NO20052474L - Amort form av esomeprazolsalter - Google Patents
Amort form av esomeprazolsalterInfo
- Publication number
- NO20052474L NO20052474L NO20052474A NO20052474A NO20052474L NO 20052474 L NO20052474 L NO 20052474L NO 20052474 A NO20052474 A NO 20052474A NO 20052474 A NO20052474 A NO 20052474A NO 20052474 L NO20052474 L NO 20052474L
- Authority
- NO
- Norway
- Prior art keywords
- salts
- amortized
- esomeprazole
- esomeprazole salts
- amorphous
- Prior art date
Links
- SUBDBMMJDZJVOS-DEOSSOPVSA-N esomeprazole Chemical class C([S@](=O)C1=NC2=CC=C(C=C2N1)OC)C1=NC=C(C)C(OC)=C1C SUBDBMMJDZJVOS-DEOSSOPVSA-N 0.000 title abstract 3
- 150000003839 salts Chemical class 0.000 abstract 2
- SUBDBMMJDZJVOS-UHFFFAOYSA-N 5-methoxy-2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfinyl}-1H-benzimidazole Chemical compound N=1C2=CC(OC)=CC=C2NC=1S(=O)CC1=NC=C(C)C(OC)=C1C SUBDBMMJDZJVOS-UHFFFAOYSA-N 0.000 abstract 1
- 229960004770 esomeprazole Drugs 0.000 abstract 1
- 229960000381 omeprazole Drugs 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Oppfinnelsen angår en amorf form av saltene av enantiomeren av omeprazol, dvs. esomeprazol. Oppfinnelsen angår også fremgangsmåter for fremstilling av amorfe salter og farmasøytiske preparater som inkluderer de amorfe esomeprazolsaltene.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1057DE2002 | 2002-10-22 | ||
| PCT/IB2003/004662 WO2004037253A1 (en) | 2002-10-22 | 2003-10-22 | Amorphous form of esomeprazole salts |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20052474D0 NO20052474D0 (no) | 2005-05-23 |
| NO20052474L true NO20052474L (no) | 2005-05-23 |
Family
ID=32170658
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20052474A NO20052474L (no) | 2002-10-22 | 2005-05-23 | Amort form av esomeprazolsalter |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US20040235903A1 (no) |
| EP (1) | EP1556043A1 (no) |
| CN (1) | CN1728997A (no) |
| AU (1) | AU2003278406A1 (no) |
| BR (1) | BR0315574A (no) |
| EA (1) | EA200500673A1 (no) |
| NO (1) | NO20052474L (no) |
| WO (1) | WO2004037253A1 (no) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070224260A1 (en) * | 2004-04-15 | 2007-09-27 | Dr. Reddy's Laboratories Limited | Dosage Form Having Polymorphic Stability |
| BRPI0512522A (pt) | 2004-06-24 | 2008-03-11 | Astrazeneca Ab | processo para a preparação de sal de sódio de esomeprazol, composto, formulação farmacêutica, e, método de tratamento |
| ES2246149B1 (es) | 2004-07-02 | 2007-06-01 | Esteve Quimica, S.A. | Formas solidas de la sal magnesica de s-omeprazol y procedimientos para su preparacion. |
| US20080146615A1 (en) * | 2004-12-20 | 2008-06-19 | Dr. Reddy's Laboratories Limited | Pharmaceutical Compositions Comprising Amorphous Benzimidazole Compounds |
| US8658216B2 (en) | 2004-12-23 | 2014-02-25 | Ranbaxy Laboratories Limited | Stable oral benzimidazole compositions and process of preparation thereof |
| DE102005008412A1 (de) * | 2005-02-24 | 2006-09-07 | Ratiopharm Gmbh | Piperazinsalz des Omeprazols und dessen Enantiomere |
| CA2600456A1 (en) * | 2005-03-08 | 2006-09-14 | Dr. Reddy's Laboratories Ltd. | Process for preparing amorphous salts |
| EP1904064A4 (en) * | 2005-07-07 | 2009-12-02 | Reddys Lab Ltd Dr | OMEPRAZOLE OF FORM B |
| WO2007031845A2 (en) * | 2005-09-14 | 2007-03-22 | Glenmark Pharmaceuticals Limited | Polymorphic forms of (s)-omeprazole magnesium salts and processes for their preparation |
| EP1948637A4 (en) * | 2005-11-14 | 2010-09-08 | Hetero Drugs Ltd | PROCESS FOR AMORPHES ESOMEPRAZOLE |
| US8158152B2 (en) * | 2005-11-18 | 2012-04-17 | Scidose Llc | Lyophilization process and products obtained thereby |
| US8124779B2 (en) * | 2005-12-05 | 2012-02-28 | Astrazeneca Ab | Process for the preparation of esomeprazole non-salt form |
| EP1801110A1 (en) | 2005-12-22 | 2007-06-27 | KRKA, tovarna zdravil, d.d., Novo mesto | Esomeprazole arginine salt |
| US7553857B2 (en) * | 2005-12-23 | 2009-06-30 | Lek Pharmaceuticals D.D. | S-omeprazole magnesium |
| US20090197919A1 (en) * | 2006-06-07 | 2009-08-06 | Rolf Bergman | Novel Method for Preparation of Ammonium Salts of Esomeprazole |
| EA200900985A1 (ru) | 2007-01-31 | 2009-12-30 | Крка, Товарна Здравил, Д. Д., Ново Место | Способ получения оптически чистого омепразола |
| JP2010519284A (ja) | 2007-02-21 | 2010-06-03 | シプラ・リミテッド | エソメプラゾールマグネシウム二水和物の調製方法 |
| US8106210B2 (en) * | 2007-10-08 | 2012-01-31 | Hetero Drugs Limited | Polymorphs of esomeprazole salts |
| US8911787B2 (en) | 2008-02-26 | 2014-12-16 | Ranbaxy Laboratories Limited | Stable oral benzimidazole compositions and process of preparation thereof |
| EP2147918A1 (en) | 2008-07-21 | 2010-01-27 | LEK Pharmaceuticals D.D. | Process for the preparation of S-omeprazole magnesium in a stable form |
| WO2010097583A1 (en) * | 2009-02-24 | 2010-09-02 | Cipla Limited | Esomeprazole potassium polymorph and its preparation |
| WO2011095984A1 (en) * | 2010-02-02 | 2011-08-11 | Glenmark Generics Limited | A process for the preparation of amorphous esomeprazole |
| FR3062129B1 (fr) * | 2017-01-23 | 2019-04-05 | Minakem | Procede d'obtention du sel de magnesium dihydrate de l'esomeprazole |
| CN113387929A (zh) * | 2021-06-30 | 2021-09-14 | 江苏中邦制药有限公司 | 一种艾司奥美拉唑镁三水合物的制备方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
| SE8301182D0 (sv) * | 1983-03-04 | 1983-03-04 | Haessle Ab | Novel compounds |
| SE9301830D0 (sv) * | 1993-05-28 | 1993-05-28 | Ab Astra | New compounds |
| CA2180535C (en) * | 1994-01-05 | 2004-03-23 | Lindberg, Per Lennart | A method for treatment of psoriasis, by omeprazole or related compounds |
| SE504459C2 (sv) | 1994-07-15 | 1997-02-17 | Astra Ab | Förfarande för framställning av substituerade sulfoxider |
| SE508669C2 (sv) * | 1996-04-26 | 1998-10-26 | Astra Ab | Nytt förfarande |
| SE510666C2 (sv) * | 1996-12-20 | 1999-06-14 | Astra Ab | Nya Kristallmodifikationer |
| SE510650C2 (sv) | 1997-05-30 | 1999-06-14 | Astra Ab | Ny förening |
| SE510643C2 (sv) * | 1997-06-27 | 1999-06-14 | Astra Ab | Termodynamiskt stabil omeprazol natrium form B |
| US6124816A (en) * | 1998-06-02 | 2000-09-26 | Cirrus Logic, Inc. | One bit digital to analog converter with relaxed filtering requirements |
| US6262085B1 (en) * | 1999-08-26 | 2001-07-17 | Robert R. Whittle | Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
| CA2290893C (en) * | 1999-11-16 | 2007-05-01 | Bernard Charles Sherman | Magnesium omeprazole |
| US20030212274A1 (en) * | 2000-05-15 | 2003-11-13 | Bakthavathsalan Vijayaraghavan | Novel amorphous form of omeprazole salts |
| CA2386716C (en) * | 2002-05-17 | 2012-07-24 | Bernard Charles Sherman | Magnesium salt of s-omeprazole |
| AU2001276721A1 (en) * | 2000-08-04 | 2002-02-18 | Takeda Chemical Industries Ltd. | Salts of benzimidazole compound and use thereof |
| HU230155B1 (hu) * | 2001-07-16 | 2015-09-28 | Janssen Pharmaceutica N.V. | Javított eljárás benzimidazol típusú vegyületek előállítására |
| WO2004002982A2 (en) * | 2002-06-27 | 2004-01-08 | Dr. Reddy's Laboratories Limited | A process for preparation of optically pure or optically enriched sulfoxide compounds, including amorphous esomeprazole and salts thereof |
| US7651788B2 (en) * | 2003-03-05 | 2010-01-26 | Lg Display Co., Ltd. | Organic electroluminescent device |
-
2003
- 2003-10-22 EA EA200500673A patent/EA200500673A1/ru unknown
- 2003-10-22 BR BR0315574-9A patent/BR0315574A/pt not_active IP Right Cessation
- 2003-10-22 EP EP03769712A patent/EP1556043A1/en not_active Withdrawn
- 2003-10-22 US US10/690,897 patent/US20040235903A1/en not_active Abandoned
- 2003-10-22 WO PCT/IB2003/004662 patent/WO2004037253A1/en not_active Ceased
- 2003-10-22 CN CNA200380107036XA patent/CN1728997A/zh active Pending
- 2003-10-22 AU AU2003278406A patent/AU2003278406A1/en not_active Abandoned
-
2005
- 2005-05-23 NO NO20052474A patent/NO20052474L/no unknown
-
2007
- 2007-11-28 US US11/946,193 patent/US7482463B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| BR0315574A (pt) | 2005-09-20 |
| NO20052474D0 (no) | 2005-05-23 |
| US20040235903A1 (en) | 2004-11-25 |
| CN1728997A (zh) | 2006-02-01 |
| US7482463B2 (en) | 2009-01-27 |
| AU2003278406A1 (en) | 2004-05-13 |
| WO2004037253A1 (en) | 2004-05-06 |
| US20080119654A1 (en) | 2008-05-22 |
| EA200500673A1 (ru) | 2005-12-29 |
| EP1556043A1 (en) | 2005-07-27 |
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