PE45295A1 - Peptidos inhibidores de proteasa - Google Patents

Peptidos inhibidores de proteasa

Info

Publication number
PE45295A1
PE45295A1 PE1995260194A PE26019495A PE45295A1 PE 45295 A1 PE45295 A1 PE 45295A1 PE 1995260194 A PE1995260194 A PE 1995260194A PE 26019495 A PE26019495 A PE 26019495A PE 45295 A1 PE45295 A1 PE 45295A1
Authority
PE
Peru
Prior art keywords
alkyl
compounds
formula
aralkyl
aryl
Prior art date
Application number
PE1995260194A
Other languages
English (en)
Spanish (es)
Inventor
Rainer Metternich
Anette Wienand
Carlo Tapparelli
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of PE45295A1 publication Critical patent/PE45295A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/08—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • A61K51/088—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Optics & Photonics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physics & Mathematics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PE1995260194A 1994-01-26 1995-01-24 Peptidos inhibidores de proteasa PE45295A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9401483A GB9401483D0 (en) 1994-01-26 1994-01-26 Organic compounds

Publications (1)

Publication Number Publication Date
PE45295A1 true PE45295A1 (es) 1995-12-29

Family

ID=10749357

Family Applications (1)

Application Number Title Priority Date Filing Date
PE1995260194A PE45295A1 (es) 1994-01-26 1995-01-24 Peptidos inhibidores de proteasa

Country Status (10)

Country Link
EP (1) EP0741747A1 (ja)
JP (1) JPH09509653A (ja)
AU (1) AU1576495A (ja)
CA (1) CA2179889A1 (ja)
GB (1) GB9401483D0 (ja)
IL (1) IL112423A0 (ja)
PE (1) PE45295A1 (ja)
SG (1) SG47079A1 (ja)
WO (1) WO1995020603A1 (ja)
ZA (1) ZA95636B (ja)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9515489D0 (en) * 1995-07-28 1995-09-27 Sandoz Ltd Organic compounds
DE10046514A1 (de) 2000-09-15 2002-04-25 Diagnostikforschung Inst Verfahren zur bildlichen Darstellung und Diagnose von Thromben mittels Kernspintomographie unter Verwendung partikulärer Kontrastmittel
BR0314450A (pt) 2002-09-09 2005-07-26 Trigen Ltd Sais de ácido borÈnico com adição de uma base farmaceuticamente aceitável, formulação farmacêutica, e uso dos referidos sais para preparar uma formulação farmacêutica
US7576206B2 (en) 2003-08-14 2009-08-18 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7223745B2 (en) 2003-08-14 2007-05-29 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7468383B2 (en) 2005-02-11 2008-12-23 Cephalon, Inc. Proteasome inhibitors and methods of using the same
AU2010341530B2 (en) 2009-12-22 2016-03-10 Cephalon, Inc. Proteasome inhibitors and processes for their preparation, purification and use
PL3472149T3 (pl) 2016-06-21 2024-02-12 Orion Ophthalmology LLC Heterocykliczne pochodne prolinamidu
US10526315B2 (en) 2016-06-21 2020-01-07 Orion Ophthalmology LLC Carbocyclic prolinamide derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4668503A (en) * 1982-07-26 1987-05-26 Trustees Of University Of Massachusetts Process for labeling amines with 99m Tc
US5187157A (en) * 1987-06-05 1993-02-16 Du Pont Merck Pharmaceutical Company Peptide boronic acid inhibitors of trypsin-like proteases
EP0403243B1 (en) * 1989-06-16 1995-11-08 Merck Frosst Canada Inc. Chelate derivatives of atrial natriuretic factor (ANF)
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
US5252721A (en) * 1990-09-28 1993-10-12 Neorx Corporation S3 N chelating compounds
WO1992018536A2 (en) * 1991-04-22 1992-10-29 Mallinckrodt Medical, Inc. Method for detecting an localizing tissues having neurokinine 1 receptors

Also Published As

Publication number Publication date
ZA95636B (en) 1996-07-26
EP0741747A1 (en) 1996-11-13
AU1576495A (en) 1995-08-15
SG47079A1 (en) 1998-03-20
JPH09509653A (ja) 1997-09-30
IL112423A0 (en) 1995-03-30
WO1995020603A1 (en) 1995-08-03
CA2179889A1 (en) 1995-08-03
GB9401483D0 (en) 1994-03-23

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Legal Events

Date Code Title Description
FG Grant, registration
FD Application declared void or lapsed