NO328077B1 - Anvendelse av en eksendin eller eksendinagonist for fremstilling av en farmasoytisk formulering. - Google Patents

Anvendelse av en eksendin eller eksendinagonist for fremstilling av en farmasoytisk formulering. Download PDF

Info

Publication number: NO328077B1
Authority: NO; Norway
Prior art keywords: exendin; agonist; compounds; glucagon; peptide
Prior art date: 1999-01-14

Application number

NO20013469A

Other languages

English (en)

Norwegian (no)

Other versions

NO20013469L (no

NO20013469D0 (no

Inventor

Andrew Young

Bronislava Gedulin

Original Assignee

Amylin Pharmaceuticals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-14

Filing date

2001-07-12

Publication date

2009-11-23

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27381821&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO328077(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2001-07-12 Application filed by Amylin Pharmaceuticals Inc filed Critical Amylin Pharmaceuticals Inc

2001-07-12 Publication of NO20013469D0 publication Critical patent/NO20013469D0/no

2001-09-14 Publication of NO20013469L publication Critical patent/NO20013469L/no

2009-11-23 Publication of NO328077B1 publication Critical patent/NO328077B1/no

Links

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Classifications

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- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/57563—Vasoactive intestinal peptide [VIP]; Related peptides
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A—HUMAN NECESSITIES
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Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Zoology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Gastroenterology & Hepatology (AREA)
Hematology (AREA)
Obesity (AREA)
Vascular Medicine (AREA)
Toxicology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Emergency Medicine (AREA)
Dermatology (AREA)
Immunology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)

NO20013469A 1999-01-14 2001-07-12 Anvendelse av en eksendin eller eksendinagonist for fremstilling av en farmasoytisk formulering. NO328077B1 (no)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US11638099P	1999-01-14	1999-01-14
US13201799P	1999-04-30	1999-04-30
US17536500P	2000-01-10	2000-01-10
PCT/US2000/000942 WO2000041548A2 (fr)	1999-01-14	2000-01-14	Methodes de suppression du glucagon

Publications (3)

Publication Number	Publication Date
NO20013469D0 NO20013469D0 (no)	2001-07-12
NO20013469L NO20013469L (no)	2001-09-14
NO328077B1 true NO328077B1 (no)	2009-11-23

Family

ID=27381821

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
NO20013469A NO328077B1 (no)	1999-01-14	2001-07-12	Anvendelse av en eksendin eller eksendinagonist for fremstilling av en farmasoytisk formulering.
NO2010010C NO2010010I1 (no)	1999-01-14	2010-05-11	Exendin-4 (Exenatid)
NO2010012C NO2010012I1 (no)	1999-01-14	2010-05-20	Exennatid (Eksenatid)

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
NO2010010C NO2010010I1 (no)	1999-01-14	2010-05-11	Exendin-4 (Exenatid)
NO2010012C NO2010012I1 (no)	1999-01-14	2010-05-20	Exennatid (Eksenatid)

Country Status (18)

Country	Link
US (3)	US6872700B1 (fr)
EP (2)	EP1143989B1 (fr)
JP (1)	JP2002538084A (fr)
KR (2)	KR20070051948A (fr)
CN (1)	CN100425284C (fr)
AT (2)	ATE460942T1 (fr)
AU (2)	AU770712B2 (fr)
BR (1)	BRPI0007823A8 (fr)
CA (1)	CA2356331C (fr)
CY (1)	CY1106347T1 (fr)
DE (2)	DE60032331T2 (fr)
DK (1)	DK1143989T3 (fr)
ES (2)	ES2278589T3 (fr)
HK (1)	HK1046105A1 (fr)
NO (3)	NO328077B1 (fr)
NZ (1)	NZ512657A (fr)
PT (1)	PT1143989E (fr)
WO (1)	WO2000041548A2 (fr)

Families Citing this family (114)

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Publication number	Priority date	Publication date	Assignee	Title
ATE493998T1 (de) *	1996-08-08	2011-01-15	Amylin Pharmaceuticals Inc	Pharmazeutische zusammensetzung mit einem exendin-4-peptid
KR100637433B1 (ko) *	2004-05-24	2006-10-20	삼성에스디아이 주식회사	발광 표시 장치
US6703359B1 (en) *	1998-02-13	2004-03-09	Amylin Pharmaceuticals, Inc.	Inotropic and diuretic effects of exendin and GLP-1
US20030087820A1 (en) *	1999-01-14	2003-05-08	Young Andrew A.	Novel exendin agonist formulations and methods of administration thereof
ES2278589T3 (es)	1999-01-14	2007-08-16	Amylin Pharmaceuticals, Inc.	Excendinas destinadas a la inhibicion de glucagon.
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2000
- 2000-01-14 ES ES00902415T patent/ES2278589T3/es not_active Expired - Lifetime
- 2000-01-14 KR KR1020077009281A patent/KR20070051948A/ko not_active Ceased
- 2000-01-14 DE DE60032331T patent/DE60032331T2/de not_active Expired - Lifetime
- 2000-01-14 AU AU24136/00A patent/AU770712B2/en not_active Expired
- 2000-01-14 CA CA002356331A patent/CA2356331C/fr not_active Expired - Lifetime
- 2000-01-14 EP EP00902415A patent/EP1143989B1/fr not_active Expired - Lifetime
- 2000-01-14 DE DE60044041T patent/DE60044041D1/de not_active Expired - Lifetime
- 2000-01-14 US US09/889,331 patent/US6872700B1/en not_active Expired - Lifetime
- 2000-01-14 BR BRPI0007823A patent/BRPI0007823A8/pt not_active Application Discontinuation
- 2000-01-14 HK HK02107813.8A patent/HK1046105A1/zh unknown
- 2000-01-14 EP EP06002683A patent/EP1658856B1/fr not_active Expired - Lifetime
- 2000-01-14 WO PCT/US2000/000942 patent/WO2000041548A2/fr not_active Ceased
- 2000-01-14 AT AT06002683T patent/ATE460942T1/de not_active IP Right Cessation
- 2000-01-14 AT AT00902415T patent/ATE347901T1/de active
- 2000-01-14 PT PT00902415T patent/PT1143989E/pt unknown
- 2000-01-14 CN CNB008050171A patent/CN100425284C/zh not_active Expired - Lifetime
- 2000-01-14 NZ NZ512657A patent/NZ512657A/xx not_active IP Right Cessation
- 2000-01-14 JP JP2000593169A patent/JP2002538084A/ja active Pending
- 2000-01-14 KR KR1020017008892A patent/KR20020001719A/ko not_active Ceased
- 2000-01-14 ES ES06002683T patent/ES2343072T3/es not_active Expired - Lifetime
- 2000-01-14 DK DK00902415T patent/DK1143989T3/da active
2001
- 2001-07-12 NO NO20013469A patent/NO328077B1/no not_active IP Right Cessation
2004
- 2004-05-26 AU AU2004202293A patent/AU2004202293B2/en not_active Expired
2005
- 2005-03-18 US US11/083,730 patent/US7153825B2/en not_active Expired - Lifetime
2006
- 2006-10-19 US US11/584,114 patent/US7407932B2/en not_active Expired - Fee Related
2007
- 2007-03-01 CY CY20071100286T patent/CY1106347T1/el unknown
2010
- 2010-05-11 NO NO2010010C patent/NO2010010I1/no not_active Application Discontinuation
- 2010-05-20 NO NO2010012C patent/NO2010012I1/no unknown

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Also Published As

Publication number	Publication date
CY1106347T1 (el)	2011-10-12
ES2343072T3 (es)	2010-07-22
US20070037750A1 (en)	2007-02-15
KR20070051948A (ko)	2007-05-18
DE60032331D1 (de)	2007-01-25
BRPI0007823A8 (pt)	2017-03-21
NZ512657A (en)	2004-01-30
PT1143989E (pt)	2007-03-30
KR20020001719A (ko)	2002-01-09
CN1347327A (zh)	2002-05-01
EP1143989A3 (fr)	2002-09-11
CN100425284C (zh)	2008-10-15
HK1046105A1 (zh)	2002-12-27
ES2278589T3 (es)	2007-08-16
AU2413600A (en)	2000-08-01
EP1658856B1 (fr)	2010-03-17
AU770712B2 (en)	2004-02-26
EP1143989B1 (fr)	2006-12-13
AU2004202293A1 (en)	2004-06-17
DK1143989T3 (da)	2007-04-16
US7407932B2 (en)	2008-08-05
ATE460942T1 (de)	2010-04-15
EP1658856A1 (fr)	2006-05-24
NO2010010I1 (no)	2010-06-07
JP2002538084A (ja)	2002-11-12
NO20013469L (no)	2001-09-14
US7153825B2 (en)	2006-12-26
WO2000041548A2 (fr)	2000-07-20
WO2000041548A3 (fr)	2001-11-29
EP1143989A2 (fr)	2001-10-17
DE60032331T2 (de)	2007-06-21
AU2004202293B2 (en)	2007-09-20
CA2356331C (fr)	2009-10-13
DE60044041D1 (de)	2010-04-29
BR0007823A (pt)	2001-11-20
ATE347901T1 (de)	2007-01-15
NO20013469D0 (no)	2001-07-12
CA2356331A1 (fr)	2000-07-20
US6872700B1 (en)	2005-03-29
NO2010012I1 (no)	2010-06-07
US20050171019A1 (en)	2005-08-04

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2010-06-07	SPCF	Filing of supplementary protection certificate	Free format text: PRODUCT NAME: BYETTA; NAT. REG. NO/DATE: EU/1/06/362/001-004/NO 20061120; FIRST REG. NO/DATE: EU , EU/1/06/362/001-004 20061120 Spc suppl protection certif: 2010010 Filing date: 20100511 Free format text: PRODUCT NAME: BYETTA; NAT. REG. NO/DATE: EU/1/06/362/001-4/NO 20061120; FIRST REG. NO/DATE: EU/1/06/362/001-004 20061120 Spc suppl protection certif: 2010012 Filing date: 20100520
2013-03-04	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: ASTRAZENECA PHARMACEUTICALS LP, US
2018-02-26	CHAD	Change of the owner's name or address (par. 44 patent law, par. patentforskriften)	Owner name: ASTRAZENECA PHARMACEUTICALS LP, US
2020-02-10	MK1K	Patent expired

Publication	Publication Date	Title
EP1143989B1 (fr)	2006-12-13	Exendines destines a la suppression du glucagon
US7399489B2 (en)	2008-07-15	Exendin analog formulations
AU775063C (en)	2005-05-12	Modified exendins and exendin agonists
US8445647B2 (en)	2013-05-21	Modified exendins and exendin agonists
EP1032587A1 (fr)	2000-09-06	Nouveaux composes agonistes de l'exendine
AU8772998A (en)	1999-03-01	Novel exendin agonist compounds
EP1938830A1 (fr)	2008-07-02	Nouveaux composants d'agoniste d'exendine