NO20090214L - Proteinkinase C aktivitetsforsterker inneholdende alkyleterderivat eller et salt av denne - Google Patents
Proteinkinase C aktivitetsforsterker inneholdende alkyleterderivat eller et salt av denneInfo
- Publication number
- NO20090214L NO20090214L NO20090214A NO20090214A NO20090214L NO 20090214 L NO20090214 L NO 20090214L NO 20090214 A NO20090214 A NO 20090214A NO 20090214 A NO20090214 A NO 20090214A NO 20090214 L NO20090214 L NO 20090214L
- Authority
- NO
- Norway
- Prior art keywords
- group
- protein kinase
- salt
- ether derivative
- alkyl ether
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Beskrevet er en proteinkinase C forsterker karakterisert ved at den inneholder et benzotiofenalkyleterderivat representert ved den generelle formel nedenfor eller et salt derav. (I formelen, R1 og R2 kan være like eller forskjellige og representerer én eller flere grupper valgt fra et hydrogenatom, et halogenatom, en alkylgruppe, en arylgruppe, en aralkylgruppe, en alkoksygruppe, en aryloksygruppe, en alkenylgruppe, en aminogruppe, en heterocyklisk gruppe, en eventuelt beskyttet aminogruppe, en hydroksylgruppe, en karboksylgruppe, en oksogruppe og lignende; R3 representerer en alkylaminogruppe, en aminogruppe, en hydroksylgruppe eller lignende; og m og n kan være like eller forskjellige og representerer et helt tall på 1-6.) Denne proteinkinase C forsterker er anvendelige for behandling eller forebygging av forskjellige sykdommer forbundet med proteinkinase C.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2006212722 | 2006-08-04 | ||
| PCT/JP2007/065165 WO2008016107A1 (en) | 2006-08-04 | 2007-08-02 | Protein kinase c activity enhancer containing alkyl ether derivative or salt thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20090214L true NO20090214L (no) | 2009-01-30 |
Family
ID=38997281
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20090214A NO20090214L (no) | 2006-08-04 | 2009-01-14 | Proteinkinase C aktivitetsforsterker inneholdende alkyleterderivat eller et salt av denne |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US8173633B2 (no) |
| EP (1) | EP2048145B9 (no) |
| JP (1) | JP5255441B2 (no) |
| KR (1) | KR20090038471A (no) |
| CN (1) | CN101501026B (no) |
| AT (1) | ATE491705T1 (no) |
| AU (1) | AU2007279673B2 (no) |
| BR (1) | BRPI0715056A2 (no) |
| CA (1) | CA2659835A1 (no) |
| CY (1) | CY1111691T1 (no) |
| DE (1) | DE602007011281D1 (no) |
| DK (1) | DK2048145T3 (no) |
| ES (1) | ES2355768T3 (no) |
| IL (1) | IL196754A0 (no) |
| MX (1) | MX2009001255A (no) |
| NO (1) | NO20090214L (no) |
| NZ (1) | NZ574551A (no) |
| PL (1) | PL2048145T3 (no) |
| PT (1) | PT2048145E (no) |
| SI (1) | SI2048145T1 (no) |
| WO (1) | WO2008016107A1 (no) |
| ZA (1) | ZA200900743B (no) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2464358C (en) | 2001-10-19 | 2011-05-24 | Toyama Chemical Co., Ltd. | Alkyl ether derivatives or their salts |
| ATE491705T1 (de) * | 2006-08-04 | 2011-01-15 | Toyama Chemical Co Ltd | Verstärker der aktivität von proteinkinase c, enthaltend ein alkyletherderivat oder ein salz davon |
| PL2287160T3 (pl) * | 2008-05-28 | 2014-09-30 | Toyama Chemical Co Ltd | Pochodna tlenku benzotiofenu i jej sól |
| AU2012335220B2 (en) | 2011-11-11 | 2017-06-01 | Pfizer Inc. | 2-thiopyrimidinones |
| BR112014020434B1 (pt) * | 2012-02-22 | 2021-10-13 | Fujifilm Toyama Chemical Co., Ltd. | Composição farmacêutica sólida |
| US10238632B2 (en) | 2015-06-11 | 2019-03-26 | Fujifilm Toyama Chemical Co., Ltd. | Sigma receptor-binding agent |
| WO2017111005A1 (ja) * | 2015-12-25 | 2017-06-29 | 富山化学工業株式会社 | １－（３－（２－（１－ベンゾチオフェン－５－イル）エトキシ）プロピル）アゼチジン－３－オールまたはその塩を含む錠剤 |
| EP3563846B1 (en) * | 2016-12-28 | 2023-07-19 | FUJIFILM Toyama Chemical Co., Ltd. | Pharmaceutical composition and method for producing the same |
| WO2018124284A1 (ja) * | 2016-12-28 | 2018-07-05 | 富山化学工業株式会社 | 医薬組成物 |
| WO2018124283A1 (ja) * | 2016-12-28 | 2018-07-05 | 富山化学工業株式会社 | 医薬組成物 |
| WO2018124281A1 (ja) * | 2016-12-28 | 2018-07-05 | 富山化学工業株式会社 | 外用組成物 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH09507846A (ja) * | 1993-12-30 | 1997-08-12 | スミスクライン・ビーチャム・コーポレイション | フェニルメチルヘキサンアミドおよびその使用 |
| US6809092B2 (en) | 2000-01-26 | 2004-10-26 | Ono Pharmaceutical Co., Ltd. | Benezene-fused heteroring derivatives and pharmaceutical agents comprising the same as active ingredient |
| JP4303435B2 (ja) * | 2001-02-26 | 2009-07-29 | 富山化学工業株式会社 | ミトコンドリア機能賦活剤 |
| CA2464358C (en) * | 2001-10-19 | 2011-05-24 | Toyama Chemical Co., Ltd. | Alkyl ether derivatives or their salts |
| US6825229B2 (en) * | 2002-03-07 | 2004-11-30 | Blanchette Rockefeller Neurosciences Institute | Methods for Alzheimer's Disease treatment and cognitive enhancement |
| KR100935615B1 (ko) * | 2002-06-14 | 2010-01-07 | 토야마 케미칼 컴퍼니 리미티드 | 뇌기능을 개선하는 의약조성물 및 뇌기능을 개선하기 위한방법 |
| US7335689B2 (en) * | 2003-01-23 | 2008-02-26 | Esperion Therapeutics, Inc. | Dihydroxyl compounds and compositions for cholesterol management and related uses |
| ZA200508166B (en) * | 2003-04-17 | 2007-03-28 | Toyama Chemical Co Ltd | Preventive/remedy for retinal nerve diseases containing alkyl ether derivatives or salts thereof |
| SE529122C2 (sv) * | 2004-09-24 | 2007-05-02 | Jokab Safety Ab | Skyddsanordning för områdesbegränsning och övervakning |
| SI2348022T1 (sl) * | 2005-03-28 | 2013-05-31 | Toyama Chemical Co., Ltd. | Postopek proizvodnje 1-(3-(2-(1-benzotiofen-5-il)etoksi)propil)azetidin-3-ola ali soli le-tega |
| JP4902247B2 (ja) * | 2005-04-08 | 2012-03-21 | 富山化学工業株式会社 | ２−（１−ベンゾチオフェン−５−イル）エタノールの新規製造法およびその中間体 |
| ES2518371T3 (es) * | 2006-04-26 | 2014-11-05 | Toyama Chemical Co., Ltd. | Inductor de la neurogénesis o agente terapéutico para la neuropatía que comprende un derivado de éter alquílico o una sal del mismo |
| ATE491705T1 (de) * | 2006-08-04 | 2011-01-15 | Toyama Chemical Co Ltd | Verstärker der aktivität von proteinkinase c, enthaltend ein alkyletherderivat oder ein salz davon |
-
2007
- 2007-08-02 AT AT07791845T patent/ATE491705T1/de active
- 2007-08-02 DK DK07791845.6T patent/DK2048145T3/da active
- 2007-08-02 PL PL07791845T patent/PL2048145T3/pl unknown
- 2007-08-02 KR KR1020097003927A patent/KR20090038471A/ko not_active Ceased
- 2007-08-02 AU AU2007279673A patent/AU2007279673B2/en not_active Ceased
- 2007-08-02 JP JP2008527788A patent/JP5255441B2/ja not_active Expired - Fee Related
- 2007-08-02 MX MX2009001255A patent/MX2009001255A/es active IP Right Grant
- 2007-08-02 CA CA002659835A patent/CA2659835A1/en not_active Abandoned
- 2007-08-02 BR BRPI0715056-3A patent/BRPI0715056A2/pt not_active IP Right Cessation
- 2007-08-02 WO PCT/JP2007/065165 patent/WO2008016107A1/ja not_active Ceased
- 2007-08-02 PT PT07791845T patent/PT2048145E/pt unknown
- 2007-08-02 DE DE602007011281T patent/DE602007011281D1/de active Active
- 2007-08-02 ES ES07791845T patent/ES2355768T3/es active Active
- 2007-08-02 SI SI200730516T patent/SI2048145T1/sl unknown
- 2007-08-02 CN CN2007800291310A patent/CN101501026B/zh not_active Expired - Fee Related
- 2007-08-02 US US12/376,296 patent/US8173633B2/en not_active Expired - Fee Related
- 2007-08-02 ZA ZA200900743A patent/ZA200900743B/xx unknown
- 2007-08-02 NZ NZ574551A patent/NZ574551A/en unknown
- 2007-08-02 EP EP07791845A patent/EP2048145B9/en not_active Not-in-force
-
2009
- 2009-01-14 NO NO20090214A patent/NO20090214L/no not_active Application Discontinuation
- 2009-01-27 IL IL196754A patent/IL196754A0/en unknown
-
2011
- 2011-02-14 CY CY20111100176T patent/CY1111691T1/el unknown
- 2011-06-17 US US13/163,105 patent/US20110245228A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN101501026A (zh) | 2009-08-05 |
| MX2009001255A (es) | 2009-06-12 |
| PL2048145T3 (pl) | 2011-09-30 |
| WO2008016107A1 (en) | 2008-02-07 |
| EP2048145B9 (en) | 2011-05-04 |
| CY1111691T1 (el) | 2015-10-07 |
| BRPI0715056A2 (pt) | 2013-05-28 |
| EP2048145A1 (en) | 2009-04-15 |
| ZA200900743B (en) | 2010-05-26 |
| DK2048145T3 (da) | 2011-04-04 |
| US20100184997A1 (en) | 2010-07-22 |
| US20110245228A1 (en) | 2011-10-06 |
| JP5255441B2 (ja) | 2013-08-07 |
| PT2048145E (pt) | 2011-01-14 |
| KR20090038471A (ko) | 2009-04-20 |
| JPWO2008016107A1 (ja) | 2009-12-24 |
| NZ574551A (en) | 2012-03-30 |
| EP2048145B1 (en) | 2010-12-15 |
| AU2007279673B2 (en) | 2012-04-19 |
| DE602007011281D1 (de) | 2011-01-27 |
| IL196754A0 (en) | 2009-11-18 |
| ATE491705T1 (de) | 2011-01-15 |
| EP2048145A4 (en) | 2009-09-09 |
| US8173633B2 (en) | 2012-05-08 |
| CN101501026B (zh) | 2012-04-04 |
| SI2048145T1 (sl) | 2011-04-29 |
| AU2007279673A1 (en) | 2008-02-07 |
| ES2355768T3 (es) | 2011-03-30 |
| CA2659835A1 (en) | 2008-02-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |