NO974125L - N-benzylazoliumderivater - Google Patents
N-benzylazoliumderivaterInfo
- Publication number
- NO974125L NO974125L NO974125A NO974125A NO974125L NO 974125 L NO974125 L NO 974125L NO 974125 A NO974125 A NO 974125A NO 974125 A NO974125 A NO 974125A NO 974125 L NO974125 L NO 974125L
- Authority
- NO
- Norway
- Prior art keywords
- general formula
- group
- hydrogen
- formula
- independently
- Prior art date
Links
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical compound C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 abstract 2
- 230000000843 anti-fungal effect Effects 0.000 abstract 2
- FNEQHKCQXDKYEO-UHFFFAOYSA-N 1-benzylpyrrole Chemical class C1=CC=CN1CC1=CC=CC=C1 FNEQHKCQXDKYEO-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000000066 S-methyl group Chemical group [H]C([H])([H])S* 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 150000001450 anions Chemical class 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000001434 methanylylidene group Chemical group [H]C#[*] 0.000 abstract 1
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 230000004962 physiological condition Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/08—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing alicyclic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP96114390 | 1996-09-09 | ||
| EP97114246 | 1997-08-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO974125D0 NO974125D0 (no) | 1997-09-08 |
| NO974125L true NO974125L (no) | 1998-03-10 |
Family
ID=26142161
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO974125A NO974125L (no) | 1996-09-09 | 1997-09-08 | N-benzylazoliumderivater |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US5900486A (cs) |
| JP (1) | JP2965532B2 (cs) |
| KR (1) | KR100252433B1 (cs) |
| CN (1) | CN1182739A (cs) |
| AU (1) | AU3685097A (cs) |
| CA (1) | CA2214669A1 (cs) |
| CZ (1) | CZ282897A3 (cs) |
| HU (1) | HUP9701479A3 (cs) |
| IL (1) | IL121691A0 (cs) |
| MA (1) | MA26440A1 (cs) |
| NO (1) | NO974125L (cs) |
| NZ (1) | NZ328607A (cs) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2931399A (en) | 1998-03-06 | 1999-09-20 | F. Hoffmann-La Roche Ag | 3-(4-(4-cyanophenyl)thiazol-2-y))-1-(1h-1,2,4-triazol-1-yl) -butan-2-ol derivatives having antifungal activity |
| AU1915500A (en) * | 1998-11-20 | 2000-06-13 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
| US6319933B1 (en) | 2000-04-17 | 2001-11-20 | Basilea Pharmaceutica Ag | Azole derivatives |
| CA2822457C (en) | 2001-12-14 | 2016-03-08 | The University Of Wyoming | Methods and compositions for controlled resease of drugs |
| TW200606129A (en) * | 2004-07-26 | 2006-02-16 | Chugai Pharmaceutical Co Ltd | Novel cyclohexane derivative, its prodrug, its salt and diabetic therapeutic agent containing the same |
| CN101391985B (zh) * | 2007-09-18 | 2013-09-11 | 西南大学 | 具抗微生物活性的三唑鎓类化合物及制备方法和医药用途 |
| CN103857440B (zh) * | 2011-06-22 | 2018-09-25 | 维奥姆生物科学有限公司 | 基于缀合物的抗真菌和抗细菌前药 |
| CN104974143A (zh) * | 2015-05-12 | 2015-10-14 | 深圳致君制药有限公司 | 一种季铵盐类化合物、其制备方法以及用途 |
| WO2021034627A1 (en) * | 2019-08-16 | 2021-02-25 | Purdue Research Foundation | Small molecule stimulators of the core particle of the proteasome |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH468788A (de) * | 1966-04-29 | 1969-02-28 | Basf Ag | Mischung zur Bekämpfung von Algen und Pilzen |
| US4017631A (en) * | 1974-11-19 | 1977-04-12 | Janssen Pharmaceutica N.V. | Imidazolium salts |
| DE2531031C3 (de) * | 1975-07-11 | 1978-03-16 | Schuelke & Mayr Gmbh, 2000 Norderstedt | 1 -Benzyl-3-alkyI-imidazoliumsalze |
| DE2643563A1 (de) * | 1976-09-28 | 1978-03-30 | Bayer Ag | Alpha-(4-biphenylyl)-benzyl-azolium- salze, verfahren zu ihrer herstellung sowie ihre verwendung zur bekaempfung von mikroorganismen |
| DE2714290A1 (de) * | 1977-03-31 | 1978-10-05 | Bayer Ag | Fungizide mittel |
| US4218458A (en) * | 1978-06-23 | 1980-08-19 | Janssen Pharmaceutica, N.V. | Heterocyclic derivatives of (4-aryloxy-methyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles |
| US4402957A (en) * | 1979-04-04 | 1983-09-06 | Janssen Pharmaceutica N.V. | Heterocyclic derivatives of [4-(piperazin-1-ylphenyloxymethyl)-1,3-dioxolan-2-ylmethyl]-1H-imidazoles and 1H-1,2,4-triazoles |
| FR2486079A1 (fr) * | 1980-07-07 | 1982-01-08 | Rhone Poulenc Agrochimie | Sels quaternaires d'alcoyl-1-imidazolium de l'acide phosphoreux ou ses monoesters, procedes pour les preparer et compositions fongicides les contenant |
| US4490530A (en) * | 1981-01-14 | 1984-12-25 | Janssen Pharmaceutica N.V. | Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)-methyl-1H-imidazoles and 1H-1,2,4-triazoles |
| EP0069442B1 (en) * | 1981-06-06 | 1985-02-20 | Pfizer Limited | Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them |
| DE3217963A1 (de) * | 1982-05-13 | 1983-11-17 | Basf Ag, 6700 Ludwigshafen | Dibenzofuranoxyalkyl-imidazoliumsalze, verfahren zu ihrer herstellung und ihre verwendung als mikrozide |
| US4861879A (en) * | 1983-02-28 | 1989-08-29 | Janssen Pharmaceutica N.V. | [[4-[4-Phenyl-1-piperazinyl)phenoxymethyl]-1-3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles |
| DE3319845A1 (de) * | 1983-06-01 | 1984-12-06 | Basf Ag, 6700 Ludwigshafen | Arylalkylimidazolium- und -triazoliumsalze, verfahren zu ihrer herstellung und ihre verwendung als mikrozide |
| US5128351A (en) * | 1990-05-04 | 1992-07-07 | American Cyanamid Company | Bis-aryl amide and urea antagonists of platelet activating factor |
| ES2141329T3 (es) * | 1994-01-24 | 2000-03-16 | Janssen Pharmaceutica Nv | Antifungicos azolicos solubles en agua. |
| NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
-
1997
- 1997-08-26 NZ NZ328607A patent/NZ328607A/xx unknown
- 1997-09-03 IL IL12169197A patent/IL121691A0/xx unknown
- 1997-09-04 CA CA002214669A patent/CA2214669A1/en not_active Abandoned
- 1997-09-05 HU HU9701479A patent/HUP9701479A3/hu unknown
- 1997-09-05 AU AU36850/97A patent/AU3685097A/en not_active Abandoned
- 1997-09-08 KR KR1019970046176A patent/KR100252433B1/ko not_active Expired - Fee Related
- 1997-09-08 CN CN97118228A patent/CN1182739A/zh active Pending
- 1997-09-08 NO NO974125A patent/NO974125L/no not_active Application Discontinuation
- 1997-09-08 CZ CZ972828A patent/CZ282897A3/cs unknown
- 1997-09-09 US US08/926,392 patent/US5900486A/en not_active Expired - Fee Related
- 1997-09-09 JP JP9244252A patent/JP2965532B2/ja not_active Expired - Lifetime
- 1997-09-09 MA MA24786A patent/MA26440A1/fr unknown
-
1999
- 1999-01-08 US US09/226,987 patent/US5962686A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JPH10114758A (ja) | 1998-05-06 |
| NZ328607A (en) | 1999-08-30 |
| HUP9701479A3 (en) | 2001-02-28 |
| AU3685097A (en) | 1998-03-12 |
| NO974125D0 (no) | 1997-09-08 |
| HU9701479D0 (en) | 1997-10-28 |
| HUP9701479A2 (hu) | 1999-02-01 |
| KR100252433B1 (ko) | 2000-08-01 |
| MA26440A1 (fr) | 2004-12-20 |
| IL121691A0 (en) | 1998-02-22 |
| JP2965532B2 (ja) | 1999-10-18 |
| CZ282897A3 (cs) | 1998-06-17 |
| US5962686A (en) | 1999-10-05 |
| US5900486A (en) | 1999-05-04 |
| KR19980024429A (ko) | 1998-07-06 |
| CN1182739A (zh) | 1998-05-27 |
| CA2214669A1 (en) | 1998-03-09 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CA2396738A1 (en) | Thiazole derivatives as active superoxide radical inhibitors | |
| CA2319005A1 (en) | 2-pyridylmethylamine derivatives useful as fungicides | |
| IL135537A0 (en) | Substituted fused heterocyclic compounds | |
| CA2273951A1 (en) | Parasiticidal pyrazoles | |
| AU589410B2 (en) | 5-(6-imidazo(1,2-A)pyridyl)pyridine derivative | |
| MX9701685A (es) | Nuevos derivados de bencimidazol que tienen la actividad de inhibicion de la fosfodiestearasa cgmp. | |
| MX9800718A (es) | Derivados de 2-(4-substituidos)-bencilamino-2-metil- propanamida. | |
| NO974125L (no) | N-benzylazoliumderivater | |
| AU629048B2 (en) | N-(-4-(phenyl)-1,2-dihydro-3-quinolyl)-N'-(phenyl) urea derivatives and their use | |
| EP0829478A3 (en) | N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents | |
| DE69810960D1 (de) | 2-phenoxyanilin-derivate | |
| NZ304438A (en) | Substituted triazole derivatives and antifungal compositions | |
| NZ296285A (en) | Inhibiting physiological conditions associated with bradykinin using a benzothiophene such as raloxifene | |
| EP0795326A4 (cs) | ||
| EP0291247A3 (en) | Novel cinnamoylamide derivatives | |
| SG50820A1 (en) | Novel thiouracil derivatives and metal surface- treating agent comprising thereof | |
| NZ335975A (en) | Heterocyclic substituted pyrrolidine amide derivatives useful in treating respiratory diseases | |
| NO963307L (no) | Karbamoylmetylureaderivater | |
| TW334426B (en) | Piperazine derivatives | |
| EP0443474A3 (en) | 1-phenoxycarbonyl-2-pyrrolidinone derivatives and nootropic agents | |
| TW358809B (en) | Phenylamidinothiophene compound and anti-inflammatory agent containing the same | |
| ECSP972249A (es) | Derivados de n-bencilazolio | |
| IL126548A0 (en) | Use of aspirochlorine or derivatives thereof as immunosuppressive agents | |
| DE60009301D1 (en) | Benzimidazolverbindungen | |
| CO5040060A1 (es) | Derivados de n-bencilazolio |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |