NO20091664L - Farmaoytiske preparater av HDAC-inhibitorer og chelaterbare metallforbindelser samt metall-HDAC-inhibitor-chelatkomplekser - Google Patents

Farmaoytiske preparater av HDAC-inhibitorer og chelaterbare metallforbindelser samt metall-HDAC-inhibitor-chelatkomplekser

Info

Publication number
NO20091664L
NO20091664L NO20091664A NO20091664A NO20091664L NO 20091664 L NO20091664 L NO 20091664L NO 20091664 A NO20091664 A NO 20091664A NO 20091664 A NO20091664 A NO 20091664A NO 20091664 L NO20091664 L NO 20091664L
Authority
NO
Norway
Prior art keywords
metal
hdac inhibitor
chelate complexes
hdac
well
Prior art date
Application number
NO20091664A
Other languages
English (en)
Norwegian (no)
Inventor
Arlene E Mckeown
Thomas A Miller
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of NO20091664L publication Critical patent/NO20091664L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/28—Compounds containing heavy metals
    • A61K31/295—Iron group metal compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/24—Heavy metals; Compounds thereof
    • A61K33/26—Iron; Compounds thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/24—Heavy metals; Compounds thereof
    • A61K33/30—Zinc; Compounds thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20091664A 2006-09-28 2009-04-27 Farmaoytiske preparater av HDAC-inhibitorer og chelaterbare metallforbindelser samt metall-HDAC-inhibitor-chelatkomplekser NO20091664L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US84830006P 2006-09-28 2006-09-28
PCT/US2007/020609 WO2008039421A2 (en) 2006-09-28 2007-09-24 Pharmaceutical compositions of hdac inhibitors and chelatable metal compounds, and metal-hdac inhibitor chelate complexes

Publications (1)

Publication Number Publication Date
NO20091664L true NO20091664L (no) 2009-04-27

Family

ID=39230785

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20091664A NO20091664L (no) 2006-09-28 2009-04-27 Farmaoytiske preparater av HDAC-inhibitorer og chelaterbare metallforbindelser samt metall-HDAC-inhibitor-chelatkomplekser

Country Status (14)

Country Link
US (2) US20090239946A1 (pt)
EP (2) EP2436382A1 (pt)
JP (1) JP2010504968A (pt)
KR (1) KR20090064400A (pt)
CN (1) CN101528212A (pt)
AU (1) AU2007300532A1 (pt)
BR (1) BRPI0717554A2 (pt)
CA (1) CA2663569A1 (pt)
CO (1) CO6190508A2 (pt)
IL (1) IL197718A0 (pt)
MX (1) MX2009003405A (pt)
NO (1) NO20091664L (pt)
RU (1) RU2009115860A (pt)
WO (1) WO2008039421A2 (pt)

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EP2085397A1 (en) * 2008-01-21 2009-08-05 Esteve Quimica, S.A. Crystalline form of abacavir
US7935817B2 (en) * 2008-03-31 2011-05-03 Apotex Pharmachem Inc. Salt form and cocrystals of adefovir dipivoxil and processes for preparation thereof
AR071318A1 (es) * 2008-04-15 2010-06-09 Basilea Pharmaceutica Ag Benzhidril ester del acido (6r,7r)-7-{2-(5-amino-[1,2,4]tiadiazol-3-il)-2-[(z)-tritiloxiimino]-acetilamino}-3-[(r)-1'-terc-butoxicarbonil-2-oxo-[1,3']bipirrolidinil-(3e)-ilidenometil]-8-oxo-5-tia-1-aza-biciclo[4.2.0]oct-2-eno-2-carboxilico cristalino; su elaboracion y uso
US8097719B2 (en) * 2008-07-15 2012-01-17 Genesen Labs Meropenem intermediate in novel crystalline form and a method of manufacture of meropenem
US8883851B2 (en) 2008-10-15 2014-11-11 Generics [Uk] Limited Process for the preparation of vorinostat
WO2010062333A1 (en) * 2008-10-27 2010-06-03 Plus Chemicals Sa Polymorphs of vorinostat and vorinostat potassium salt and process for preparation thereof
JP2012509929A (ja) * 2008-11-26 2012-04-26 ジェネリクス・（ユーケー）・リミテッド 多型
KR101713453B1 (ko) 2010-03-12 2017-03-07 오메로스 코포레이션 Pde10 억제제 및 관련 조성물 및 방법
JP2013536859A (ja) * 2010-09-01 2013-09-26 アリーナ ファーマシューティカルズ， インコーポレイテッド ５−ｈｔ２ｃアゴニストの非吸湿性塩
EP2760859A1 (en) * 2011-09-30 2014-08-06 Sunshine Lake Pharma Co., Ltd Crystalline forms of azilsartan and preparation and uses thereof
US20150141470A1 (en) 2012-05-08 2015-05-21 The Broad Institute, Inc. Diagnostic and treatment methods in patients having or at risk of developing resistance to cancer therapy
TWI483721B (zh) 2013-09-05 2015-05-11 Profeat Biotechnology Co Ltd The use of a composition containing a ferrous amino acid chelate for the manufacture of anti-cancer medicaments
JP5973684B2 (ja) * 2013-09-05 2016-08-23 普惠徳生技股▲ふん▼有限公司 癌治療のための使用
NZ630803A (en) 2014-04-28 2016-03-31 Omeros Corp Optically active pde10 inhibitor
NZ716494A (en) 2014-04-28 2017-07-28 Omeros Corp Processes and intermediates for the preparation of a pde10 inhibitor
US10413517B2 (en) * 2014-06-12 2019-09-17 University Of Notre Dame Du Lac Composition and method for the treatment of neurological diseases and cerebral injury
KR20170139074A (ko) 2015-04-24 2017-12-18 오메로스 코포레이션 Pde10 억제제 및 관련 조성물 및 방법
WO2017079678A1 (en) 2015-11-04 2017-05-11 Omeros Corporation Solid state forms of a pde10 inhibitor
CN107362148B (zh) * 2017-07-27 2020-04-21 东曜药业有限公司 一种治疗肿瘤的药物组合物及其制备方法和应用
IL326637A (en) * 2017-09-07 2026-04-01 Atnx Spv Llc Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-N-benzylacetamide
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
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CN111303230B (zh) * 2020-03-09 2021-07-13 中国食品药品检定研究院 一种黄体酮共晶物及其制备方法和用途

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Also Published As

Publication number Publication date
WO2008039421A3 (en) 2008-07-24
CO6190508A2 (es) 2010-08-19
EP2079462A4 (en) 2009-12-02
MX2009003405A (es) 2009-04-09
US20090239946A1 (en) 2009-09-24
RU2009115860A (ru) 2010-11-20
CA2663569A1 (en) 2008-04-03
WO2008039421A2 (en) 2008-04-03
IL197718A0 (en) 2009-12-24
AU2007300532A1 (en) 2008-04-03
US20120142770A1 (en) 2012-06-07
CN101528212A (zh) 2009-09-09
EP2079462A2 (en) 2009-07-22
BRPI0717554A2 (pt) 2013-10-29
JP2010504968A (ja) 2010-02-18
EP2436382A1 (en) 2012-04-04
KR20090064400A (ko) 2009-06-18

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