NO931697L - Lhrh-antagonister - Google Patents

Lhrh-antagonister

Info

Publication number
NO931697L
NO931697L NO93931697A NO931697A NO931697L NO 931697 L NO931697 L NO 931697L NO 93931697 A NO93931697 A NO 93931697A NO 931697 A NO931697 A NO 931697A NO 931697 L NO931697 L NO 931697L
Authority
NO
Norway
Prior art keywords
parent compound
dala10
leu7
ser4
pro9
Prior art date
Application number
NO93931697A
Other languages
English (en)
Norwegian (no)
Other versions
NO931697D0 (no
Inventor
Shabo Tianjin Xiao
Original Assignee
Asta Medica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Medica Ag filed Critical Asta Medica Ag
Publication of NO931697D0 publication Critical patent/NO931697D0/no
Publication of NO931697L publication Critical patent/NO931697L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Medicinal Preparation (AREA)
NO93931697A 1990-11-10 1993-05-10 Lhrh-antagonister NO931697L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN90108955A CN1036343C (zh) 1990-11-10 1990-11-10 新促黄体生成素释放激素拮抗类似物的制备方法
PCT/EP1991/002110 WO1992008733A1 (en) 1990-11-10 1991-11-08 Lhrh-antagonists

Publications (2)

Publication Number Publication Date
NO931697D0 NO931697D0 (no) 1993-05-10
NO931697L true NO931697L (no) 1993-07-07

Family

ID=4881223

Family Applications (1)

Application Number Title Priority Date Filing Date
NO93931697A NO931697L (no) 1990-11-10 1993-05-10 Lhrh-antagonister

Country Status (29)

Country Link
EP (1) EP0564466B1 (pl)
KR (1) KR100244624B1 (pl)
CN (1) CN1036343C (pl)
AT (1) ATE149520T1 (pl)
AU (1) AU662496B2 (pl)
CA (1) CA2095932C (pl)
CZ (1) CZ284168B6 (pl)
DE (1) DE69125024T2 (pl)
DK (1) DK0564466T3 (pl)
EE (1) EE03141B1 (pl)
ES (1) ES2100965T3 (pl)
FI (1) FI933156A0 (pl)
GR (1) GR3023389T3 (pl)
HR (1) HRP920585B1 (pl)
IE (1) IE913915A1 (pl)
LT (1) LT3971B (pl)
LV (1) LV10106B (pl)
NO (1) NO931697L (pl)
NZ (1) NZ240505A (pl)
PH (1) PH31178A (pl)
PL (1) PL170564B1 (pl)
PT (1) PT99458B (pl)
RU (1) RU2123499C1 (pl)
SI (1) SI9111779B (pl)
SK (1) SK281319B6 (pl)
UA (1) UA41300C2 (pl)
WO (1) WO1992008733A1 (pl)
YU (1) YU48831B (pl)
ZA (1) ZA918847B (pl)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3568952B2 (ja) * 1992-12-18 2004-09-22 アボット・ラボラトリーズ ５位及び６位に修飾アミノアシル残基を有するｌｈｒｈ拮抗薬
DE4305225A1 (de) * 1993-02-19 1994-08-25 Asta Medica Ag Neues Herstellverfahren für Cetrorelix Lyophilisat
US6828415B2 (en) 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
DE4338015A1 (de) * 1993-11-08 1995-05-11 Asta Medica Ag Verwendung von D-glucopyranuronsäuren und deren Derivaten zum Einbau in pharmakologisch wirksame Peptide und deren Salze
US5843901A (en) * 1995-06-07 1998-12-01 Advanced Research & Technology Institute LHRH antagonist peptides
DE19544212A1 (de) * 1995-11-28 1997-06-05 Asta Medica Ag Neue LH-RH-Antagonisten mit verbesserter Wirkung
US5968547A (en) 1997-02-24 1999-10-19 Euro-Celtique, S.A. Method of providing sustained analgesia with buprenorphine
DE19911771B4 (de) * 1999-03-17 2006-03-30 Zentaris Gmbh LHRH-Antagonist, Verfahren zu seiner Herstellung und seiner Verwendung
CN101037472B (zh) * 2006-03-14 2013-03-27 中国人民解放军军事医学科学院毒物药物研究所 具有低组胺释放作用的促黄体生成素释放激素拮抗剂
CN102675418B (zh) * 2011-03-15 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物、其制备方法及用途
CN103524599B (zh) * 2012-07-05 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 环肽lhrh拮抗剂衍生物及其药物用途
CN104418936B (zh) * 2013-08-20 2018-06-05 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物及其药物用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4801577A (en) * 1987-02-05 1989-01-31 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US4851385A (en) * 1987-07-15 1989-07-25 Indiana University Foundation LHRH antagonist analogs having low histamine-release activity

Also Published As

Publication number Publication date
DE69125024D1 (de) 1997-04-10
LTIP1513A (en) 1995-06-26
PT99458A (pt) 1992-10-30
UA41300C2 (uk) 2001-09-17
HRP920585A2 (en) 1997-04-30
KR930703353A (ko) 1993-11-29
LT3971B (en) 1996-05-27
ES2100965T3 (es) 1997-07-01
DK0564466T3 (da) 1997-08-25
NZ240505A (en) 1993-04-28
SI9111779A (en) 1997-04-30
EE03141B1 (et) 1998-12-15
EP0564466B1 (en) 1997-03-05
FI933156A7 (fi) 1993-07-09
YU48831B (sh) 2002-03-18
IE913915A1 (en) 1992-05-20
EP0564466A1 (en) 1993-10-13
SI9111779B (en) 2001-12-31
PL170564B1 (pl) 1996-12-31
SK281319B6 (sk) 2001-02-12
GR3023389T3 (en) 1997-08-29
CA2095932C (en) 2003-02-25
NO931697D0 (no) 1993-05-10
ATE149520T1 (de) 1997-03-15
PT99458B (pt) 1999-02-26
AU8861291A (en) 1992-06-11
CZ84893A3 (en) 1994-02-16
RU2123499C1 (ru) 1998-12-20
PH31178A (en) 1998-03-20
DE69125024T2 (de) 1997-07-17
KR100244624B1 (ko) 2000-02-15
WO1992008733A1 (en) 1992-05-29
PL295427A1 (en) 1993-09-06
CN1036343C (zh) 1997-11-05
LV10106B (en) 1995-04-20
CN1061605A (zh) 1992-06-03
YU177991A (sh) 1994-06-24
ZA918847B (en) 1992-08-26
CZ284168B6 (cs) 1998-09-16
CA2095932A1 (en) 1992-05-11
LV10106A (lv) 1994-05-10
FI933156A0 (fi) 1993-07-09
HRP920585B1 (en) 2000-08-31
AU662496B2 (en) 1995-09-07
SK45393A3 (en) 1993-10-06

Similar Documents

Publication Publication Date Title
RU95114376A (ru) Нитроэфиры, обладающие фармакологической активностью, и способ их получения
CA2104873A1 (en) Compositions and Methods of Treatment of Sympathetically Maintained Pain
EA199800563A1 (ru) Антагонисты гормона, высвобождающего гонадотропин
RU92016471A (ru) Твердая непористая микросфера, способ ее получения и применение в фармакологическом препарате
BG50924A3 (bg) Метод за получаване на фармацевтичен състав
EP0695171A1 (en) GONADOTROPINE CONTAINING FREEZER DRIED DROPS
LV10949A (lv) Aizvietoti 4-fenil-4piperidinkarboksamidi to iegusanas panemiens farmaceitiska kompozicija
KR920700201A (ko) 신규 1α-히드록시비타민D 2 에피머 및 유도체
ATE160344T1 (de) Heterozyklische alkylamine, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen die sie enthalten
DE69310602D1 (de) 3',5'-Ditertbutyl-4'-Hydroxyflavone, Verfahren zu ihrer Herstellung und pharmazeutische Zusammensetzung mit Antioxidations- und Antivasokonstriktionsaktivität
ATE104273T1 (de) Benzolsulfonamide und verfahren zu ihrer herstellung.
UA42819C2 (uk) Ін`єкційний та інфузійний розчин, що містить енрофлокcацин
ATE149520T1 (de) Lhrh-antagonisten
HUT54113A (en) Process for producing butenecarboxylic acid derivatives and pharmaceutical compositions comprising such compounds
ATE177424T1 (de) N-substituierte naphthalimide, ihre herstellung und verwendung
ES2054186T3 (es) Composicion antihepatopatica.
KR870010036A (ko) 유기 아연 착화합물의 제조방법 및 활성 성분으로서 그를 함유하는 약학 조성물
EA199700302A1 (ru) Биологически активные уреидо-производные, полезные при лечении рассеянного склероза
RU94045890A (ru) Трициклические соединения-антагонисты тахикинина, их получение и фармацевтические композиции, содержащие такие соединения
KR940021524A (ko) 1,2,5,6-테트라하이드로피리딘 유도체와 이의 제조 방법 및 치료시 이의 이용방법
ES8407039A1 (es) Un procedimiento para preparacion de una quinalozina.
EP0254179A3 (de) Neue Tetrahydrobenzothiazolo-chinoline ihre Herstellung und Verwendung
RU94017615A (ru) Способ получения пептида
Caselli et al. Antihistaminic/antiallergic activity of 2-dialkylaminoalkylthio (OXY) 1-substituted benzimidazoles, evaluation “in vitro” and “in vivo”
TH19999A (th) ไดไฮโดรพิริดีนที่แสดงฤทธิ์ในระยะเวลาสั้น

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application