NO20072687L - Pharmaceutical contraceptive preparation - Google Patents

Pharmaceutical contraceptive preparation

Info

Publication number
NO20072687L
NO20072687L NO20072687A NO20072687A NO20072687L NO 20072687 L NO20072687 L NO 20072687L NO 20072687 A NO20072687 A NO 20072687A NO 20072687 A NO20072687 A NO 20072687A NO 20072687 L NO20072687 L NO 20072687L
Authority
NO
Norway
Prior art keywords
daily dosage
ethinyl estradiol
administered
dienogest
pharmaceutically acceptable
Prior art date
Application number
NO20072687A
Other languages
Norwegian (no)
Inventor
Thomas Graser
Claus Claussen
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of NO20072687L publication Critical patent/NO20072687L/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Oppfinnelsen vedrører et farmasøytisk preparat som inneholder dienogest ved en mengde som tilsvarer en daglig doseringsenhet på 1,5 mg eller 2,0 mg når preparatet blir administrert, og etinyløstradiol ved en mengde som tilsvarer en daglig doseringsenhet på 0,015 mg eller 0,020 mg når preparatet blir administrert, sammen med én eller flere farmasøytisk akseptable bærere i minst 21 daglige doseringsenheter. Oppfinnelsen vedrører ytterligere et oralt, farmasøytisk prevensjonspreparat inneholdende 1,5 mg 17a-cyanometyl-17ß-hydroksyøstra-4,9-dien-3-on (dienogest) og 0,015 eller 0,020 mg 17a-etinyløstradiol (etinyløstradiol) eller 2,0 mg dienogest og 0,015 mg etinyløstradiol sammen med én eller flere farmasøytisk akseptable bærer i minst 21 daglige doseringsenheter i en 28-dagers menstruasjonssyklus.The invention relates to a pharmaceutical composition containing dienogest at an amount corresponding to a daily dosage unit of 1.5 mg or 2.0 mg when administered, and ethinyl estradiol at an amount corresponding to a daily dosage unit of 0.015 mg or 0.020 mg when the preparation is administered. administered with one or more pharmaceutically acceptable carriers in at least 21 daily dosage units. The invention further relates to an oral pharmaceutical contraceptive composition containing 1.5 mg of 17α-cyanomethyl-17β-hydroxyester-4,9-dien-3-one (dienogest) and 0.015 or 0.020 mg of 17α-ethinyl estradiol (ethinyl estradiol) or 2.0 mg dienogest and 0.015 mg of ethinyl estradiol together with one or more pharmaceutically acceptable carriers in at least 21 daily dosage units during a 28-day menstrual cycle.

NO20072687A 2005-02-15 2007-05-25 Pharmaceutical contraceptive preparation NO20072687L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05003179A EP1690543A1 (en) 2005-02-15 2005-02-15 Pharmaceutical composition for contraception
PCT/EP2006/001354 WO2006087173A1 (en) 2005-02-15 2006-02-15 Contraceptive pharmaceutical preparation

Publications (1)

Publication Number Publication Date
NO20072687L true NO20072687L (en) 2007-11-13

Family

ID=34933759

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072687A NO20072687L (en) 2005-02-15 2007-05-25 Pharmaceutical contraceptive preparation

Country Status (20)

Country Link
EP (2) EP1690543A1 (en)
JP (1) JP2008527018A (en)
KR (1) KR20070086380A (en)
CN (1) CN101119732A (en)
AR (1) AR053545A1 (en)
AU (1) AU2006215818A1 (en)
BR (1) BRPI0606724A2 (en)
CA (1) CA2590004A1 (en)
CR (1) CR9324A (en)
DO (1) DOP2006000035A (en)
EA (1) EA200701091A1 (en)
IL (1) IL183635A0 (en)
MX (1) MX2007009061A (en)
NO (1) NO20072687L (en)
PA (1) PA8663401A1 (en)
PE (1) PE20061291A1 (en)
TW (1) TW200640468A (en)
UA (1) UA85003C2 (en)
WO (1) WO2006087173A1 (en)
ZA (1) ZA200707910B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1774970A1 (en) * 2005-10-13 2007-04-18 Bayer Schering Pharma AG Method for preparing a monophase pharnmaceutical preparation containing ethinyl estradiol and dienogest for the treatment of dysfunctional uterine bleeding
DE102008051140B4 (en) * 2007-10-11 2010-06-10 Bayer Schering Pharma Aktiengesellschaft A process for the preparation of a monophasic pharmaceutical preparation for limiting / reducing the risk of deep vein thrombosis in unit with oral contraception
AT12800U1 (en) * 2007-11-05 2012-11-15 Bayer Schering Pharma Ag A pharmaceutical preparation for use in the oral contraception of lactose intolerant women

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998004269A1 (en) * 1996-07-26 1998-02-05 American Home Products Corporation Monophasic contraceptive method and kit comprising a combination of a progestin and estrogen

Also Published As

Publication number Publication date
WO2006087173A1 (en) 2006-08-24
EA200701091A1 (en) 2008-02-28
UA85003C2 (en) 2008-12-10
IL183635A0 (en) 2007-10-31
TW200640468A (en) 2006-12-01
CN101119732A (en) 2008-02-06
PE20061291A1 (en) 2006-12-07
PA8663401A1 (en) 2006-12-07
MX2007009061A (en) 2007-09-11
AU2006215818A1 (en) 2006-08-24
BRPI0606724A2 (en) 2009-07-14
CR9324A (en) 2007-10-11
EP1690543A1 (en) 2006-08-16
CA2590004A1 (en) 2006-08-24
KR20070086380A (en) 2007-08-27
ZA200707910B (en) 2009-08-26
DOP2006000035A (en) 2006-09-15
JP2008527018A (en) 2008-07-24
AR053545A1 (en) 2007-05-09
EP1853273A1 (en) 2007-11-14

Similar Documents

Publication Publication Date Title
ES2558030T3 (en) Long-cycle multiphase oral contraceptive method
HRP20070188B1 (en) PHARMACEUTICAL COMBINATION OF ETHINYLESTRADIOL AND DROSPIRENONE FOR USE AS A CONTRACEPTIC
EA200900491A1 (en) USE OF ESTRADIOL VALERAT OR 17B-ESTRADIOL IN COMBINATION WITH DIENOGEST FOR ORAL TREATMENT TO MAINTAIN AND / OR INCREASE SEXUAL TREATMENT IN THE SPECIAL WOMAN
BG66095B1 (en) Pregelatinized starch in a controlled release preparation
NO327588B1 (en) Pharmaceutical composition and composition comprising ethinylostradiol and drospirenone for use as a contraceptive
NO20072893L (en) Solid oral contraceptive
HRP20090256T1 (en) Use of estradiolvalerate and dienogest for oral treatment of dysfunctional uterine bleeding in a contraceptive method
CR9324A (en) PHARMACEUTICAL PREPARATION FOR ORAL ANTI-CONCEPTION
WO2005092441A3 (en) Extended cycle multiphasic oral contraceptive method
TW200638951A (en) Solid oral pharmaceutical form for contraception
NO20091057L (en) Oral form of birth control
UY29378A1 (en) PHARMACEUTICAL PREPARATION FOR ORAL ANTI-CONCEPTION
CY1112775T1 (en) USE OF VALERIAN OSTRADIOLIS IN CONNECTION WITH DIENOGEST FOR ORAL TREATMENT OF MUTRAL DISORDER BLOOD TREATMENT IN AITITA
TH80557A (en) Pharmaceutical products for oral contraception
JO2213B1 (en) A pharmaceutical composition for use as a contraceptive
RU2009140372A (en) NEW MODE WITH DROSPIRENONE / 17B-ESTRADIOL, PHARMACEUTICAL COMBINED PRODUCT AND KIT FOR THE PERFORMANCE OF THIS MODE
HRP20020666B1 (en) DROSPIRENON FOR HORMONAL REPLACEMENT THERAPY

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application