OA12244A - Oxazole derivatives and their uses as tyrosine kinase inhibitors. - Google Patents

Oxazole derivatives and their uses as tyrosine kinase inhibitors. Download PDF

Info

Publication number: OA12244A
Authority: OA; OAPI
Prior art keywords: compound; sait; formula; cancer; agent
Prior art date: 2000-04-07

Application number

OA1200200311A

Other languages

English (en)

Inventor

Takenori Hitaka

Etsuya Matsutani

Akihiro Tasaka

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-07

Filing date

2001-04-05

Publication date

2006-05-10

2001-04-05 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

2006-05-10 Publication of OA12244A publication Critical patent/OA12244A/en

Links

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

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Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

OA1200200311A 2000-04-07 2001-04-05 Oxazole derivatives and their uses as tyrosine kinase inhibitors. OA12244A (en)

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JP2000106836		2000-04-07

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US (2)	US6716863B2 (pl)
EP (1)	EP1268473A1 (pl)
KR (1)	KR20020028865A (pl)
CN (1)	CN1444582A (pl)
AU (1)	AU2001244726A1 (pl)
BR (1)	BR0109851A (pl)
CA (1)	CA2404760A1 (pl)
CO (1)	CO5261589A1 (pl)
CZ (1)	CZ20023264A3 (pl)
EE (1)	EE200200576A (pl)
HU (1)	HUP0300434A3 (pl)
IL (1)	IL152115A0 (pl)
MX (1)	MXPA02009621A (pl)
NO (1)	NO20024742L (pl)
OA (1)	OA12244A (pl)
PE (1)	PE20011178A1 (pl)
PL (1)	PL365787A1 (pl)
SK (1)	SK14132002A3 (pl)
WO (1)	WO2001077107A1 (pl)

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HUP0103761A3 (en) *	1998-10-08	2002-11-28	Takeda Chemical Industries Ltd	Compositions for retarding change of hormone-dependent cancer into hormone-independent cancer and their use
KR20030013360A (ko) *	2000-07-19	2003-02-14	다케다 야쿠힌 고교 가부시키가이샤	1-치환-1,2,3-트리아졸 유도체의 제조 방법
EP1382350A4 (en) *	2001-04-25	2006-01-04	Takeda Pharmaceutical	MEANS AGAINST THE PROPHYLAXIS BEFORE POSTOPERATIVE REPEAT OF PREMOPEOPAUSAL BREAST CANCER
US20040116330A1 (en) *	2001-04-27	2004-06-17	Kenichiro Naito	Preventive/therapeutic method for cancer
WO2002087619A1 (en) *	2001-04-27	2002-11-07	Takeda Chemical Industries, Ltd.	Preventive/therapeutic method for cancer
WO2003015820A1 (en) *	2001-08-10	2003-02-27	Takeda Chemical Industries, Ltd.	GnRH AGONIST COMBINATION DRUGS
EP1439178A4 (en) *	2001-10-05	2005-11-16	Takeda Pharmaceutical	Heterocyclic compounds, oxazole derivatives, process for their preparation and their use
EP1444988A4 (en)	2001-11-13	2007-04-25	Takeda Pharmaceutical	CANCER AGENT
AU2002349477A1 (en) *	2001-11-26	2003-06-10	Takeda Chemical Industries, Ltd.	Bicyclic derivative, process for producing the same, and use
WO2003059907A1 (en) *	2002-01-17	2003-07-24	Takeda Chemical Industries, Ltd.	Nitrogenous heterocyclic compounds, process for preparation of the same and use thereof
AU2003231098A1 (en)	2002-04-25	2003-11-10	University Of Connecticut Health Center	Using heat shock proteins to improve the therapeutic benefit of a non-vaccine treatment modality
HRP20050544B1 (hr) *	2002-12-16	2017-12-01	Kissei Pharmaceutical Co., Ltd.	Čvrsti oblik za oralnu upotrebu
TW200505913A (en) *	2003-03-28	2005-02-16	Hoffmann La Roche	Novel oxazole derivatives, their manufacture and use as pharmaceutical agents
TW200423931A (en)	2003-04-30	2004-11-16	Hoffmann La Roche	Novel aniline derivatives, their manufacture and use as pharmaceutical agents
US7247649B2 (en)	2003-08-13	2007-07-24	Hoffmann-La Roche Inc.	Oxazoles, their manufacture and use as pharmaceutical agents
US7259262B2 (en)	2003-10-24	2007-08-21	Hoffmann-La Roche Inc.	Arylazole derivatives, their manufacture and use as pharmaceutical agents
US20050186275A1 (en) *	2004-02-23	2005-08-25	Standard Chem. & Pharm. Co. Ltd.	Sustained release tamsulosin formulations
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2001
- 2001-04-03 PE PE2001000307A patent/PE20011178A1/es not_active Application Discontinuation
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- 2001-04-05 CN CN01807792A patent/CN1444582A/zh active Pending
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Publication number	Publication date
US20040024035A1 (en)	2004-02-05
MXPA02009621A (es)	2003-05-14
US6716863B2 (en)	2004-04-06
AU2001244726A1 (en)	2001-10-23
SK14132002A3 (sk)	2003-04-01
EP1268473A1 (en)	2003-01-02
US20020173526A1 (en)	2002-11-21
CN1444582A (zh)	2003-09-24
WO2001077107A8 (en)	2003-02-13
WO2001077107B1 (en)	2001-12-20
CO5261589A1 (es)	2003-03-31
CZ20023264A3 (cs)	2003-02-12
PE20011178A1 (es)	2001-11-19
PL365787A1 (pl)	2005-01-10
WO2001077107A1 (en)	2001-10-18
CA2404760A1 (en)	2001-10-18
BR0109851A (pt)	2003-06-03
HUP0300434A2 (hu)	2003-06-28
KR20020028865A (ko)	2002-04-17
IL152115A0 (en)	2003-05-29
NO20024742L (no)	2002-11-25
NO20024742D0 (no)	2002-10-02
HUP0300434A3 (en)	2004-11-29
EE200200576A (et)	2004-06-15

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