PH20029A - Benzodiazepine derivatives - Google Patents

Benzodiazepine derivatives

Info

Publication number: PH20029A
Authority: PH; Philippines
Prior art keywords: benzodiazepine derivatives; benzodiazepine; derivatives
Prior art date: 1983-08-25

Application number

PH31144A

Inventor

Rodney Ian Fryer

Armin Walser

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-08-25

Filing date

1984-08-24

Publication date

1986-09-04

1984-08-24 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1986-09-04 Publication of PH20029A publication Critical patent/PH20029A/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C247/00—Compounds containing azido groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
- C07D239/76—N-oxides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Anesthesiology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

PH31144A 1983-08-25 1984-08-24 Benzodiazepine derivatives PH20029A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US52619483A	1983-08-25	1983-08-25

Publications (1)

Publication Number	Publication Date
PH20029A true PH20029A (en)	1986-09-04

Family

ID=24096318

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PH31144A PH20029A (en)	1983-08-25	1984-08-24	Benzodiazepine derivatives

Country Status (16)

Country	Link
EP (1)	EP0135770A3 (en)
JP (1)	JPS6067480A (en)
KR (1)	KR850001756A (en)
AU (1)	AU3237984A (en)
DK (1)	DK406384A (en)
ES (2)	ES535392A0 (en)
FI (1)	FI843356A7 (en)
GR (1)	GR80197B (en)
HU (1)	HU193588B (en)
IL (1)	IL72757A0 (en)
MC (1)	MC1616A1 (en)
NO (1)	NO843376L (en)
NZ (1)	NZ209316A (en)
PH (1)	PH20029A (en)
PT (1)	PT79131B (en)
ZA (1)	ZA845757B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2635776B1 (en) *	1988-09-01	1993-06-11	Rhone Poulenc Agrochimie	AMIDE DERIVATIVES, PROCESS FOR THEIR MANUFACTURE AND FUNGICIDE COMPOSITIONS CONTAINING THEM
IL91418A (en) *	1988-09-01	1997-11-20	Rhone Poulenc Agrochimie	(hetero) cyclic amide derivatives, process for their preparation and fungicidal compositions containing them
US5317018A (en) *	1992-06-09	1994-05-31	Armin Walser	Benzodiazepines and compositions for treating anxiety and panic disorders, and idiopathic and psychomotor epilepsy
TW234123B (en) *	1992-12-16	1994-11-11	Takeda Pharm Industry Co Ltd
US6063921A (en) *	1997-11-20	2000-05-16	Pharm-Eco Laboratories, Inc.	Synthesis of 11-aryl-5,6-dihydro-11H-dibenz[b,e]azepines
US8119629B2 (en)	2007-10-03	2012-02-21	Bristol-Meyers Squibb Company	Carboxamide GABAA α2 modulators
AU2017313753B2 (en)	2016-08-16	2022-01-27	The Trustees Of Columbia University In The City Of New York	GABA(A) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA755418B (en) *	1974-09-11	1977-06-29	Hoffmann La Roche	Diazepine derivatives
AT361486B (en) *	1975-08-07	1981-03-10	Hoffmann La Roche	METHOD FOR PRODUCING NEW IMIDAZO (1,5 -A) (1,4) DIAZEPINE COMPOUNDS, THEIR SALTS AND OPTICALLY ACTIVE FORMS
US4125726A (en) *	1977-03-11	1978-11-14	Hoffmann-La Roche Inc.	Imidazo[1,5-a][1,4]benzodiazepines
DK151808C (en) *	1982-11-16	1988-06-20	Ferrosan As	ANALOGY PROCEDURE FOR THE PREPARATION OF OXADIAZOLYLIMIDAZO-OE1,4AA-BENZODIAZEPINE DERIVATIVES

1984
- 1984-07-25 ZA ZA845757A patent/ZA845757B/en unknown
- 1984-08-13 EP EP84109639A patent/EP0135770A3/en not_active Withdrawn
- 1984-08-23 NO NO843376A patent/NO843376L/en unknown
- 1984-08-23 NZ NZ209316A patent/NZ209316A/en unknown
- 1984-08-23 IL IL72757A patent/IL72757A0/en unknown
- 1984-08-23 MC MC841721A patent/MC1616A1/en unknown
- 1984-08-23 GR GR80197A patent/GR80197B/en unknown
- 1984-08-24 PT PT79131A patent/PT79131B/en unknown
- 1984-08-24 ES ES535392A patent/ES535392A0/en active Granted
- 1984-08-24 DK DK406384A patent/DK406384A/en not_active Application Discontinuation
- 1984-08-24 AU AU32379/84A patent/AU3237984A/en not_active Abandoned
- 1984-08-24 JP JP59175328A patent/JPS6067480A/en active Pending
- 1984-08-24 KR KR1019840005134A patent/KR850001756A/en not_active Withdrawn
- 1984-08-24 HU HU843179A patent/HU193588B/en unknown
- 1984-08-24 PH PH31144A patent/PH20029A/en unknown
- 1984-08-24 FI FI843356A patent/FI843356A7/en not_active Application Discontinuation
1985
- 1985-05-31 ES ES543717A patent/ES8603433A1/en not_active Expired

Also Published As

Publication number	Publication date
PT79131A (en)	1984-09-01
FI843356A7 (en)	1985-02-26
NZ209316A (en)	1987-04-30
IL72757A0 (en)	1984-11-30
FI843356A0 (en)	1984-08-24
KR850001756A (en)	1985-04-01
HU193588B (en)	1987-10-28
GR80197B (en)	1985-01-03
ES8602700A1 (en)	1985-12-01
ES543717A0 (en)	1986-01-01
NO843376L (en)	1985-02-26
ZA845757B (en)	1985-04-24
EP0135770A2 (en)	1985-04-03
EP0135770A3 (en)	1988-01-13
ES8603433A1 (en)	1986-01-01
DK406384A (en)	1985-02-26
MC1616A1 (en)	1985-07-18
ES535392A0 (en)	1985-12-01
AU3237984A (en)	1985-02-28
JPS6067480A (en)	1985-04-17
HUT34978A (en)	1985-05-28
DK406384D0 (en)	1984-08-24
PT79131B (en)	1986-11-14

Publication	Publication Date	Title
GB8334499D0 (en)	1984-02-01	Derivatives
EP0129513A3 (en)	1985-11-27	Oxamic-acid derivatives
EP0135177A3 (en)	1986-07-16	Benzocycloalkane derivatives
GB8405980D0 (en)	1984-04-11	N-pyridylpyrazole derivatives
GB8416172D0 (en)	1984-08-01	Spirosuccinide derivatives
GB2145084B (en)	1987-01-28	Fredericamycin derivatives
IL72157A0 (en)	1984-10-31	2-alkylthiopenem derivatives
GB8415032D0 (en)	1984-07-18	3-phenyl-4-cyano-pyrrole derivatives
PT79448B (en)	1986-11-13	Pyrazolopyridine-cycloalkanone derivatives
GB2144119B (en)	1986-12-10	Fluoromethylthiooxacephalosporin derivatives
DE3475621D1 (en)	1989-01-19	2-dioxacycloalkylthiopenem derivatives
GR80371B (en)	1985-01-15	3-indolecarboxamide derivatives
ZA845757B (en)	1985-04-24	Benzodiazepine derivatives
GB2146991B (en)	1987-04-15	Fluorenylalkylimidazole derivatives
EG16589A (en)	1989-03-30	2-azacycloalkylthiopenem derivatives
GB2152046B (en)	1987-06-03	2-arylbenzothiazoline derivatives
GB8408128D0 (en)	1984-05-10	Gonadoliberine derivatives
DE3460649D1 (en)	1986-10-16	Cyanotercyclohexane derivatives
AR243155A1 (en)	1993-07-30	Benzoamide derivatives
EP0143001A3 (en)	1986-03-19	Pyrimidoisoquinoline derivatives
GR80582B (en)	1985-02-04	Azolyl-tetrahydrofuran-2-yliden-methan derivatives
GR82491B (en)	1985-04-08	Iminomethyl - azolyl derivatives
GR80442B (en)	1985-01-21	Triazolylmethyl-pyridyloxymethyl-carbinol derivatives
ZA844658B (en)	1986-02-26	2-alkylthiopenem derivatives
GB8402968D0 (en)	1984-03-07	Benzazepine derivatives