NO20061655L - Behandling eller forebyggelse av restless legs syndron ved anvendelse av prodrug av GABA analoger - Google Patents
Behandling eller forebyggelse av restless legs syndron ved anvendelse av prodrug av GABA analogerInfo
- Publication number
- NO20061655L NO20061655L NO20061655A NO20061655A NO20061655L NO 20061655 L NO20061655 L NO 20061655L NO 20061655 A NO20061655 A NO 20061655A NO 20061655 A NO20061655 A NO 20061655A NO 20061655 L NO20061655 L NO 20061655L
- Authority
- NO
- Norway
- Prior art keywords
- prodrug
- prevention
- treatment
- restless legs
- legs syndrome
- Prior art date
Links
- BTCSSZJGUNDROE-UHFFFAOYSA-N gamma-aminobutyric acid Chemical class NCCCC(O)=O BTCSSZJGUNDROE-UHFFFAOYSA-N 0.000 title abstract 5
- 208000005793 Restless legs syndrome Diseases 0.000 title abstract 3
- 239000000651 prodrug Substances 0.000 title abstract 2
- 229940002612 prodrug Drugs 0.000 title abstract 2
- 230000002265 prevention Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- OGNSCSPNOLGXSM-UHFFFAOYSA-N (+/-)-DABA Natural products NCCC(N)C(O)=O OGNSCSPNOLGXSM-UHFFFAOYSA-N 0.000 abstract 1
- 229960003692 gamma aminobutyric acid Drugs 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/075—Ethers or acetals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Emergency Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US50417203P | 2003-09-17 | 2003-09-17 | |
| US50472603P | 2003-09-18 | 2003-09-18 | |
| US51227903P | 2003-10-17 | 2003-10-17 | |
| US53849504P | 2004-01-22 | 2004-01-22 | |
| PCT/US2004/030698 WO2005027850A2 (en) | 2003-09-17 | 2004-09-17 | Treating or preventing restless legs syndrome using prodrugs of gaba analogs |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20061655L true NO20061655L (no) | 2006-06-15 |
Family
ID=34382174
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20061655A NO20061655L (no) | 2003-09-17 | 2006-04-11 | Behandling eller forebyggelse av restless legs syndron ved anvendelse av prodrug av GABA analoger |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8114909B2 (pt) |
| EP (1) | EP1677812A4 (pt) |
| JP (1) | JP5107576B2 (pt) |
| KR (1) | KR101157436B1 (pt) |
| CN (1) | CN1871021B (pt) |
| AU (1) | AU2004274002B2 (pt) |
| BR (1) | BRPI0414481A (pt) |
| CA (1) | CA2538802C (pt) |
| IL (2) | IL174282A (pt) |
| MX (1) | MXPA06003043A (pt) |
| NO (1) | NO20061655L (pt) |
| NZ (2) | NZ579515A (pt) |
| SG (1) | SG146643A1 (pt) |
| WO (1) | WO2005027850A2 (pt) |
| ZA (1) | ZA200602182B (pt) |
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| EP1811986B1 (en) | 2004-11-04 | 2014-03-26 | XenoPort, Inc. | Gabapentin prodrug sustained release oral dosage forms |
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| CN102341098A (zh) * | 2009-03-06 | 2012-02-01 | 什诺波特有限公司 | 具有高负荷的加巴喷丁前药的口服剂型 |
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| CN105169266A (zh) * | 2015-10-02 | 2015-12-23 | 陈爱华 | 一种用于治疗不安腿综合征的药物制剂 |
| CN105777586A (zh) * | 2016-04-14 | 2016-07-20 | 安徽省逸欣铭医药科技有限公司 | S（+）氨己烯酸酯衍生物及其制备方法和用途 |
| RS65663B1 (sr) | 2018-02-15 | 2024-07-31 | Intrabio Ltd | Acetil leucin za upotrebu u lečenju sindroma nemirnih nogu |
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-
2004
- 2004-09-17 CA CA2538802A patent/CA2538802C/en not_active Expired - Lifetime
- 2004-09-17 AU AU2004274002A patent/AU2004274002B2/en not_active Expired
- 2004-09-17 WO PCT/US2004/030698 patent/WO2005027850A2/en not_active Ceased
- 2004-09-17 JP JP2006527100A patent/JP5107576B2/ja not_active Expired - Lifetime
- 2004-09-17 KR KR1020067005448A patent/KR101157436B1/ko not_active Expired - Lifetime
- 2004-09-17 MX MXPA06003043A patent/MXPA06003043A/es active IP Right Grant
- 2004-09-17 SG SG200806876-9A patent/SG146643A1/en unknown
- 2004-09-17 NZ NZ579515A patent/NZ579515A/en not_active IP Right Cessation
- 2004-09-17 EP EP04788836A patent/EP1677812A4/en not_active Withdrawn
- 2004-09-17 US US10/969,196 patent/US8114909B2/en not_active Expired - Lifetime
- 2004-09-17 CN CN2004800311096A patent/CN1871021B/zh not_active Expired - Fee Related
- 2004-09-17 NZ NZ545989A patent/NZ545989A/en not_active IP Right Cessation
- 2004-09-17 BR BRPI0414481-3A patent/BRPI0414481A/pt not_active Application Discontinuation
-
2006
- 2006-03-13 IL IL174282A patent/IL174282A/en not_active IP Right Cessation
- 2006-03-15 ZA ZA2006/02182A patent/ZA200602182B/en unknown
- 2006-04-11 NO NO20061655A patent/NO20061655L/no not_active Application Discontinuation
-
2009
- 2009-09-01 IL IL200687A patent/IL200687A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL174282A0 (en) | 2006-08-01 |
| WO2005027850A2 (en) | 2005-03-31 |
| IL174282A (en) | 2012-12-31 |
| KR20060106815A (ko) | 2006-10-12 |
| AU2004274002A1 (en) | 2005-03-31 |
| CA2538802A1 (en) | 2005-03-31 |
| CN1871021A (zh) | 2006-11-29 |
| US8114909B2 (en) | 2012-02-14 |
| AU2004274002B2 (en) | 2011-04-28 |
| IL200687A0 (en) | 2011-08-01 |
| CN1871021B (zh) | 2010-07-28 |
| CA2538802C (en) | 2015-01-27 |
| KR101157436B1 (ko) | 2012-07-05 |
| NZ579515A (en) | 2011-09-30 |
| ZA200602182B (en) | 2012-07-25 |
| EP1677812A2 (en) | 2006-07-12 |
| JP2007511464A (ja) | 2007-05-10 |
| NZ545989A (en) | 2009-10-30 |
| BRPI0414481A (pt) | 2006-11-14 |
| MXPA06003043A (es) | 2006-05-31 |
| WO2005027850A3 (en) | 2005-06-16 |
| EP1677812A4 (en) | 2010-03-24 |
| US20050192353A1 (en) | 2005-09-01 |
| SG146643A1 (en) | 2008-10-30 |
| JP5107576B2 (ja) | 2012-12-26 |
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