NO884467L - Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-cykloalkylbenzenderivater. - Google Patents

Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-cykloalkylbenzenderivater.

Info

Publication number: NO884467L
Authority: NO; Norway
Prior art keywords: aminomethyloxooxazolidinyl; cycloalkyl; preparation; analogy procedure; benzen
Prior art date: 1987-10-09

Application number

NO88884467A

Other languages

English (en)

Other versions

NO172890B (no

NO884467D0 (no

NO172890C (no

Inventor

Chia-Lin Jeffrey Wang

Mark Arvid Wuonola

Original Assignee

Du Pont

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-10-09

Filing date

1988-10-07

Publication date

1989-04-10

1988-10-07 Application filed by Du Pont filed Critical Du Pont

1988-10-07 Publication of NO884467D0 publication Critical patent/NO884467D0/no

1989-04-10 Publication of NO884467L publication Critical patent/NO884467L/no

1993-06-14 Publication of NO172890B publication Critical patent/NO172890B/no

1993-09-22 Publication of NO172890C publication Critical patent/NO172890C/no

Links

UHOVQNZJYSORNB-UHFFFAOYSA-N Benzene Chemical class C1=CC=CC=C1 UHOVQNZJYSORNB-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO884467A 1987-10-09 1988-10-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive aminomethyloxooxazolidinyl-cykloalkylbenzenderivater NO172890C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/106,358 US4801600A (en)	1987-10-09	1987-10-09	Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents

Publications (4)

Publication Number	Publication Date
NO884467D0 NO884467D0 (no)	1988-10-07
NO884467L true NO884467L (no)	1989-04-10
NO172890B NO172890B (no)	1993-06-14
NO172890C NO172890C (no)	1993-09-22

Family

ID=22310972

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO884467A NO172890C (no)	1987-10-09	1988-10-07	Analogifremgangsmaate for fremstilling av terapeutisk aktive aminomethyloxooxazolidinyl-cykloalkylbenzenderivater

Country Status (16)

Country	Link
US (1)	US4801600A (no)
EP (1)	EP0311090A1 (no)
JP (1)	JPH01132569A (no)
KR (1)	KR890006632A (no)
AU (1)	AU613669B2 (no)
CA (1)	CA1322001C (no)
DK (1)	DK562888A (no)
FI (1)	FI884610A7 (no)
HU (1)	HU202216B (no)
IL (1)	IL87972A (no)
MY (1)	MY103618A (no)
NO (1)	NO172890C (no)
NZ (1)	NZ226493A (no)
PT (1)	PT88713B (no)
SU (1)	SU1616518A3 (no)
ZA (1)	ZA887550B (no)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
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US4985429A (en) *	1987-10-09	1991-01-15	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4942183A (en) *	1987-10-16	1990-07-17	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A (en) *	1987-10-21	1990-12-11	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US4948801A (en) *	1988-07-29	1990-08-14	E. I. Du Pont De Nemours And Company	Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5164510A (en) *	1988-09-15	1992-11-17	The Upjohn Company	5'Indolinyl-5β-amidomethyloxazolidin-2-ones
US5182403A (en) *	1988-09-15	1993-01-26	The Upjohn Company	Substituted 3(5'indazolyl) oxazolidin-2-ones
US5225565A (en) *	1988-09-15	1993-07-06	The Upjohn Company	Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones
AU617871B2 (en) *	1988-09-15	1991-12-05	Pharmacia & Upjohn Company	In position 3 substituted-5-beta-amidomethyl-oxazolidin-2- ones
US5231188A (en) *	1989-11-17	1993-07-27	The Upjohn Company	Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents
PT97888B (pt) *	1990-06-07	1998-12-31	Zeneca Ltd	Processo para a preparacao de compostos heterociclicos derivados de indol e de composicoes farmaceuticas que os contem
JP2669579B2 (ja) *	1991-10-23	1997-10-29	エーザイ株式会社	オキサゾリドン誘導体
ATE146783T1 (de) *	1991-11-01	1997-01-15	Upjohn Co	Substituierte aryl- und heteroaryl- phenyloxazolidinone
SK283420B6 (sk) *	1992-05-08	2003-07-01	Pharmacia & Upjohn Company	Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
EP0673370B1 (en) *	1992-12-08	1998-01-07	PHARMACIA & UPJOHN COMPANY	Tropone-substituted phenyloxazolidinone antibacterial agents
US5688792A (en) *	1994-08-16	1997-11-18	Pharmacia & Upjohn Company	Substituted oxazine and thiazine oxazolidinone antimicrobials
EP0730591B1 (en) *	1993-11-22	1999-07-14	PHARMACIA & UPJOHN COMPANY	Esters of substituted-hydroxyacetyl piperazine phenyl oxazolidinones
DE4425612A1 (de) *	1994-07-20	1996-04-04	Bayer Ag	6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
DE4425609A1 (de) *	1994-07-20	1996-01-25	Bayer Ag	Benzofuranyl- und Benzothienyloxazolidinone
DE4425613A1 (de) *	1994-07-20	1996-01-25	Bayer Ag	5-gliedrige Heteroaryl-oxazolidinone
DE19514313A1 (de)	1994-08-03	1996-02-08	Bayer Ag	Benzoxazolyl- und Benzothiazolyloxazolidinone
BR9509673A (pt) *	1994-11-15	1997-09-30	Upjohn Co	Compostos e uso dos mesmos
DK0807112T3 (da) *	1995-02-03	2001-12-17	Upjohn Co	Antimikrobiel heteroaromatisk ringsubstitueret phenyloxazolidinon
HRP960159A2 (en) *	1995-04-21	1997-08-31	Bayer Ag	Benzocyclopentane oxazolidinones containing heteroatoms
NZ306310A (en) *	1995-05-11	2001-05-25	Upjohn Co	Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones
US5883093A (en) *	1995-09-12	1999-03-16	Pharmacia & Upjohn Company	Phenyloxazolidinone antimicrobials
DE19601264A1 (de)	1996-01-16	1997-07-17	Bayer Ag	Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone
DE19601265A1 (de) *	1996-01-16	1997-07-17	Bayer Ag	2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone
DE19601627A1 (de) *	1996-01-18	1997-07-24	Bayer Ag	Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone
HRP970049A2 (en) *	1996-02-06	1998-04-30	Bayer Ag	New heteroaryl oxazolidinones
DE19604223A1 (de) *	1996-02-06	1997-08-07	Bayer Ag	Neue substituierte Oxazolidinone
MY116093A (en) *	1996-02-26	2003-11-28	Upjohn Co	Azolyl piperazinyl phenyl oxazolidinone antimicrobials
BR9813985A (pt) *	1997-11-12	2000-09-26	Upjohn Co	Derivados de oxazolidinona e composições farmacêuticas
DE19802235A1 (de) *	1998-01-22	1999-07-29	Bayer Ag	Mit tricyclischen Indolen substituierte Oxazolidinone
KR20010015910A (ko) *	1998-01-23	2001-02-26	로렌스 티. 마이젠헬더	옥사졸리디논 조합 라이브러리, 조성물 및 제조 방법
JP2002535680A (ja)	1999-01-27	2002-10-22	ファルマシア・アンド・アップジョン・カンパニー	延長因子ｐ活性モジュレーターのアッセイ方法
ES2203473T3 (es) *	1999-05-27	2004-04-16	PHARMACIA & UPJOHN COMPANY	Oxazolidinonas biciclicas como agentes antibacterianos.
US6444813B2 (en) *	2000-02-02	2002-09-03	Pharmacia & Upjohn Company	Linezolid-crystal form II
BR0112826A (pt)	2000-07-17	2003-06-24	Ranbaxy Lab Ltd	Derivados da oxazolidinona como antimicrobianos
PE20020689A1 (es) *	2000-11-17	2002-08-03	Upjohn Co	Oxazolidinonas con un heterociclo de 6 o 7 miembros unidos con enlace anular al benceno
ES2256331T3 (es)	2000-12-21	2006-07-16	PHARMACIA & UPJOHN COMPANY LLC	Derivados de quinolina antimicrobianos y uso de los mismos para tratar infecciones bacterianas.
US6956040B2 (en)	2001-07-16	2005-10-18	Ranbaxy Laboratories Limited	Oxazolidinone piperazinyl derivatives as potential antimicrobials
EP1409464A4 (en) *	2001-07-16	2005-11-02	Ranbaxy Lab Ltd	OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS
US20050209248A1 (en) *	2002-05-15	2005-09-22	Biswajit Das	Plymorphic forms of phenyl oxazolidinone derivatives
MXPA05001199A (es) *	2002-07-29	2005-05-16	Ranbaxy Lab Ltd	Derivados de oxazolidinona como antimicrobianos.
JP2006516989A (ja) *	2003-02-07	2006-07-13	ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー	抗菌剤として使用するための二環式環によりｎ−置換されたオキサゾリジノン誘導体
US20080214565A1 (en) *	2003-04-07	2008-09-04	Anita Mehta	Oxazolidinone Derivatives as Antimicrobials
EP1866295A2 (en)	2005-02-24	2007-12-19	Teva Pharmaceutical Industries Ltd	Processes for the preparation of linezolid intermediate
US20100298384A1 (en) *	2006-12-04	2010-11-25	Mohamed Takhi	Novel oxazolidinone compounds as antiinfective agents
CA2712613C (en) *	2008-03-26	2017-02-28	Global Alliance For Tb Drug Development	Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones
US12479816B2 (en)	2019-02-08	2025-11-25	University of Pittsburgh—of the Commonwealth System of Higher Education	20-HETE formation inhibitors

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US29607A (en) *		1860-08-14		Portable scaffold
GB1222708A (en) *	1968-10-22	1971-02-17	Delalande Sa	Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
USRE29607E (en)	1969-03-18	1978-04-11	Delalande S. A.	Derivatives of 5-hydroxymethyl-3-substituted-2-oxazolidinones, process of preparation thereof and therapeutic application
LU80081A1 (fr) *	1977-08-26	1979-05-15	Delalande Sa	Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique
US4128654A (en) *	1978-02-10	1978-12-05	E. I. Du Pont De Nemours And Company	5-Halomethyl-3-phenyl-2-oxazolidinones
CA1171865A (en) *	1980-06-04	1984-07-31	Alain Lacour	N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics
US4340606A (en) *	1980-10-23	1982-07-20	E. I. Du Pont De Nemours And Company	3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents
FR2500450A1 (fr) *	1981-02-25	1982-08-27	Delalande Sa	Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
US4461773A (en) *	1982-09-15	1984-07-24	E. I. Dupont De Nemours And Company	P-Oxooxazolidinylbenzene compounds as antibacterial agents
US4705799A (en) *	1983-06-07	1987-11-10	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
ES8506659A1 (es) *	1983-06-07	1985-08-01	Du Pont	Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno.
CA1260948A (en) *	1984-12-05	1989-09-26	E. I. Du Pont De Nemours And Company	Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents

1987
- 1987-10-09 US US07/106,358 patent/US4801600A/en not_active Expired - Lifetime
1988
- 1988-10-04 CA CA000579301A patent/CA1322001C/en not_active Expired - Fee Related
- 1988-10-06 AU AU23507/88A patent/AU613669B2/en not_active Ceased
- 1988-10-06 SU SU884356653A patent/SU1616518A3/ru active
- 1988-10-07 NO NO884467A patent/NO172890C/no unknown
- 1988-10-07 IL IL87972A patent/IL87972A/xx unknown
- 1988-10-07 JP JP63252207A patent/JPH01132569A/ja active Pending
- 1988-10-07 MY MYPI88001123A patent/MY103618A/en unknown
- 1988-10-07 EP EP88116621A patent/EP0311090A1/en not_active Withdrawn
- 1988-10-07 DK DK562888A patent/DK562888A/da not_active Application Discontinuation
- 1988-10-07 ZA ZA887550A patent/ZA887550B/xx unknown
- 1988-10-07 KR KR1019880013071A patent/KR890006632A/ko not_active Ceased
- 1988-10-07 HU HU885214A patent/HU202216B/hu not_active IP Right Cessation
- 1988-10-07 PT PT88713A patent/PT88713B/pt not_active IP Right Cessation
- 1988-10-07 NZ NZ226493A patent/NZ226493A/xx unknown
- 1988-10-07 FI FI884610A patent/FI884610A7/fi not_active Application Discontinuation

Also Published As

Publication number	Publication date
PT88713B (pt)	1992-12-31
NO172890B (no)	1993-06-14
ZA887550B (en)	1990-06-27
US4801600A (en)	1989-01-31
KR890006632A (ko)	1989-06-14
IL87972A (en)	1993-05-13
MY103618A (en)	1993-08-28
DK562888D0 (da)	1988-10-07
HUT53359A (en)	1990-10-28
EP0311090A1 (en)	1989-04-12
NO884467D0 (no)	1988-10-07
JPH01132569A (ja)	1989-05-25
FI884610A0 (fi)	1988-10-07
DK562888A (da)	1989-04-10
HU202216B (en)	1991-02-28
AU2350788A (en)	1989-04-13
AU613669B2 (en)	1991-08-08
IL87972A0 (en)	1989-03-31
FI884610A7 (fi)	1989-04-10
NO172890C (no)	1993-09-22
NZ226493A (en)	1990-09-26
CA1322001C (en)	1993-09-07
SU1616518A3 (ru)	1990-12-23

Publication	Publication Date	Title
NO884467L (no)	1989-04-10	Analogifremgangsmaate for fremstilling av aminomethyloxooxazolidinyl-cykloalkylbenzenderivater.
NO893076L (no)	1990-01-30	Fremgangsmaate for fremstilling av aminomethyloxooxa-zolidinylarylbenzenderivater.
NO870579L (no)	1987-08-17	Fremgangsmaate for fremstilling av indolizin-derivater.
NO842273L (no)	1984-12-10	Fremgangsmaate ved fremstilling av aminomethyloxooxazolidinylbenzenderivater.
NO892936D0 (no)	1989-07-17	Fremgangsmaate for fremstilling av furanderivater.
NO880910D0 (no)	1988-03-01	Fremgangsmaate for fremstilling av chromonderivater.
NO884900D0 (no)	1988-11-03	Fremgangsmaate for fremstilling av ginkolid-derivater.
NO891588L (no)	1989-10-20	Fremgangsmaate for fremstilling av fosfonoalkylpurinderivater.
NO883145D0 (no)	1988-07-14	Fremgangsmaate til fremstilling av tienoimidazolderivater.
NO167807C (no)	1991-12-11	Analogifremgangsmaate til fremstilling av 3',4'-dinitrogensubstituerte epipodofyllotoksinglukosidderivater.
NO170022C (no)	1992-09-02	Fremgangsmaate for fremstilling av sialocylglycerolipider.
NO882730D0 (no)	1988-06-21	Fremgangsmaate for fremstilling av aminocyklopentyletere.
NO874199D0 (no)	1987-10-07	Fremgangsmaate for fremstilling av imidazo-pyridinonderivater.
NO884100L (no)	1989-03-17	Fremgangsmaate for fremstilling av halogentiazolderivater.
NO883398D0 (no)	1988-08-01	Fremgangsmaate for fremstilling av benzoksazinderivater.
NO871721D0 (no)	1987-04-24	Fremgangsmaate for fremstilling av ergolenderivater.
NO883610L (no)	1989-02-16	Fremgangsmaate til fremstilling av substituerte tienoimidazol-derivater.
NO894707L (no)	1990-05-28	Fremgangsmaate for fremstilling av benzoksazinderivater.
NO880834D0 (no)	1988-02-25	Fremgangsmaate for fremstilling av heterocyclyl-2-propyn-1-aminer.
NO874698L (no)	1988-05-13	Fremgangsmaate for fremstilling av 2-guanidinothiazolderivater.
NO873019D0 (no)	1987-07-20	Fremgangsmaate for fremstilling av tetrahydrobenzotiazolkinolin-derivater.
NO871521D0 (no)	1987-04-10	Fremgangsmaate for fremstilling av benzoksa- henholdsvis benzotia-diazolderivater.
NO884901L (no)	1989-05-05	Fremgangsmaate for fremstilling av nye indenofuran-derivater.
NO903254L (no)	1990-09-20	Fremgangsmaate for fremstilling av kinuklidin-derivater.
NO883525L (no)	1989-02-13	Framgangsmaate for framstilling av 1,5-benzotiazepinderivater.