not_active Expired - Fee Related
- 2003-09-26 DE DE60315479T patent/DE60315479T2/de not_active Expired - Lifetime
- 2003-09-26 DK DK03750639T patent/DK1546127T3/da active
- 2003-09-26 JP JP2004539039A patent/JP4463685B2/ja not_active Expired - Fee Related
- 2003-09-26 NZ NZ538930A patent/NZ538930A/en unknown
- 2003-09-26 PL PL03374443A patent/PL374443A1/xx not_active Application Discontinuation
- 2003-09-26 ES ES03750639T patent/ES2288615T3/es not_active Expired - Lifetime
- 2003-09-26 CA CA2499822A patent/CA2499822C/en not_active Expired - Fee Related
2005
- 2005-03-18 ZA ZA200502304A patent/ZA200502304B/en unknown
- 2005-03-23 EC EC2005005701A patent/ECSP055701A/es unknown
- 2005-04-22 NO NO20051966A patent/NO20051966L/no not_active Application Discontinuation
2009
- 2009-10-09 JP JP2009235252A patent/JP5178681B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US20060142577A1 (en)	2006-06-29
DK1546127T3 (da)	2007-12-10
GB0222514D0 (en)	2002-11-06
BR0314797A (pt)	2005-07-26
EP1546127A1 (en)	2005-06-29
KR20070098940A (ko)	2007-10-05
JP5178681B2 (ja)	2013-04-10
NZ538930A (en)	2008-04-30
ECSP055701A (es)	2005-05-30
MXPA05003253A (es)	2005-06-08
JP4463685B2 (ja)	2010-05-19
WO2004029038A1 (en)	2004-04-08
JP2010043113A (ja)	2010-02-25
CA2499822C (en)	2012-04-10
AU2003270277A1 (en)	2004-04-19
US7655669B2 (en)	2010-02-02
CN100404528C (zh)	2008-07-23
CA2499822A1 (en)	2004-04-08
RU2378267C2 (ru)	2010-01-10
KR20050047128A (ko)	2005-05-19
ES2288615T3 (es)	2008-01-16
AU2003270277B2 (en)	2007-08-23
JP2006508064A (ja)	2006-03-09
ZA200502304B (en)	2006-04-26
ATE369355T1 (de)	2007-08-15
KR100876055B1 (ko)	2008-12-26
CN1684951A (zh)	2005-10-19
EP1546127B1 (en)	2007-08-08
PL374443A1 (en)	2005-10-17
RU2005113153A (ru)	2006-11-10
PT1546127E (pt)	2007-11-07
DE60315479T2 (de)	2008-04-30
DE60315479D1 (de)	2007-09-20
HK1080459A1 (en)	2006-04-28
SI1546127T1 (sl)	2008-08-31

Legal Events

Date	Code	Title	Description
2010-04-26	FC2A	Withdrawal, rejection or dismissal of laid open patent application

Publication	Publication Date	Title
DK1546127T3 (da)	2007-12-10	Nye pyrimidinamidderivater og anvendelse deraf
DE602004017194D1 (de)	2008-11-27	Pyridylpyrrol-derivate als wirksame kinase-hemmer
DK1636236T3 (da)	2013-12-09	Pyrazolo-quinazolin-derivater, en fremgangsmåde til fremstilling deraf, og deres anvendelse som kinase-inhibitorer
WO2004005281A8 (en)	2004-05-06	Inhibitors of tyrosine kinases
MXPA06000302A (es)	2006-04-18	Derivados de pirazolil-indol activos como inhibidores de cinasa, procedimientos para su preparacion y composiciones farmaceuticas que los comprenden.
TW200615266A (en)	2006-05-16	Organic compounds
NO20055863L (no)	2001-09-12	W-karboksyarylsubstituerte difenylureaforbindelser som raf-kinaseinhibitorer
NO20062504L (no)	2006-07-21	Sammensetninger og doseringsformer for forbedret absorpsjon
CY1108932T1 (el)	2014-07-02	Ενωσεις 4-(ετεροκυκλυλ)-βενζολοσουλφοξιμινης για την θεραπευτικη αγωγη φλεγμονωδων ασθενειων
NO20040547L (no)	2004-03-03	Amino-ftalazinonderivater aktive som kinaseinhibitorer, fremgangsmate for deres fremstilling og farmasoytiske sammensetninger inneholdende disse.
DE50310516D1 (de)	2008-10-30	Fredericamycin-derivate
BRPI0413438A (pt)	2006-10-17	derivados de pirimidilpirrol ativos como inibidores de cinase
BR0312722A (pt)	2005-05-10	Derivados de pirazol heterobicìclico como inibidores de qinase
SE0101932D0 (sv)	2001-05-31	Pharmaceutical combinations
BR0316458A (pt)	2005-10-11	Composto, composição farmacêutica, método de tratamento ou prevenção de doenças, método para intensificar a cognição em um paciente saudável, e, uso de um composto
SE0002729D0 (sv)	2000-07-20	Novel compound form
DE50312224D1 (de)	2010-01-21	Deuterierte catecholaminderivate sowie diese verbindungen enthaltende arzneimittel
MXPA05014143A (es)	2006-02-24	Derivados de cumarina para el tratamiento de trastornos oftalmicos.
NO20030021D0 (no)	2003-01-03	Heterosykliske forbindelser som er inhibitorer for enzymet DPP-IV
NO20034985L (no)	2003-11-10	Nye 5-tio-SS-D-xylopyranosid-derivater, fremgangsmåte for fremstilling derav, farmasöytiske blandinger inneholdende dem og den terapeutiskeanvendelse derav
DE60327249D1 (de)	2009-05-28	Anthranilsäureamide und ihre pharmazeutische verwendung
DE50304524D1 (de)	2006-09-14	Arzneimittel enthaltend substituierte 2,5-diaminomethyl-1h-pyrrole
ECSP12005525A (es)	2014-01-31	Inhibidores de cinasas de tirosina