NO943280L - Fremgangsmåte for fremstilling av ger derav - Google Patents

Fremgangsmåte for fremstilling av ger derav

Info

Publication number: NO943280L
Authority: NO; Norway
Prior art keywords: pct; general formula; date sep; sec; ger
Prior art date: 1992-03-10

Application number

NO943280A

Other languages

English (en)

Other versions

NO304515B1 (no

NO943280D0 (no

Inventor

Jean-Dominique Bourzat

Alain Commercon

Original Assignee

Rhone Poulenc Rorer Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-03-10

Filing date

1994-09-05

Publication date

1994-09-05

1994-09-05 Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa

1994-09-05 Publication of NO943280L publication Critical patent/NO943280L/no

1994-09-05 Publication of NO943280D0 publication Critical patent/NO943280D0/no

1999-01-04 Publication of NO304515B1 publication Critical patent/NO304515B1/no

Links

RZARFIRJROUVLM-GVHYBUMESA-N (3r)-3-amino-2-hydroxy-3-phenylpropanoic acid Chemical compound OC(=O)C(O)[C@H](N)C1=CC=CC=C1 RZARFIRJROUVLM-GVHYBUMESA-N 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
150000007513 acids Chemical class 0.000 abstract 1
230000000719 anti-leukaemic effect Effects 0.000 abstract 1
230000000259 anti-tumor effect Effects 0.000 abstract 1
150000003934 aromatic aldehydes Chemical class 0.000 abstract 1
150000003951 lactams Chemical class 0.000 abstract 1
DKPFODGZWDEEBT-QFIAKTPHSA-N taxane Chemical class C([C@]1(C)CCC[C@@H](C)[C@H]1C1)C[C@H]2[C@H](C)CC[C@@H]1C2(C)C DKPFODGZWDEEBT-QFIAKTPHSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Epoxy Compounds (AREA)
Steroid Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

NO943280A 1992-03-10 1994-09-05 FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt NO304515B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9202821A FR2688499B1 (fr)	1992-03-10	1992-03-10	Procede de preparation de la beta-phenylisoserine et de ses analogues.
PCT/FR1993/000224 WO1993017997A1 (fr)	1992-03-10	1993-03-08	PROCEDE DE PREPARATION DE LA β-PHENYLISOSERINE ET DE SES ANALOGUES

Publications (3)

Publication Number	Publication Date
NO943280L true NO943280L (no)	1994-09-05
NO943280D0 NO943280D0 (no)	1994-09-05
NO304515B1 NO304515B1 (no)	1999-01-04

Family

ID=9427518

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO943280A NO304515B1 (no)	1992-03-10	1994-09-05	FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt

Country Status (25)

Country	Link
US (2)	US5608102A (no)
EP (1)	EP0630365B1 (no)
JP (1)	JP3278768B2 (no)
KR (1)	KR100272650B1 (no)
AT (1)	ATE159512T1 (no)
AU (1)	AU667886B2 (no)
CA (1)	CA2130333C (no)
CZ (1)	CZ283613B6 (no)
DE (1)	DE69314779T2 (no)
DK (1)	DK0630365T3 (no)
ES (1)	ES2109509T3 (no)
FI (1)	FI113640B (no)
FR (1)	FR2688499B1 (no)
GE (1)	GEP19981430B (no)
GR (1)	GR3025117T3 (no)
HU (1)	HU213621B (no)
MX (1)	MX9301268A (no)
NO (1)	NO304515B1 (no)
NZ (1)	NZ249899A (no)
PL (1)	PL171551B1 (no)
RU (1)	RU2103258C1 (no)
SK (1)	SK281297B6 (no)
TW (1)	TW252971B (no)
WO (1)	WO1993017997A1 (no)
ZA (1)	ZA931677B (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU684218B2 (en) *	1994-07-26	1997-12-04	Indena S.P.A.	Semi-synthetic taxanes with anti-tumoural activity
US6765015B2 (en) *	1995-12-13	2004-07-20	Xechem International, Inc.	Halogenated paclitaxel derivatives
KR100225535B1 (ko)	1996-08-27	1999-10-15	정지석	파클리탁셀의 제조방법
EP1019347B1 (en) *	1997-08-21	2003-03-19	Florida State University	Method for the synthesis of taxanes
AU1701699A (en) *	1997-11-19	1999-06-07	Xechem International, Inc.	Halogenated paclitaxel derivatives
ITMI991483A1 (it)	1999-07-06	2001-01-06	Indena Spa	Derivati tassanici e procedimenti per la loro preparazione
JP4776843B2 (ja)	1999-10-01	2011-09-21	イムノゲンインコーポレーティッド	免疫複合体及び化学療法剤を用いる癌治療用組成物及び方法
JP2002080435A (ja) *	2000-06-26	2002-03-19	Kanegafuchi Chem Ind Co Ltd	３−アミノ−２−ヒドロキシプロピオン酸誘導体の製造法
US7126003B2 (en)	2001-03-07	2006-10-24	Daiichi Pharmaceutical Co., Ltd.	Method for producing 2-azetidinone derivative
EP1961735B1 (en) *	2007-02-22	2009-11-18	Indena S.P.A.	Process for the preparation of (2r,3s)-3-phenylisoserine methyl ester acetate salt
EP2080764B1 (en)	2008-01-18	2012-08-22	INDENA S.p.A.	Solid forms of ortataxel
CN102408356A (zh) *	2011-09-28	2012-04-11	北京东方协和医药生物技术有限公司	一种多西他赛手性侧链中间体的制备方法
EP3102195B1 (en) *	2014-02-03	2021-10-06	Quadriga Biosciences, Inc.	Beta-substituted beta-amino acids and analogs as chemotherapeutic agents
CN111100026A (zh) *	2019-12-30	2020-05-05	重庆市碚圣医药科技股份有限公司	一种紫杉醇恶唑环侧链中间体的制备方法
CN112574134A (zh) *	2020-12-30	2021-03-30	重庆市碚圣医药科技股份有限公司	一种多西紫杉醇侧链的合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2629819B1 (fr) *	1988-04-06	1990-11-16	Rhone Poulenc Sante	Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
IT1231751B (it) *	1989-04-12	1991-12-21	Sigma Tau Ind Farmaceuti	Procedimento per la produzione di r(+) amminocarnitina e s(-) amminocarnitina
US5175315A (en) *	1989-05-31	1992-12-29	Florida State University	Method for preparation of taxol using β-lactam
US5304670A (en) *	1989-08-23	1994-04-19	Centre National De La Recherche Scientifique	Process for the enantioselective preparation of phenylisoserine derivatives
FR2658510B1 (fr) *	1990-02-21	1992-04-30	Rhone Poulenc Sante	Nouveau derive de la beta-phenylisoserine, sa preparation et son emploi.
US5294737A (en) *	1992-02-27	1994-03-15	The Research Foundation State University Of New York	Process for the production of chiral hydroxy-β-lactams and hydroxyamino acids derived therefrom

1992
- 1992-03-10 FR FR9202821A patent/FR2688499B1/fr not_active Expired - Fee Related
1993
- 1993-03-08 DK DK93918746.4T patent/DK0630365T3/da active
- 1993-03-08 ES ES93918746T patent/ES2109509T3/es not_active Expired - Lifetime
- 1993-03-08 GE GEAP19932472A patent/GEP19981430B/en unknown
- 1993-03-08 DE DE69314779T patent/DE69314779T2/de not_active Expired - Lifetime
- 1993-03-08 PL PL93305059A patent/PL171551B1/pl unknown
- 1993-03-08 JP JP51539493A patent/JP3278768B2/ja not_active Expired - Lifetime
- 1993-03-08 SK SK1085-94A patent/SK281297B6/sk not_active IP Right Cessation
- 1993-03-08 MX MX9301268A patent/MX9301268A/es unknown
- 1993-03-08 US US08/295,677 patent/US5608102A/en not_active Expired - Lifetime
- 1993-03-08 KR KR1019940703156A patent/KR100272650B1/ko not_active Expired - Lifetime
- 1993-03-08 WO PCT/FR1993/000224 patent/WO1993017997A1/fr not_active Ceased
- 1993-03-08 CZ CZ942185A patent/CZ283613B6/cs not_active IP Right Cessation
- 1993-03-08 HU HU9402590A patent/HU213621B/hu unknown
- 1993-03-08 CA CA002130333A patent/CA2130333C/fr not_active Expired - Lifetime
- 1993-03-08 RU RU94045799A patent/RU2103258C1/ru active
- 1993-03-08 EP EP93918746A patent/EP0630365B1/fr not_active Expired - Lifetime
- 1993-03-08 AT AT93918746T patent/ATE159512T1/de active
- 1993-03-08 AU AU37557/93A patent/AU667886B2/en not_active Expired
- 1993-03-08 NZ NZ249899A patent/NZ249899A/en not_active IP Right Cessation
- 1993-03-09 ZA ZA931677A patent/ZA931677B/xx unknown
- 1993-03-10 TW TW082101775A patent/TW252971B/zh not_active IP Right Cessation
1994
- 1994-09-05 NO NO943280A patent/NO304515B1/no not_active IP Right Cessation
- 1994-09-09 FI FI944169A patent/FI113640B/fi not_active IP Right Cessation
1996
- 1996-08-23 US US08/697,420 patent/US5763628A/en not_active Expired - Lifetime
1997
- 1997-10-23 GR GR970401615T patent/GR3025117T3/el unknown

Also Published As

Publication number	Publication date
TW252971B (no)	1995-08-01
GEP19981430B (en)	1998-10-30
US5763628A (en)	1998-06-09
EP0630365A1 (fr)	1994-12-28
HU213621B (en)	1997-08-28
FI944169A0 (fi)	1994-09-09
ATE159512T1 (de)	1997-11-15
SK281297B6 (sk)	2001-02-12
CZ218594A3 (en)	1995-11-15
EP0630365B1 (fr)	1997-10-22
CA2130333A1 (fr)	1993-09-16
AU3755793A (en)	1993-10-05
FR2688499A1 (fr)	1993-09-17
CZ283613B6 (cs)	1998-05-13
RU2103258C1 (ru)	1998-01-27
AU667886B2 (en)	1996-04-18
MX9301268A (es)	1993-09-01
PL171551B1 (pl)	1997-05-30
JP3278768B2 (ja)	2002-04-30
FI113640B (fi)	2004-05-31
HUT68540A (en)	1995-06-28
NZ249899A (en)	1996-01-26
FR2688499B1 (fr)	1994-05-06
CA2130333C (fr)	2002-11-26
RU94045799A (ru)	1996-07-20
DE69314779T2 (de)	1998-02-26
SK108594A3 (en)	1995-02-08
NO304515B1 (no)	1999-01-04
ES2109509T3 (es)	1998-01-16
ZA931677B (en)	1993-10-06
DK0630365T3 (da)	1998-03-02
JPH07504425A (ja)	1995-05-18
US5608102A (en)	1997-03-04
WO1993017997A1 (fr)	1993-09-16
HU9402590D0 (en)	1994-11-28
FI944169L (fi)	1994-09-09
GR3025117T3 (en)	1998-01-30
DE69314779D1 (de)	1997-11-27
KR950700234A (ko)	1995-01-16
KR100272650B1 (ko)	2000-11-15
NO943280D0 (no)	1994-09-05

Legal Events

Date	Code	Title	Description
2013-04-15	MK1K	Patent expired

Publication	Publication Date	Title
AU699480B2 (en)	1998-12-03	2,2-Dichloroalkane carboxylic acids, processes for their production and pharmaceutical agents containing these
NO943280D0 (no)	1994-09-05	Fremgangsmåte for fremstilling av ger derav
DE69725608D1 (de)	2003-11-20	Indolin-2-one derivate, verfahren zu ihrer herstellung und dieseenthaltende arzneimittel
ATE215078T1 (de)	2002-04-15	Verbessertes verfahren zum herstellen von geschützten 3,4-dihydroxybuttersäure estern
DK0696281T3 (da)	1999-11-01	Hidtil ukendte 5-pyrrolyl-2-pyridylmethylsulfinylbenzimidazolderivater
ZA952771B (en)	1996-10-04	Novel compound
GB9126725D0 (en)	1992-02-12	Process
ATE246515T1 (de)	2003-08-15	Verfahren zur herstellung von oralen dosierungsformulierungen enthaltend diclofenac
AU5644296A (en)	1996-11-21	Novel heterocyclic chemistry
DE69104220D1 (de)	1994-10-27	Verfahren zur Herstellung von direktkomprimierten, Cephalosporansäure Derivate enthaltendenTabletten.
DE69330601D1 (de)	2001-09-20	Serotoninergische ergolin derivate
BR9610175A (pt)	1998-08-11	Composto processo de preparação do composto composição farmacêutica e utilização do composto
BG90414A (bg)	1993-12-24	2-азабицикло (2,2,1)-хепт-5- ен-2-оцетна киселина и нейни производни, метод за получаване и приложението им
HU886767D0 (en)	1990-09-28	Process for the preparation of new 20,21-dinor-eburnamenine derivatives, new intermediates thereof, as well as pharmaceutical compositions containing said compounds as active ingredients
AU6878900A (en)	2001-03-19	1,4-dihydropyridine-5-carboxylic acid ester derivatives and method for the preparation thereof
DE69414586D1 (de)	1998-12-17	Verfahren zur herstellung von indolizinderivaten
ATE188694T1 (de)	2000-01-15	Verfahren zur herstellung von benzopyranderivaten
AU1466592A (en)	1992-11-17	Gem-diphosphonic acid nitrosocarbamoyl derivatives, a process for the preparation thereof and pharmaceutical compositions containing them
AU1459192A (en)	1992-11-17	Aminoacyl derivatives of gem-diphosphonic acids, a process for the preparation thereof and pharmaceutical compositions containing them
DE69620244D1 (de)	2002-05-02	Verfahren zur herstellung von prostaglandin e1