NO884467L - Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-cykloalkylbenzenderivater. - Google Patents

Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-cykloalkylbenzenderivater.

Info

Publication number: NO884467L
Authority: NO; Norway
Prior art keywords: aminomethyloxooxazolidinyl; cycloalkyl; preparation; analogy procedure; benzen
Prior art date: 1987-10-09

Application number

NO88884467A

Other languages

English (en)

Other versions

NO172890B (no

NO172890C (no

NO884467D0 (no

Inventor

Chia-Lin Jeffrey Wang

Mark Arvid Wuonola

Original Assignee

Du Pont

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-10-09

Filing date

1988-10-07

Publication date

1989-04-10

1988-10-07 Application filed by Du Pont filed Critical Du Pont

1988-10-07 Publication of NO884467D0 publication Critical patent/NO884467D0/no

1989-04-10 Publication of NO884467L publication Critical patent/NO884467L/no

1993-06-14 Publication of NO172890B publication Critical patent/NO172890B/no

1993-09-22 Publication of NO172890C publication Critical patent/NO172890C/no

Links

UHOVQNZJYSORNB-UHFFFAOYSA-N Benzene Chemical class C1=CC=CC=C1 UHOVQNZJYSORNB-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO884467A 1987-10-09 1988-10-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive aminomethyloxooxazolidinyl-cykloalkylbenzenderivater NO172890C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/106,358 US4801600A (en)	1987-10-09	1987-10-09	Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents

Publications (4)

Publication Number	Publication Date
NO884467D0 NO884467D0 (no)	1988-10-07
NO884467L true NO884467L (no)	1989-04-10
NO172890B NO172890B (no)	1993-06-14
NO172890C NO172890C (no)	1993-09-22

Family

ID=22310972

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO884467A NO172890C (no)	1987-10-09	1988-10-07	Analogifremgangsmaate for fremstilling av terapeutisk aktive aminomethyloxooxazolidinyl-cykloalkylbenzenderivater

Country Status (16)

Country	Link
US (1)	US4801600A (no)
EP (1)	EP0311090A1 (no)
JP (1)	JPH01132569A (no)
KR (1)	KR890006632A (no)
AU (1)	AU613669B2 (no)
CA (1)	CA1322001C (no)
DK (1)	DK562888A (no)
FI (1)	FI884610A7 (no)
HU (1)	HU202216B (no)
IL (1)	IL87972A (no)
MY (1)	MY103618A (no)
NO (1)	NO172890C (no)
NZ (1)	NZ226493A (no)
PT (1)	PT88713B (no)
SU (1)	SU1616518A3 (no)
ZA (1)	ZA887550B (no)

Families Citing this family (50)

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US4985429A (en) *	1987-10-09	1991-01-15	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4942183A (en) *	1987-10-16	1990-07-17	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A (en) *	1987-10-21	1990-12-11	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US4948801A (en) *	1988-07-29	1990-08-14	E. I. Du Pont De Nemours And Company	Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5182403A (en) *	1988-09-15	1993-01-26	The Upjohn Company	Substituted 3(5'indazolyl) oxazolidin-2-ones
US5164510A (en) *	1988-09-15	1992-11-17	The Upjohn Company	5'Indolinyl-5β-amidomethyloxazolidin-2-ones
US5225565A (en) *	1988-09-15	1993-07-06	The Upjohn Company	Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones
ATE112773T1 (de) *	1988-09-15	1994-10-15	Upjohn Co	5-indolinyl-5-beta-amidomethyloxazolidin-2-one, 3-(substituierte kondensierte)phenyl-5-beta amidomethyloxazolidin-2-one und 3-(nitrogen- substituierte)phenyl-5-beta-amidomethyloxazolid n-2-one.
US5231188A (en) *	1989-11-17	1993-07-27	The Upjohn Company	Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents
KR100215627B1 (ko) *	1990-06-07	1999-08-16	레슬리 제인 에드워즈	치료용 헤테로사이클 화합물
JP2669579B2 (ja) *	1991-10-23	1997-10-29	エーザイ株式会社	オキサゾリドン誘導体
AU667198B2 (en) *	1991-11-01	1996-03-14	Pharmacia & Upjohn Company	Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents
SK283420B6 (sk) *	1992-05-08	2003-07-01	Pharmacia & Upjohn Company	Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
JP3558088B2 (ja) *	1992-12-08	2004-08-25	ファルマシア・アンド・アップジョン・カンパニー	トロポン−置換のフェニルオキサゾリジノン抗菌剤
US5688792A (en) *	1994-08-16	1997-11-18	Pharmacia & Upjohn Company	Substituted oxazine and thiazine oxazolidinone antimicrobials
JP3698724B2 (ja) *	1993-11-22	2005-09-21	ファルマシア・アンド・アップジョン・カンパニー	置換−ヒドロキシアセチルピペラジンフェニルオキサゾリジノンのエステル
DE4425612A1 (de) *	1994-07-20	1996-04-04	Bayer Ag	6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
DE4425613A1 (de) *	1994-07-20	1996-01-25	Bayer Ag	5-gliedrige Heteroaryl-oxazolidinone
DE4425609A1 (de) *	1994-07-20	1996-01-25	Bayer Ag	Benzofuranyl- und Benzothienyloxazolidinone
DE19514313A1 (de)	1994-08-03	1996-02-08	Bayer Ag	Benzoxazolyl- und Benzothiazolyloxazolidinone
BR9509673A (pt) *	1994-11-15	1997-09-30	Upjohn Co	Compostos e uso dos mesmos
CA2208603A1 (en) *	1995-02-03	1996-08-08	The Upjohn Company	Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials
HRP960159A2 (en) *	1995-04-21	1997-08-31	Bayer Ag	Benzocyclopentane oxazolidinones containing heteroatoms
AU702752B2 (en) *	1995-05-11	1999-03-04	Pharmacia & Upjohn Company	Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones
US5883093A (en) *	1995-09-12	1999-03-16	Pharmacia & Upjohn Company	Phenyloxazolidinone antimicrobials
DE19601265A1 (de)	1996-01-16	1997-07-17	Bayer Ag	2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone
DE19601264A1 (de)	1996-01-16	1997-07-17	Bayer Ag	Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone
DE19601627A1 (de) *	1996-01-18	1997-07-24	Bayer Ag	Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone
DE19604223A1 (de) *	1996-02-06	1997-08-07	Bayer Ag	Neue substituierte Oxazolidinone
HRP970049A2 (en) *	1996-02-06	1998-04-30	Bayer Ag	New heteroaryl oxazolidinones
MY116093A (en) *	1996-02-26	2003-11-28	Upjohn Co	Azolyl piperazinyl phenyl oxazolidinone antimicrobials
US5998406A (en) *	1997-11-12	1999-12-07	Pharmacia & Upjohn Company	Oxazolidinone derivatives and pharmaceutical compositions
DE19802235A1 (de) *	1998-01-22	1999-07-29	Bayer Ag	Mit tricyclischen Indolen substituierte Oxazolidinone
WO1999037630A1 (en) *	1998-01-23	1999-07-29	Versicor, Inc.	Oxazolidinone combinatorial libraries, compositions and methods of preparation
EP1147422A1 (en)	1999-01-27	2001-10-24	Pharmacia & Upjohn Company	Assays for modulators of "elongation factor p" activity
JP2003501351A (ja) *	1999-05-27	2003-01-14	ファルマシア・アンド・アップジョン・カンパニー	抗菌剤としての二環系オキサゾリジノン
US6444813B2 (en) *	2000-02-02	2002-09-03	Pharmacia & Upjohn Company	Linezolid-crystal form II
WO2002006278A1 (en) *	2000-07-17	2002-01-24	Ranbaxy Laboratories Limited	Oxazolidinone derivatives as antimicrobials
PE20020689A1 (es) *	2000-11-17	2002-08-03	Upjohn Co	Oxazolidinonas con un heterociclo de 6 o 7 miembros unidos con enlace anular al benceno
ATE319710T1 (de)	2000-12-21	2006-03-15	Pharmacia & Upjohn Co Llc	Antimikrobielle chinolonderivate und ihre verwendung zur behandlung bakterieller infektionen
EP1409464A4 (en) *	2001-07-16	2005-11-02	Ranbaxy Lab Ltd	OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS
US6956040B2 (en)	2001-07-16	2005-10-18	Ranbaxy Laboratories Limited	Oxazolidinone piperazinyl derivatives as potential antimicrobials
BR0310074A (pt) *	2002-05-15	2005-03-08	Ranbaxy Lab Ltd	Formas polimórficas de derivados de fenil oxazolidinona
CN1668308A (zh) *	2002-07-29	2005-09-14	兰贝克赛实验室有限公司	作为抗菌剂的噁唑烷酮衍生物
EP1594494A1 (en) *	2003-02-07	2005-11-16	Warner-Lambert Company LLC	Oxazolidinone derivatives n-substituted by a bicyclic ring, for use as antibacterial agents
AU2003215861A1 (en) *	2003-04-07	2004-11-01	Ranbaxy Laboratories Limited	Oxazolidinone derivatives as antimicrobials
CA2602073A1 (en) *	2005-02-24	2006-08-31	Teva Pharmaceutical Industries Ltd.	Processes for the preparation of linezolid intermediate
US20100298384A1 (en) *	2006-12-04	2010-11-25	Mohamed Takhi	Novel oxazolidinone compounds as antiinfective agents
CN101965353B (zh) *	2008-03-26	2014-12-17	丹诺医药(苏州）有限公司	共价连接到取代苯基噁唑烷酮的双环硝基咪唑类
WO2020163689A1 (en)	2019-02-08	2020-08-13	University Of Pittsburgh - Of The Commonwealth System Of Higher Education	20-hete formation inhibitors

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US29607A (en) *		1860-08-14		Portable scaffold
GB1222708A (en) *	1968-10-22	1971-02-17	Delalande Sa	Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
USRE29607E (en)	1969-03-18	1978-04-11	Delalande S. A.	Derivatives of 5-hydroxymethyl-3-substituted-2-oxazolidinones, process of preparation thereof and therapeutic application
LU80081A1 (fr) *	1977-08-26	1979-05-15	Delalande Sa	Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique
US4128654A (en) *	1978-02-10	1978-12-05	E. I. Du Pont De Nemours And Company	5-Halomethyl-3-phenyl-2-oxazolidinones
CA1171865A (en) *	1980-06-04	1984-07-31	Alain Lacour	N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics
US4340606A (en) *	1980-10-23	1982-07-20	E. I. Du Pont De Nemours And Company	3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents
FR2500450A1 (fr) *	1981-02-25	1982-08-27	Delalande Sa	Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
US4461773A (en) *	1982-09-15	1984-07-24	E. I. Dupont De Nemours And Company	P-Oxooxazolidinylbenzene compounds as antibacterial agents
ES8506659A1 (es) *	1983-06-07	1985-08-01	Du Pont	Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno.
US4705799A (en) *	1983-06-07	1987-11-10	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
CA1260948A (en) *	1984-12-05	1989-09-26	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents

1987
- 1987-10-09 US US07/106,358 patent/US4801600A/en not_active Expired - Lifetime
1988
- 1988-10-04 CA CA000579301A patent/CA1322001C/en not_active Expired - Fee Related
- 1988-10-06 AU AU23507/88A patent/AU613669B2/en not_active Ceased
- 1988-10-06 SU SU884356653A patent/SU1616518A3/ru active
- 1988-10-07 DK DK562888A patent/DK562888A/da not_active Application Discontinuation
- 1988-10-07 ZA ZA887550A patent/ZA887550B/xx unknown
- 1988-10-07 MY MYPI88001123A patent/MY103618A/en unknown
- 1988-10-07 PT PT88713A patent/PT88713B/pt not_active IP Right Cessation
- 1988-10-07 JP JP63252207A patent/JPH01132569A/ja active Pending
- 1988-10-07 KR KR1019880013071A patent/KR890006632A/ko not_active Ceased
- 1988-10-07 EP EP88116621A patent/EP0311090A1/en not_active Withdrawn
- 1988-10-07 NO NO884467A patent/NO172890C/no unknown
- 1988-10-07 HU HU885214A patent/HU202216B/hu not_active IP Right Cessation
- 1988-10-07 FI FI884610A patent/FI884610A7/fi not_active Application Discontinuation
- 1988-10-07 IL IL87972A patent/IL87972A/xx unknown
- 1988-10-07 NZ NZ226493A patent/NZ226493A/xx unknown

Also Published As

Publication number	Publication date
HUT53359A (en)	1990-10-28
FI884610A7 (fi)	1989-04-10
SU1616518A3 (ru)	1990-12-23
DK562888D0 (da)	1988-10-07
HU202216B (en)	1991-02-28
DK562888A (da)	1989-04-10
FI884610A0 (fi)	1988-10-07
US4801600A (en)	1989-01-31
ZA887550B (en)	1990-06-27
IL87972A0 (en)	1989-03-31
EP0311090A1 (en)	1989-04-12
PT88713B (pt)	1992-12-31
AU613669B2 (en)	1991-08-08
NO172890B (no)	1993-06-14
NO172890C (no)	1993-09-22
AU2350788A (en)	1989-04-13
IL87972A (en)	1993-05-13
MY103618A (en)	1993-08-28
KR890006632A (ko)	1989-06-14
NO884467D0 (no)	1988-10-07
NZ226493A (en)	1990-09-26
JPH01132569A (ja)	1989-05-25
CA1322001C (en)	1993-09-07

Publication	Publication Date	Title
NO893076D0 (no)	1989-07-28	Fremgangsmaate for fremstilling av aminomethyloxooxa-zolidinylarylbenzenderivater.
NO884467D0 (no)	1988-10-07	Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-ycloalkylbenzenderivater.
NO870579L (no)	1987-08-17	Fremgangsmaate for fremstilling av indolizin-derivater.
NO842273L (no)	1984-12-10	Fremgangsmaate ved fremstilling av aminomethyloxooxazolidinylbenzenderivater.
NO892936L (no)	1990-01-19	Fremgangsmaate for fremstilling av furanderivater.
NO880910D0 (no)	1988-03-01	Fremgangsmaate for fremstilling av chromonderivater.
NO884900D0 (no)	1988-11-03	Fremgangsmaate for fremstilling av ginkolid-derivater.
NO891588D0 (no)	1989-04-18	Fremgangsmaate for fremstilling av fosfonoalkylpurinderivater.
NO883145L (no)	1989-01-16	Fremgangsmaate til fremstilling av tienoimidazol-derivater.
NO167807C (no)	1991-12-11	Analogifremgangsmaate til fremstilling av 3',4'-dinitrogensubstituerte epipodofyllotoksinglukosidderivater.
NO882730D0 (no)	1988-06-21	Fremgangsmaate for fremstilling av aminocyklopentyletere.
NO885002D0 (no)	1988-11-09	Fremgangsmte for fremstilling av sialocylglycerolipider.
NO874199D0 (no)	1987-10-07	Fremgangsmaate for fremstilling av imidazo-pyridinonderivater.
NO900972L (no)	1990-09-04	Fremgangsmaate for fremstilling av terapeutisk aktive naftalen-derivater.
NO883398D0 (no)	1988-08-01	Fremgangsmaate for fremstilling av benzoksazinderivater.
NO884100L (no)	1989-03-17	Fremgangsmaate for fremstilling av halogentiazolderivater.
NO871721D0 (no)	1987-04-24	Fremgangsmaate for fremstilling av ergolenderivater.
NO883610D0 (no)	1988-08-12	Fremgangsmaate til fremstilling av substituerte tienoimidazol-derivater.
NO894707L (no)	1990-05-28	Fremgangsmaate for fremstilling av benzoksazinderivater.
NO880834L (no)	1988-08-29	Fremgangsmaate for fremstilling av heterocyclyl-2-propyn-1-aminer.
NO873019D0 (no)	1987-07-20	Fremgangsmaate for fremstilling av tetrahydrobenzotiazolkinolin-derivater.
NO874698D0 (no)	1987-11-11	Fremgangsmaate for fremstilling av 2-guanidinothiazolderivater.
NO871521L (no)	1988-10-11	Fremgangsmaate for fremstilling av benzoksa- henholdsvis benzotia-diazolderivater.
NO884901L (no)	1989-05-05	Fremgangsmaate for fremstilling av nye indenofuran-derivater.
NO903254L (no)	1990-09-20	Fremgangsmaate for fremstilling av kinuklidin-derivater.