NO800501L - ANTIBACTERIAL AND BETA-LACTAMA INHIBITORS AND PROCEDURE FOR THEIR PREPARATION - Google Patents

ANTIBACTERIAL AND BETA-LACTAMA INHIBITORS AND PROCEDURE FOR THEIR PREPARATION

Info

Publication number
NO800501L
NO800501L NO800501A NO800501A NO800501L NO 800501 L NO800501 L NO 800501L NO 800501 A NO800501 A NO 800501A NO 800501 A NO800501 A NO 800501A NO 800501 L NO800501 L NO 800501L
Authority
NO
Norway
Prior art keywords
lactama
antibacterial
inhibitors
beta
procedure
Prior art date
Application number
NO800501A
Other languages
Norwegian (no)
Other versions
NO161000B (en
NO161000C (en
Inventor
Maurizio Foglio
Giovanni Franceschi
Cosimo Scarafile
Federico Arcamone
Aurora Sanfilippo
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NO800501L publication Critical patent/NO800501L/en
Publication of NO161000B publication Critical patent/NO161000B/en
Publication of NO161000C publication Critical patent/NO161000C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568—Four-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
NO800501A 1979-02-24 1980-02-22 ANALOGUE PROCEDURE FOR PREPARING A THERAPEUTIC ACTIVE PENEMKARBOXYLIC ACID OR ESTER. NO161000C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7906634 1979-02-24
GB7932591 1979-09-20

Publications (3)

Publication Number Publication Date
NO800501L true NO800501L (en) 1980-08-25
NO161000B NO161000B (en) 1989-03-13
NO161000C NO161000C (en) 1989-06-21

Family

ID=26270697

Family Applications (1)

Application Number Title Priority Date Filing Date
NO800501A NO161000C (en) 1979-02-24 1980-02-22 ANALOGUE PROCEDURE FOR PREPARING A THERAPEUTIC ACTIVE PENEMKARBOXYLIC ACID OR ESTER.

Country Status (24)

Country Link
AT (1) AT368506B (en)
AU (1) AU535080B2 (en)
CA (2) CA1154010A (en)
CH (2) CH654831A5 (en)
CS (1) CS226010B2 (en)
DE (1) DE3006273A1 (en)
DK (1) DK159448C (en)
ES (2) ES8200685A1 (en)
FI (1) FI75163C (en)
FR (1) FR2449690B1 (en)
GB (1) GB2043639B (en)
GR (1) GR73623B (en)
HK (1) HK74487A (en)
HU (1) HU182664B (en)
IE (1) IE49407B1 (en)
IT (1) IT1193922B (en)
LU (1) LU82192A1 (en)
NL (1) NL192265C (en)
NO (1) NO161000C (en)
NZ (1) NZ192949A (en)
PT (1) PT70849A (en)
SE (1) SE449489B (en)
UA (1) UA6041A1 (en)
YU (1) YU42964B (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
DE3121510A1 (en) * 1980-07-04 1982-06-16 Farmitalia Carlo Erba S.p.A., 20159 Milano 6-Alkyl-2-subst. penems and process for their preparation
JPS588084A (en) * 1981-07-08 1983-01-18 Takeda Chem Ind Ltd (6r)-substituted-(5r)-penem-3-carboxylic acid derivative and its preparation
DE3277696D1 (en) * 1981-07-15 1987-12-23 Sumitomo Pharma Carboxylic beta-lactam compounds and the preparation thereof
US4508649A (en) * 1981-12-11 1985-04-02 Farmitalia Carlo Erba Process for preparing optically active penems
NO831160L (en) * 1982-04-08 1983-10-10 Erba Farmitalia PREPARATION OF SUBSTITUTED PENEM DERIVATIVES
PH21930A (en) * 1982-11-16 1988-04-08 Ciba Geigy Ag 6-hydroxy-lower alkylpenem compounds,pharmaceutical composition containing same and method of use thereof
EP0112283B1 (en) * 1982-11-16 1987-08-12 Ciba-Geigy Ag Heterocyclyl-thio compounds, process for their preparation, pharmaceutical compositions containing them and their use
GB8300295D0 (en) * 1983-01-06 1983-02-09 Erba Farmitalia Penem esters
JPS59152387A (en) * 1983-02-10 1984-08-31 Shionogi & Co Ltd Novel penem compound
GB8321677D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia Preparation of penems
US4656165A (en) * 1983-09-02 1987-04-07 Ciba-Geigy Corporation Aminomethyl penem compounds
US4711886A (en) * 1984-07-02 1987-12-08 Merck & Co., Inc. β-lactam derivatives as anti-inflammatory and antidegenerative agents
US4761408A (en) * 1984-11-02 1988-08-02 Ciba-Geigy Corporation Crystalline aminomethyl compound
EP0278911B1 (en) * 1987-02-11 1993-08-04 Ciba-Geigy Ag Bicyclic beta-lactam carboxylic acids
GB2206578B (en) * 1987-07-07 1991-07-03 Erba Carlo Spa Process for the preparation of penems
US5364768A (en) * 1987-07-07 1994-11-15 Farmitalia Carlo Erba S.R.L. Process for the preparation of penems
IT1286558B1 (en) * 1996-02-27 1998-07-15 Menarini Farma Ind PROCESS FOR THE PREPARATION OF 2-HALOGENOMETHYL-PENEMS AND THEIR USE FOR THE PREPARATION OF ANTIBACTERIAL PENEMS
US6156745A (en) 1997-12-29 2000-12-05 Research Corporation Technologies, Inc. 2β-substituted-6-alkylidene penicillanic acid derivatives as β-lactamase inhibitors
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
US6720445B2 (en) * 2000-12-21 2004-04-13 Beacon Laboratories, Inc. Acetyloxymethyl esters and methods for using the same
ATE339424T1 (en) 2001-07-24 2006-10-15 Univ Southern Methodist 3-SUBSTITUTED 7-ALKYLIDENE-3-CEPHEM-4-CARBOXYLIC ACIDS AS BETA-LACTAMASE INHIBITORS
AU2003224874A1 (en) 2002-04-04 2003-10-27 Alamx, L.L.C. INHIBITORS OF SERINE AND METALLO-ss-LACTAMASES

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU77306A1 (en) * 1977-05-09 1979-01-18
AU3796278A (en) * 1977-07-13 1980-01-17 Glaxo Group Ltd Penams and azetidinones
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4155912A (en) * 1977-12-14 1979-05-22 Bristol-Myers Company 2-Methylpenem-3-carboxylic acid antibiotics
JPS54117459A (en) * 1978-01-20 1979-09-12 Glaxo Group Ltd Novel lactam compound
EP0003960B1 (en) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-substituted thia-aza-compounds, their preparation and pharmaceutical compositions containing them
JPS5559193A (en) * 1978-09-20 1980-05-02 Glaxo Group Ltd Bblactam compound
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
EP0013067A1 (en) * 1978-12-22 1980-07-09 Beecham Group Plc Bicyclic beta-lactam antibacterial agents, their use in pharmaceutical compositions, processes for their preparation and intermediates for use in such processes

Also Published As

Publication number Publication date
FI800493A7 (en) 1980-08-25
NL192265B (en) 1996-12-02
FI75163B (en) 1988-01-29
IT1193922B (en) 1988-08-31
DE3006273A1 (en) 1980-09-04
NO161000B (en) 1989-03-13
IE800338L (en) 1980-08-24
GB2043639A (en) 1980-10-08
NL8001012A (en) 1980-08-26
UA6041A1 (en) 1994-12-29
DK159448B (en) 1990-10-15
HK74487A (en) 1987-10-23
GB2043639B (en) 1983-07-20
SE449489B (en) 1987-05-04
FR2449690B1 (en) 1986-06-13
CH654831A5 (en) 1986-03-14
LU82192A1 (en) 1980-06-06
NZ192949A (en) 1984-03-16
FR2449690A1 (en) 1980-09-19
AT368506B (en) 1982-10-25
NL192265C (en) 1997-04-03
NO161000C (en) 1989-06-21
SE8001424L (en) 1980-08-25
HU182664B (en) 1984-02-28
ES488886A0 (en) 1981-11-16
CH651570A5 (en) 1985-09-30
YU42964B (en) 1989-02-28
AU535080B2 (en) 1984-03-01
CA1154010A (en) 1983-09-20
AU5567080A (en) 1980-09-11
PT70849A (en) 1980-03-01
DK159448C (en) 1991-03-04
FI75163C (en) 1988-05-09
ES8107224A1 (en) 1981-10-01
DK77580A (en) 1980-08-25
GR73623B (en) 1984-03-26
ES495977A0 (en) 1981-10-01
IE49407B1 (en) 1985-10-02
ES8200685A1 (en) 1981-11-16
CA1212665B (en) 1986-10-14
CS226010B2 (en) 1984-03-19
YU46180A (en) 1983-02-28
IT8020021A0 (en) 1980-02-19
ATA91980A (en) 1982-02-15
IT8020021A1 (en) 1981-08-19

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