NO772493L - 5- (2-FUROYL) -, 5- (2-THENOYL) -, 5- (3-FUROYL) -OG 5- (3-THENOYL) -1,2-DIHYDRO-3H-PYRROLO (1,2-A ) PYRROL-1-CARBOXYLIC ACID DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION. - Google Patents

5- (2-FUROYL) -, 5- (2-THENOYL) -, 5- (3-FUROYL) -OG 5- (3-THENOYL) -1,2-DIHYDRO-3H-PYRROLO (1,2-A ) PYRROL-1-CARBOXYLIC ACID DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION.

Info

Publication number: NO772493L
Authority: NO; Norway
Prior art keywords: thenoyl; furoyl; pyrrol; pyrrolo; dihydro
Prior art date: 1976-07-14

Application number

NO772493A

Other languages

Norwegian (no)

Other versions

NO147563B (en

NO147563C (en

Inventor

Joseph M Muchowski

Arthur F Kluge

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1977-07-13

Publication date

1978-01-17

1977-02-23 Priority claimed from US05/771,283 external-priority patent/US4087539A/en

1977-07-13 Application filed by Syntex Inc filed Critical Syntex Inc

1978-01-17 Publication of NO772493L publication Critical patent/NO772493L/en

1983-01-24 Publication of NO147563B publication Critical patent/NO147563B/en

1983-05-18 Publication of NO147563C publication Critical patent/NO147563C/en

Links

-1 3-FUROYL Chemical class 0.000 title 1
QXJGPMJZRCHZPM-UHFFFAOYSA-N 5-(thiophene-3-carbonyl)-2,3-dihydro-1h-pyrrolizine-1-carboxylic acid Chemical class OC(=O)C1CCN2C1=CC=C2C(=O)C=1C=CSC=1 QXJGPMJZRCHZPM-UHFFFAOYSA-N 0.000 title 1
238000000034 method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

NO772493A 1976-07-14 1977-07-13 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVITY 5- (2-FUROYL, 5- (2-TENOYL) -, 5- (3-FUROYL) - AND 5- (3-TENOYL) -1,2-DIHYDRO-3H-PYRROLO ( 1,2-A) pyrrole-1-carboxylic acid derivatives NO147563C (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70485776A	1976-07-14	1976-07-14
US05/771,283 US4087539A (en)	1976-07-14	1977-02-23	5-(2-Furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- and 5-(3-thenoyl)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (3)

Publication Number	Publication Date
NO772493L true NO772493L (en)	1978-01-17
NO147563B NO147563B (en)	1983-01-24
NO147563C NO147563C (en)	1983-05-18

Family

ID=27107392

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO772493A NO147563C (en)	1976-07-14	1977-07-13	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVITY 5- (2-FUROYL, 5- (2-TENOYL) -, 5- (3-FUROYL) - AND 5- (3-TENOYL) -1,2-DIHYDRO-3H-PYRROLO ( 1,2-A) pyrrole-1-carboxylic acid derivatives

Country Status (26)

Country	Link
JP (1)	JPS539789A (en)
AR (1)	AR218631A1 (en)
AU (1)	AU513385B2 (en)
CA (1)	CA1100140A (en)
CH (2)	CH651045A5 (en)
CS (1)	CS208724B2 (en)
DE (1)	DE2731662A1 (en)
DK (1)	DK152652C (en)
ES (2)	ES460705A1 (en)
FI (1)	FI63407C (en)
FR (1)	FR2361396A1 (en)
GB (1)	GB1554076A (en)
GR (1)	GR61607B (en)
HK (1)	HK17581A (en)
IE (1)	IE45302B1 (en)
IL (1)	IL52492A (en)
IT (1)	IT1117314B (en)
MY (1)	MY8100371A (en)
NL (1)	NL7707652A (en)
NO (1)	NO147563C (en)
NZ (1)	NZ184611A (en)
PL (1)	PL111408B1 (en)
PT (1)	PT66779B (en)
SE (1)	SE434644B (en)
SU (2)	SU664566A3 (en)
YU (2)	YU43156B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4097579A (en) *	1977-03-31	1978-06-27	Syntex (U.S.A.) Inc.	5-(2-Pyrroyl)-1,2-dihydro-3H-pyrrolo 1,2-a!pyrrole-1-carboxylic acid derivatives and process for the production thereof
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (en) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
HU198927B (en) *	1987-01-14	1989-12-28	Richter Gedeon Vegyeszet	Process for producing 1-/substituted aminomethyl/-octa-hydroindolo-(2,3-a)quinolizine derivatives, pharmaceutically applicable acid addition salts thereof, as well as pharmaceutical compositions comprising same
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds

1977
- 1977-05-17 JP JP5697877A patent/JPS539789A/en active Granted
- 1977-07-07 DK DK307677A patent/DK152652C/en not_active IP Right Cessation
- 1977-07-07 AR AR268357A patent/AR218631A1/en active
- 1977-07-07 GR GR53906A patent/GR61607B/en unknown
- 1977-07-08 CH CH4005/84A patent/CH651045A5/en not_active IP Right Cessation
- 1977-07-08 IL IL52492A patent/IL52492A/en unknown
- 1977-07-08 IE IE1422/77A patent/IE45302B1/en unknown
- 1977-07-08 NL NL7707652A patent/NL7707652A/en not_active Application Discontinuation
- 1977-07-08 CH CH848877A patent/CH644861A5/en not_active IP Right Cessation
- 1977-07-08 PT PT66779A patent/PT66779B/en unknown
- 1977-07-11 FI FI772154A patent/FI63407C/en not_active IP Right Cessation
- 1977-07-11 NZ NZ184611A patent/NZ184611A/en unknown
- 1977-07-11 GB GB28923/77A patent/GB1554076A/en not_active Expired
- 1977-07-12 CS CS774647A patent/CS208724B2/en unknown
- 1977-07-12 CA CA282,600A patent/CA1100140A/en not_active Expired
- 1977-07-12 FR FR7721559A patent/FR2361396A1/en active Granted
- 1977-07-13 SE SE7708142A patent/SE434644B/en not_active IP Right Cessation
- 1977-07-13 NO NO772493A patent/NO147563C/en unknown
- 1977-07-13 PL PL1977199602A patent/PL111408B1/en unknown
- 1977-07-13 SU SU772504151A patent/SU664566A3/en active
- 1977-07-13 ES ES460705A patent/ES460705A1/en not_active Expired
- 1977-07-13 AU AU26976/77A patent/AU513385B2/en not_active Expired
- 1977-07-13 DE DE19772731662 patent/DE2731662A1/en active Granted
- 1977-07-13 IT IT68631/77A patent/IT1117314B/en active
- 1977-12-29 SU SU772558960A patent/SU793400A3/en active
1978
- 1978-05-24 ES ES470213A patent/ES470213A1/en not_active Expired
1981
- 1981-04-30 HK HK175/81A patent/HK17581A/en unknown
- 1981-12-30 MY MY371/81A patent/MY8100371A/en unknown
1983
- 1983-02-28 YU YU475/83A patent/YU43156B/en unknown
- 1983-02-28 YU YU476/83A patent/YU43157B/en unknown

Also Published As

Publication number	Publication date
SE7708142L (en)	1978-01-15
AR218631A1 (en)	1980-06-30
CH644861A5 (en)	1984-08-31
GR61607B (en)	1978-12-02
YU43157B (en)	1989-04-30
CA1100140A (en)	1981-04-28
DE2731662A1 (en)	1978-01-19
FI63407B (en)	1983-02-28
HK17581A (en)	1981-05-08
GB1554076A (en)	1979-10-17
FR2361396B1 (en)	1981-11-27
NZ184611A (en)	1979-03-28
SU664566A3 (en)	1979-05-25
SU793400A3 (en)	1980-12-30
IE45302L (en)	1978-01-14
PT66779A (en)	1977-08-01
FR2361396A1 (en)	1978-03-10
ES460705A1 (en)	1979-10-01
JPS539789A (en)	1978-01-28
PL199602A1 (en)	1979-01-29
FI772154A7 (en)	1978-01-15
MY8100371A (en)	1981-12-31
SE434644B (en)	1984-08-06
YU43156B (en)	1989-04-30
IL52492A0 (en)	1977-10-31
ES470213A1 (en)	1979-09-16
IE45302B1 (en)	1982-07-28
CS208724B2 (en)	1981-09-15
AU2697677A (en)	1979-01-18
DK152652C (en)	1988-09-12
DK152652B (en)	1988-04-05
IT1117314B (en)	1986-02-17
PT66779B (en)	1978-12-18
YU47683A (en)	1984-04-30
YU47583A (en)	1984-06-30
FI63407C (en)	1983-06-10
AU513385B2 (en)	1980-11-27
DK307677A (en)	1978-01-15
NO147563B (en)	1983-01-24
IL52492A (en)	1981-06-29
CH651045A5 (en)	1985-08-30
NO147563C (en)	1983-05-18
PL111408B1 (en)	1980-08-30
NL7707652A (en)	1978-01-17
JPS6254110B2 (en)	1987-11-13
DE2731662C2 (en)	1989-11-09

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