NO329206B1 - Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. - Google Patents

Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. Download PDF

Info

Publication number
NO329206B1
NO329206B1 NO20002526A NO20002526A NO329206B1 NO 329206 B1 NO329206 B1 NO 329206B1 NO 20002526 A NO20002526 A NO 20002526A NO 20002526 A NO20002526 A NO 20002526A NO 329206 B1 NO329206 B1 NO 329206B1
Authority
NO
Norway
Prior art keywords
drug content
preparation
high drug
methylene
methyl
Prior art date
Application number
NO20002526A
Other languages
English (en)
Norwegian (no)
Other versions
NO20002526L (no
NO20002526D0 (no
Inventor
Gopadi M Venkatesh
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of NO20002526L publication Critical patent/NO20002526L/no
Publication of NO20002526D0 publication Critical patent/NO20002526D0/no
Publication of NO329206B1 publication Critical patent/NO329206B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
NO20002526A 1997-11-17 2000-05-16 Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat. NO329206B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6591897P 1997-11-17 1997-11-17
PCT/US1998/024502 WO1999025321A1 (fr) 1997-11-17 1998-11-17 Formes posologiques orales a forte dose medicamenteuse et a liberation immediate et modifiee et leurs procedes de fabrication

Publications (3)

Publication Number Publication Date
NO20002526L NO20002526L (no) 2000-05-16
NO20002526D0 NO20002526D0 (no) 2000-05-16
NO329206B1 true NO329206B1 (no) 2010-09-13

Family

ID=22066009

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20002526A NO329206B1 (no) 1997-11-17 2000-05-16 Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat.

Country Status (14)

Country Link
EP (1) EP1033974B1 (fr)
JP (1) JP4880118B2 (fr)
KR (1) KR100597922B1 (fr)
CN (1) CN1285739A (fr)
AU (1) AU750611B2 (fr)
BR (1) BR9814877A (fr)
CA (1) CA2310028C (fr)
HU (1) HUP0004407A3 (fr)
IL (1) IL136142A0 (fr)
NO (1) NO329206B1 (fr)
NZ (1) NZ504565A (fr)
PL (1) PL340587A1 (fr)
TR (1) TR200001412T2 (fr)
WO (1) WO1999025321A1 (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ509378A (en) * 1998-07-20 2003-04-29 Smithkline Beecham Corp Amorphous ammonium salts of eprosartan and pharmaceuticals thereof, useful for blocking angiotensin II receptors and useful for treating hypertension, congestive heart disease and renal failure
HK1050135A1 (zh) 1999-11-02 2003-06-13 Depomed, Inc. 用於促进将药物给予胃的饭後模式药理学诱导
GB0209265D0 (en) 2002-04-23 2002-06-05 Novartis Ag Organic compounds
GB0228878D0 (en) * 2002-06-21 2003-01-15 Unilever Plc Hair conditioning composition
KR20120058618A (ko) 2003-01-31 2012-06-07 다이이찌 산쿄 가부시키가이샤 동맥 경화 및 고혈압증의 예방 및 치료를 위한 의약
EP2382975A3 (fr) * 2006-05-09 2012-02-29 Braincells, Inc. Neurogénèse par modulation d'angiotensine
NZ584686A (en) * 2007-11-06 2013-03-28 Novartis Ag Compositions of trisodium [3-((1S,3R)-1-biphenyl-4-ylmethyl-3-ethoxycarbonyl-1-butylcarbamoyl) propionate(S)-3'-methyl-2' -(pentanoyl{ 2 -(tetrazol-5-ylate)biphenyl-4'-ylmethyl} amino)butyrate]hemipentahydrate
AR072477A1 (es) * 2008-07-11 2010-09-01 Solvay Pharm Bv Formulacion farmaceutica de eprosartan. uso.
JP5476782B2 (ja) * 2009-04-21 2014-04-23 大正製薬株式会社 アルギニン含有錠剤の製造方法
JP5446716B2 (ja) * 2009-10-21 2014-03-19 大正製薬株式会社 アルギニン及びカルニチン含有錠剤の製造方法
TR201007508A1 (tr) * 2010-09-14 2012-04-24 Sanovel İlaç San. Ve Ti̇c. A.Ş. Oral yolla dağılan bileşimler
CN104546779A (zh) * 2013-10-14 2015-04-29 深圳海王药业有限公司 高药物荷载的枸橼酸西地那非片剂及其制备方法
US11510877B2 (en) 2017-10-10 2022-11-29 Capsugel Belgium Nv Gelling multiparticulates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5185351A (en) * 1989-06-14 1993-02-09 Smithkline Beecham Corporation Imidazolyl-alkenoic acids useful as angiotensin II receptor antagonists
JP3214856B2 (ja) * 1990-12-14 2001-10-02 スミスクライン・ビーチャム・コーポレイション イミダゾリル−アルケン酸
AU7475694A (en) * 1993-08-02 1995-02-28 Prizm Pharmaceuticals, Inc. Monogenous preparations of cytotoxic conjugates
BR9708336A (pt) * 1996-03-29 1999-08-03 Smithkline Beecham Corp Diidrato de eprosartan e processo para sua produção e formulação

Also Published As

Publication number Publication date
HUP0004407A1 (hu) 2002-02-28
WO1999025321A1 (fr) 1999-05-27
EP1033974A1 (fr) 2000-09-13
EP1033974A4 (fr) 2007-05-02
NO20002526L (no) 2000-05-16
CA2310028C (fr) 2008-06-10
IL136142A0 (en) 2001-05-20
PL340587A1 (en) 2001-02-12
TR200001412T2 (tr) 2000-09-21
JP4880118B2 (ja) 2012-02-22
CN1285739A (zh) 2001-02-28
BR9814877A (pt) 2000-10-03
AU1588799A (en) 1999-06-07
HUP0004407A3 (en) 2002-03-28
NO20002526D0 (no) 2000-05-16
JP2001522872A (ja) 2001-11-20
KR20010032129A (ko) 2001-04-16
AU750611B2 (en) 2002-07-25
CA2310028A1 (fr) 1999-05-27
EP1033974B1 (fr) 2014-01-22
NZ504565A (en) 2002-11-26
KR100597922B1 (ko) 2006-07-10

Similar Documents

Publication Publication Date Title
KR100634953B1 (ko) 에프로사르탄을 포함하는 생물학적으로 강화된 경구 고형투여 형태의 제제
US6558699B2 (en) High drug load immediate and modified release oral dosage formulations and processes for their manufacture
US6630498B2 (en) Eprosartan arginyl charge-neutralization-complex and a process for its preparation and formulation
NO329206B1 (no) Granulering og preparat med hoyt legemiddelinnhold, fremgangsmate for fremstilling derav og farmasoytisk preparat.
KR101778050B1 (ko) 칼슘 길항약／안지오텐신 ｉｉ 수용체 길항약 함유 의약 제제의 제조 방법
JP4463975B2 (ja) エプロサルタン・アルギニル電荷中和複合体およびその製造方法および処方
CZ20001802A3 (cs) Orální dávkové prostředky s okamžitým nebo modifikovaným uvolňováním vysoké náplně léčiva a způsoby jejich přípravy
MXPA00004791A (en) High drug load immediate and modified release oral dosage formulations and processes for their manufacture
CZ2001227A3 (cs) Biologicky zlepšené prostředky obsahující eprosartan v orální pevné dávkové formě
HK1031688B (en) Eprosartan arginyl charge-neutralization-complex and a process for its production and formulation
MXPA00001385A (en) Eprosartan arginyl charge-neutralization-complex and a process for its production and formulation

Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees