PH12960A - Derivatives of 4,6-di-(aminoglycosyl)-1,3-diaminocy-clitols and pharmaceutical compositions thereof - Google Patents

Derivatives of 4,6-di-(aminoglycosyl)-1,3-diaminocy-clitols and pharmaceutical compositions thereof

Info

Publication number
PH12960A
PH12960A PH16732A PH16732A PH12960A PH 12960 A PH12960 A PH 12960A PH 16732 A PH16732 A PH 16732A PH 16732 A PH16732 A PH 16732A PH 12960 A PH12960 A PH 12960A
Authority
PH
Philippines
Prior art keywords
diaminocy
clitols
aminoglycosyl
derivatives
pharmaceutical compositions
Prior art date
Application number
PH16732A
Other languages
English (en)
Inventor
P Daniels
Original Assignee
Scherico Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scherico Ltd filed Critical Scherico Ltd
Publication of PH12960A publication Critical patent/PH12960A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
PH16732A 1974-03-19 1975-01-21 Derivatives of 4,6-di-(aminoglycosyl)-1,3-diaminocy-clitols and pharmaceutical compositions thereof PH12960A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US45257174A 1974-03-19 1974-03-19

Publications (1)

Publication Number Publication Date
PH12960A true PH12960A (en) 1979-10-19

Family

ID=23797003

Family Applications (1)

Application Number Title Priority Date Filing Date
PH16732A PH12960A (en) 1974-03-19 1975-01-21 Derivatives of 4,6-di-(aminoglycosyl)-1,3-diaminocy-clitols and pharmaceutical compositions thereof

Country Status (5)

Country Link
US (1) US4117221A (fr)
BE (1) BE824657A (fr)
CA (1) CA1046512A (fr)
DO (1) DOP1975002538A (fr)
PH (1) PH12960A (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5461151A (en) * 1977-10-25 1979-05-17 Shionogi & Co Ltd Novel aminoglycoside derivative
JPS5492951A (en) * 1977-12-29 1979-07-23 Shionogi & Co Ltd Novel aminoglycoside derivative
FR2435481A1 (fr) * 1978-09-06 1980-04-04 Roussel Uclaf Nouveaux aminoglycosides derives de la desoxystreptamine et leurs sels, procede de preparation et application a titre de medicaments
DE2840907A1 (de) * 1978-09-20 1980-04-03 Bayer Ag Selektiv geschuetzte 4,6-di-o-(aminoglykosyl)-1,3-diaminocyclitole
DE2921973A1 (de) * 1979-05-30 1980-12-11 Bayer Ag Sisomicin-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
US4387219A (en) * 1979-11-13 1983-06-07 Sterling Drug Inc. 2-Hydroxy gentamicin compounds
US4288547A (en) * 1979-11-13 1981-09-08 Haruo Yamamoto Fermentative process for preparing antibiotics of the gentamicin class
US4412068A (en) * 1981-06-08 1983-10-25 Sterling Drug Inc. Novel compounds of the gentamicin class
US7794713B2 (en) 2004-04-07 2010-09-14 Lpath, Inc. Compositions and methods for the treatment and prevention of hyperproliferative diseases
US7862812B2 (en) 2006-05-31 2011-01-04 Lpath, Inc. Methods for decreasing immune response and treating immune conditions
CN101152195B (zh) * 2007-10-09 2010-09-08 常州方圆制药有限公司 一种氨基糖苷类抗生素在制备治疗耐药菌感染的药物组合物中的应用
BRPI0819319B8 (pt) 2007-11-21 2021-05-25 Achaogen Inc análogos de aminoglicosídeo antibacteriano
WO2010132759A1 (fr) 2009-05-15 2010-11-18 Achaogen, Inc. Dérivés antibactériens de la dibékacine
WO2010132760A1 (fr) 2009-05-15 2010-11-18 Achaogen, Inc. Dérivés antibactériens de tobramycine
WO2010132757A2 (fr) 2009-05-15 2010-11-18 Achaogen, Inc. Analogues d'aminoglycoside antibactériens
WO2010132768A1 (fr) 2009-05-15 2010-11-18 Achaogen, Inc. Dérivés antibactériens de sisomicine
WO2010132765A2 (fr) 2009-05-15 2010-11-18 Achaogen, Inc. Analogues d'aminoglycoside antibactériens
US8906868B2 (en) * 2010-05-12 2014-12-09 Rempex Pharmaceuticals, Inc. Aminoglycoside derivatives
EA202090753A1 (ru) * 2017-06-16 2020-06-15 Борис Славинович ФАРБЕР Комбинаторные производные антибиотиков на основе супрамолекулярных структур

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3920628A (en) * 1972-10-24 1975-11-18 Schering Corp 2{41 -Deoxyaminoglycosides and 2{41 -epi-amino-3{41 -desamino derivatives thereof, methods for their manufacture and novel intermediates useful therein
US4029882A (en) * 1974-03-19 1977-06-14 Schering Corporation Selective acylation of the C-1 amino group of aminoglycoside antibiotics
US4002742A (en) * 1974-03-19 1977-01-11 Schering Corporation 1-N-alkyl-4,6-di-(aminoglycosyl)-1,3-diaminocyclitols, methods for their manufacture, methods for their use as antibacterial agents, and compositions useful therefor

Also Published As

Publication number Publication date
CA1046512A (fr) 1979-01-16
US4117221A (en) 1978-09-26
BE824657A (fr) 1975-07-22
DOP1975002538A (es) 1988-11-03

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