NO325501B1 - Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. - Google Patents
Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. Download PDFInfo
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- NO325501B1 NO325501B1 NO20032390A NO20032390A NO325501B1 NO 325501 B1 NO325501 B1 NO 325501B1 NO 20032390 A NO20032390 A NO 20032390A NO 20032390 A NO20032390 A NO 20032390A NO 325501 B1 NO325501 B1 NO 325501B1
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Classifications
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Anesthesiology (AREA)
- Reproductive Health (AREA)
- Nutrition Science (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25330100P | 2000-11-28 | 2000-11-28 | |
| US29781401P | 2001-06-13 | 2001-06-13 | |
| PCT/US2001/043160 WO2002044142A2 (en) | 2000-11-28 | 2001-11-27 | Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20032390D0 NO20032390D0 (no) | 2003-05-27 |
| NO20032390L NO20032390L (no) | 2003-07-22 |
| NO325501B1 true NO325501B1 (no) | 2008-05-26 |
Family
ID=26943115
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20032390A NO325501B1 (no) | 2000-11-28 | 2003-05-27 | Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. |
Country Status (24)
| Country | Link |
|---|---|
| US (3) | US6469007B2 (de) |
| EP (1) | EP1339406B1 (de) |
| JP (1) | JP4198989B2 (de) |
| KR (1) | KR100835552B1 (de) |
| CN (1) | CN100352437C (de) |
| AR (1) | AR035603A1 (de) |
| AT (1) | ATE269078T1 (de) |
| AU (2) | AU2002237654B2 (de) |
| BR (1) | BR0115609A (de) |
| CA (1) | CA2428039C (de) |
| DE (1) | DE60103927T2 (de) |
| DK (1) | DK1339406T3 (de) |
| EA (1) | EA005925B1 (de) |
| ES (1) | ES2222401T3 (de) |
| HU (1) | HUP0400551A2 (de) |
| IL (1) | IL156098A0 (de) |
| MX (1) | MXPA03004677A (de) |
| NO (1) | NO325501B1 (de) |
| NZ (1) | NZ526150A (de) |
| PL (1) | PL363219A1 (de) |
| PT (1) | PT1339406E (de) |
| TR (1) | TR200401546T4 (de) |
| TW (1) | TWI224102B (de) |
| WO (1) | WO2002044142A2 (de) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US6432826B1 (en) * | 1999-11-29 | 2002-08-13 | Applied Materials, Inc. | Planarized Cu cleaning for reduced defects |
| US20060287335A1 (en) | 2000-11-28 | 2006-12-21 | Wyeth | Serotonergic agents for treating sexual dysfunction |
| US20060223824A1 (en) * | 2000-11-28 | 2006-10-05 | Wyeth | Serotonergic agents |
| ES2323451T7 (es) | 2001-07-20 | 2011-08-01 | Psychogenics Inc. | Tratamiento para el trastorno de hiperactividad con deficit de atencion. |
| ES2329122T3 (es) | 2002-03-12 | 2009-11-23 | Wyeth | Procedimiento para sintetizar n-aril piperazinas quirales. |
| US7091349B2 (en) | 2002-03-12 | 2006-08-15 | Wyeth | Process for synthesizing N-aryl piperazines with chiral N′-1-[benzoyl(2-pyridyl)amino]-2-propane substitution |
| BR0308347A (pt) | 2002-03-12 | 2005-01-25 | Wyeth Corp | Processo para fabricação de piperazinas 1,4-dissubstituìdas quirais |
| US7361773B2 (en) | 2002-03-12 | 2008-04-22 | Wyeth | Preparation of N1-(2'-pyridyl)-1,2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines |
| GB0219961D0 (en) * | 2002-08-28 | 2002-10-02 | Pfizer Ltd | Oxytocin inhibitors |
| WO2004082686A2 (en) * | 2003-03-13 | 2004-09-30 | Dynogen Pharmaceuticals, Inc. | Use of compounds with combined 5-ht1a and ssri activities to treat sexual dysfunction |
| US20050215561A1 (en) * | 2004-03-19 | 2005-09-29 | Krishnendu Ghosh | Pharmaceutical dosage forms and compositions |
| US20050209245A1 (en) * | 2004-03-19 | 2005-09-22 | Wyeth | Process for preparing N-aryl-piperazine derivatives |
| US20070099931A1 (en) * | 2004-03-19 | 2007-05-03 | Wyeth | Pharmaceutical dosage forms and compositions |
| KR100646337B1 (ko) * | 2004-06-30 | 2006-11-23 | 주식회사 롯데기공 | 보일러의 누수 감지방법 |
| AU2005295640B2 (en) * | 2004-10-15 | 2011-07-28 | The Government Of The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services | Multi-domain amphipathic helical peptides and methods of their use |
| TW200700413A (en) * | 2005-03-01 | 2007-01-01 | Wyeth Corp | Crystalline and amorphous 4-cyano-n-{(2r)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-n-pyridin-2-yl-benzamide hydrochloride |
| TW200800959A (en) * | 2005-06-10 | 2008-01-01 | Wyeth Corp | Piperazine-piperidine antagonists and agonists of the 5-HT1a receptor |
| BRPI0611948A2 (pt) * | 2005-06-17 | 2010-10-13 | Wyeth Corp | compostos úteis como inibidores de serotonina e agonistas de antagonista de 5-ht1a |
| CA2640569A1 (en) * | 2006-01-26 | 2007-08-09 | The University Of Rochester | Inhibiting amyloid-beta peptide/rage interaction at the blood-brain barrier |
| TW200808741A (en) * | 2006-06-09 | 2008-02-16 | Wyeth Corp | 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline hydrochloric acid salts |
| TW200811144A (en) * | 2006-06-09 | 2008-03-01 | Wyeth Corp | Crystalline forms of 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline |
| TW200808740A (en) * | 2006-06-09 | 2008-02-16 | Wyeth Corp | Succinate salts of 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline and crystalline forms thereof |
| CL2007003410A1 (es) * | 2006-11-28 | 2008-04-11 | Wyeth Corp | Compuestos derivados de 5-fluoro-8-{4-[4-(6-metoxiquinolin-8-il)piperazin-1-il]piperidin-1-il}quinolina; procedimiento de preparacion; compuestos intermediarios; procedimiento de preparacion; composicion farmaceutica; y uso en el tratamiento de trast |
| TW200901974A (en) * | 2007-01-16 | 2009-01-16 | Wyeth Corp | Compounds, compositions, and methods of making and using them |
| US8936787B2 (en) * | 2008-04-15 | 2015-01-20 | The United States Of America As Represented By The Secretary, Department Of Health And Human Services | Peptides promoting lipid efflux |
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| MX9201991A (es) | 1991-05-02 | 1992-11-01 | Jonh Wyeth & Brother Limited | Derivados de piperazina y procedimiento para su preparacion. |
| GB9514901D0 (en) | 1995-07-20 | 1995-09-20 | American Home Prod | Piperazine derivatives |
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2001
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- 2001-11-27 AT AT01986458T patent/ATE269078T1/de not_active IP Right Cessation
- 2001-11-27 JP JP2002546512A patent/JP4198989B2/ja not_active Expired - Fee Related
- 2001-11-27 TW TW090129285A patent/TWI224102B/zh not_active IP Right Cessation
- 2001-11-27 BR BR0115609-8A patent/BR0115609A/pt not_active Application Discontinuation
- 2001-11-27 EA EA200300619A patent/EA005925B1/ru not_active IP Right Cessation
- 2001-11-27 CA CA2428039A patent/CA2428039C/en not_active Expired - Fee Related
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2002
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2003
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- 2003-05-27 NO NO20032390A patent/NO325501B1/no not_active IP Right Cessation
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