PE20099A1 - Derivados de espiro-piperidina y su uso como agentes terapeuticos - Google Patents

Derivados de espiro-piperidina y su uso como agentes terapeuticos

Info

Publication number: PE20099A1
Authority: PE; Peru
Prior art keywords: fenil; spiro; piperidine; derivatives; therapeutic agents
Prior art date: 1996-12-02

Application number

PE00108297A

Other languages

English (en)

Spanish (es)

Inventor

Brian John Williams

Raymond Baker

Timothy Harrison

Janusz Jozef Kulagowski

Christopher John Swain

Neil Roy Curtis

Gregory John Hollingworth

Eileen Mary Seward

Jason Matthew Elliott

Philip Stephen Jackson

Original Assignee

Merck Sharp & Dohme

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-12-02

Filing date

1997-12-01

Publication date

1999-03-05

1996-12-02 Priority claimed from GB9625051A external-priority patent/GB9625051D0/en

1997-01-24 Priority claimed from GB9701459A external-priority patent/GB9701459D0/en

1997-12-01 Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme

1999-03-05 Publication of PE20099A1 publication Critical patent/PE20099A1/es

Links

JUXAVSAMVBLDKO-UHFFFAOYSA-N 1-(1-azabicyclo[2.2.2]octan-3-yl)-3-[3-(1h-indol-3-yl)-1-oxo-1-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylpropan-2-yl]urea Chemical class C1N(CC2)CCC2C1NC(=O)NC(C(=O)N1CCC2(C3=CC=CC=C3CC2)CC1)CC1=CNC2=CC=CC=C12 JUXAVSAMVBLDKO-UHFFFAOYSA-N 0.000 title 1
239000003814 drug Substances 0.000 title 1
229940124597 therapeutic agent Drugs 0.000 title 1
HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical compound C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 2
RZVAJINKPMORJF-UHFFFAOYSA-N Acetaminophen Chemical compound CC(=O)NC1=CC=C(O)C=C1 RZVAJINKPMORJF-UHFFFAOYSA-N 0.000 abstract 2
206010061218 Inflammation Diseases 0.000 abstract 1
206010036376 Postherpetic Neuralgia Diseases 0.000 abstract 1
206010047700 Vomiting Diseases 0.000 abstract 1
239000005557 antagonist Substances 0.000 abstract 1
NRUQNUIWEUZVLI-UHFFFAOYSA-O diethanolammonium nitrate Chemical compound [O-][N+]([O-])=O.OCC[NH2+]CCO NRUQNUIWEUZVLI-UHFFFAOYSA-O 0.000 abstract 1
230000004054 inflammatory process Effects 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
239000000126 substance Substances 0.000 abstract 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Other In-Based Heterocyclic Compounds (AREA)

PE00108297A 1996-12-02 1997-12-01 Derivados de espiro-piperidina y su uso como agentes terapeuticos PE20099A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB9625051A GB9625051D0 (en)	1996-12-02	1996-12-02	Therapeutic agents
GB9701459A GB9701459D0 (en)	1997-01-24	1997-01-24	Therapeutic agents

Publications (1)

Publication Number	Publication Date
PE20099A1 true PE20099A1 (es)	1999-03-05

Family

ID=26310534

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PE00108297A PE20099A1 (es)	1996-12-02	1997-12-01	Derivados de espiro-piperidina y su uso como agentes terapeuticos

Country Status (4)

Country	Link
CO (1)	CO4910154A1 (id)
HR (1)	HRP970648A2 (id)
ID (1)	ID19017A (id)
PE (1)	PE20099A1 (id)

1997
- 1997-11-27 ID IDP973779A patent/ID19017A/id unknown
- 1997-12-01 CO CO97070178A patent/CO4910154A1/es unknown
- 1997-12-01 HR HRP970648 patent/HRP970648A2/hr not_active Application Discontinuation
- 1997-12-01 PE PE00108297A patent/PE20099A1/es not_active Application Discontinuation

Also Published As

Publication number	Publication date
ID19017A (id)	1998-06-04
HRP970648A2 (en)	1998-08-31
CO4910154A1 (es)	2000-04-24

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Legal Events

Date	Code	Title	Description
2001-03-15	FG	Grant, registration
2002-07-18	FD	Application declared void or lapsed