NO975578L - Vinyl sulfosides and a process for their preparation - Google Patents

Vinyl sulfosides and a process for their preparation

Info

Publication number
NO975578L
NO975578L NO975578A NO975578A NO975578L NO 975578 L NO975578 L NO 975578L NO 975578 A NO975578 A NO 975578A NO 975578 A NO975578 A NO 975578A NO 975578 L NO975578 L NO 975578L
Authority
NO
Norway
Prior art keywords
sulfosides
vinyl
preparation
arylalkoxy
alkoxy
Prior art date
Application number
NO975578A
Other languages
Norwegian (no)
Other versions
NO975578D0 (en
Inventor
James A Aikins
Randal S Miller
Tony Y Zhang
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/483,130 external-priority patent/US6372945B1/en
Priority claimed from US08/478,706 external-priority patent/US5659087A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO975578D0 publication Critical patent/NO975578D0/en
Publication of NO975578L publication Critical patent/NO975578L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/16—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)

Abstract

Det er beskrevet nye diarylvenylsulfoksyder av formelen hvor RI er hydrogen, Ci-C* alkoksy, arylalk oksy, halogen eller amino; R2 er hydrogen, C|-C< alkoksy, arylalkoksy, halogen eller amino; og R3 er en termisk labil eller syrelabil CrC10 alkyl, C4-C|0 alkenyl eller aryl (C,-C1 alkyl) gruppe. Det er videre beskrevet fremgangmåter for fremstilling av disse forbindelsene.There are disclosed novel diarylvenyl sulfoxides of the formula wherein R 1 is hydrogen, C 1 -C 4 alkoxy, arylalkoxy, halogen or amino; R 2 is hydrogen, C 1 -C 4 alkoxy, arylalkoxy, halogen or amino; and R 3 is a thermally labile or acid labile C 1 -C 10 alkyl, C 4 -C 20 alkenyl or aryl (C 1 -C 1 alkyl) group. Methods for preparing these compounds are further described.

NO975578A 1995-06-07 1997-12-03 Vinyl sulfosides and a process for their preparation NO975578L (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/483,130 US6372945B1 (en) 1995-06-07 1995-06-07 Process for the synthesis of vinyl sulfoxides
US08/478,706 US5659087A (en) 1995-06-07 1995-06-07 Diarylvinyl sulfoxides
PCT/US1996/009163 WO1996040691A1 (en) 1995-06-07 1996-06-04 Vinyl sulfoxides and a process for their synthesis

Publications (2)

Publication Number Publication Date
NO975578D0 NO975578D0 (en) 1997-12-03
NO975578L true NO975578L (en) 1997-12-03

Family

ID=27045988

Family Applications (2)

Application Number Title Priority Date Filing Date
NO975578A NO975578L (en) 1995-06-07 1997-12-03 Vinyl sulfosides and a process for their preparation
NO20005987A NO20005987D0 (en) 1995-06-07 2000-11-27 Process for the preparation of vinyl sulfoxides

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20005987A NO20005987D0 (en) 1995-06-07 2000-11-27 Process for the preparation of vinyl sulfoxides

Country Status (16)

Country Link
EP (1) EP0830361A4 (en)
JP (1) JPH11507061A (en)
KR (1) KR19990022362A (en)
CN (2) CN1192741A (en)
AU (1) AU697352B2 (en)
BR (1) BR9608579A (en)
CA (1) CA2220145A1 (en)
CZ (1) CZ393097A3 (en)
EA (1) EA000405B1 (en)
HU (1) HUP9900922A3 (en)
IL (1) IL122090A0 (en)
NO (2) NO975578L (en)
NZ (1) NZ310179A (en)
PL (1) PL324035A1 (en)
TR (3) TR199801495T2 (en)
WO (1) WO1996040691A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4596651B2 (en) * 1999-04-02 2010-12-08 テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション (E) -styrylsulfone anticancer agent
EP1546138B1 (en) 2002-09-30 2012-01-18 A/S GEA Farmaceutisk Fabrik Raloxifene l-lactate or a hemihydrate thereof, their uses, pharmaceutical compositions and preparation processes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5514826A (en) * 1995-06-07 1996-05-07 Eli Lilly And Company Vinyl sulfenic acid derivatives
US5512701A (en) * 1995-06-07 1996-04-30 Eli Lilly And Company Process for the synthesis of vinyl sulfenic acid derivatives
CA2224225A1 (en) * 1995-06-07 1996-12-19 Wayne Douglas Luke Process for the synthesis of vinyl sulfenic acid derivatives

Also Published As

Publication number Publication date
IL122090A0 (en) 1998-04-05
CZ393097A3 (en) 1998-06-17
KR19990022362A (en) 1999-03-25
JPH11507061A (en) 1999-06-22
EP0830361A4 (en) 1998-12-30
CN1192741A (en) 1998-09-09
NO20005987D0 (en) 2000-11-27
NZ310179A (en) 1999-09-29
HUP9900922A3 (en) 2000-06-28
CN1341596A (en) 2002-03-27
EA000405B1 (en) 1999-06-24
TR199801495T2 (en) 1998-09-21
PL324035A1 (en) 1998-05-11
TR199801494T2 (en) 1998-09-21
TR199701510T1 (en) 1998-03-21
EP0830361A1 (en) 1998-03-25
AU697352B2 (en) 1998-10-01
EA199800028A1 (en) 1998-08-27
NO975578D0 (en) 1997-12-03
HUP9900922A2 (en) 1999-07-28
NO5987A (en) 1997-12-03
WO1996040691A1 (en) 1996-12-19
CA2220145A1 (en) 1996-12-19
AU6092096A (en) 1996-12-30
BR9608579A (en) 1999-01-05

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application