NO20073387L - Benzdioksanpiperazinderivater med en kombinasjon av affinitet for dopamin-D2-reseptorer og serotoninreopptaksseter - Google Patents

Benzdioksanpiperazinderivater med en kombinasjon av affinitet for dopamin-D2-reseptorer og serotoninreopptaksseter

Info

Publication number
NO20073387L
NO20073387L NO20073387A NO20073387A NO20073387L NO 20073387 L NO20073387 L NO 20073387L NO 20073387 A NO20073387 A NO 20073387A NO 20073387 A NO20073387 A NO 20073387A NO 20073387 L NO20073387 L NO 20073387L
Authority
NO
Norway
Prior art keywords
dopamine
receptors
affinity
serotonin reuptake
benz
Prior art date
Application number
NO20073387A
Other languages
English (en)
Inventor
Cornelis G Kruse
Roelof Van Hes
Pieter Smid
Martinus Th M Tulp
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2005/056503 external-priority patent/WO2006061374A1/en
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of NO20073387L publication Critical patent/NO20073387L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Den foreliggende oppfinnelsen vedrører en gruppe nye 3-(2-piperidin-4-yl-etyl)-1H-indol derivater med todelt virkemåte: serotonin-reopptaksinhibisjon og affinitet for dopamin-D2 reseptorer, og fremgangsmåter for fremstilling av disse forbindelsene. Oppfinnelsen vedrører også anvendelsen av en forbindelse som her er beskrevet for fremstilling av et medikament som gir en fordelaktig effekt. Forbindelsene har den generelle formel (I) der symbolene har betydningene som er gitt i teksten.
NO20073387A 2004-12-07 2007-07-02 Benzdioksanpiperazinderivater med en kombinasjon av affinitet for dopamin-D2-reseptorer og serotoninreopptaksseter NO20073387L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63344704P 2004-12-07 2004-12-07
EP04106361 2004-12-07
PCT/EP2005/056503 WO2006061374A1 (en) 2004-12-07 2005-12-06 Benzdioxane piperazine derivatives with a combination of affinity for dopamine-d2 receptors and serotonin reuptake sites

Publications (1)

Publication Number Publication Date
NO20073387L true NO20073387L (no) 2007-07-02

Family

ID=35781191

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20073387A NO20073387L (no) 2004-12-07 2007-07-02 Benzdioksanpiperazinderivater med en kombinasjon av affinitet for dopamin-D2-reseptorer og serotoninreopptaksseter

Country Status (3)

Country Link
DE (1) DE602005013424D1 (no)
IL (1) IL183203A0 (no)
NO (1) NO20073387L (no)

Also Published As

Publication number Publication date
DE602005013424D1 (de) 2009-04-30
IL183203A0 (en) 2007-08-19

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Legal Events

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