PH26584A - Beta-amino-boronic acid derivatives - Google Patents

Beta-amino-boronic acid derivatives Download PDF

Info

Publication number
PH26584A
PH26584A PH39613A PH39613A PH26584A PH 26584 A PH26584 A PH 26584A PH 39613 A PH39613 A PH 39613A PH 39613 A PH39613 A PH 39613A PH 26584 A PH26584 A PH 26584A
Authority
PH
Philippines
Prior art keywords
alkyl
amino
methyl
denotes
formula
Prior art date
Application number
PH39613A
Other languages
English (en)
Inventor
Heinz-Werner Kleeman
Hansjorg Urbach
Dieter Ruppert
Bernward Scholkens
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PH26584A publication Critical patent/PH26584A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH39613A 1988-12-01 1989-11-29 Beta-amino-boronic acid derivatives PH26584A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3840452A DE3840452A1 (de) 1988-12-01 1988-12-01 (beta)-amino-boronsaeure-derivate

Publications (1)

Publication Number Publication Date
PH26584A true PH26584A (en) 1992-08-19

Family

ID=6368210

Family Applications (1)

Application Number Title Priority Date Filing Date
PH39613A PH26584A (en) 1988-12-01 1989-11-29 Beta-amino-boronic acid derivatives

Country Status (14)

Country Link
EP (1) EP0371467A3 (ja)
JP (1) JPH02193997A (ja)
KR (1) KR900009663A (ja)
AU (1) AU616819B2 (ja)
CA (1) CA2004303A1 (ja)
DE (1) DE3840452A1 (ja)
DK (1) DK605489A (ja)
FI (1) FI895718A7 (ja)
IL (1) IL92497A0 (ja)
NO (1) NO894790L (ja)
NZ (1) NZ231578A (ja)
PH (1) PH26584A (ja)
PT (1) PT92442A (ja)
ZA (1) ZA899152B (ja)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL90244A (en) * 1988-05-11 1993-05-13 Du Pont Merck Pharma Peptide-drug compositions, for buccal and nasal administration, containing :-aminoboronic acid derivatives
US4983589A (en) * 1989-12-14 1991-01-08 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes and derivatives thereof
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
GB9024775D0 (en) * 1990-11-14 1991-01-02 Axis Research Chemical compounds
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
US6825169B1 (en) 1991-10-22 2004-11-30 Trustees Of Tufts College Inhibitors of dipeptidyl-aminopeptidase type IV
US5888992A (en) * 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
ATE253050T1 (de) 1992-03-11 2003-11-15 Narhex Ltd Aminderivate von oxo- und hydroxy- substituierten kohlenwasserstoffen
US6071895A (en) * 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
JPH07504654A (ja) * 1992-03-11 1995-05-25 ナルヘックス　リミテッド オキソ及びヒドロキシ置換炭化水素のアミン誘導体
US5559256A (en) * 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
WO1994004543A1 (en) * 1992-08-14 1994-03-03 The Procter & Gamble Company PROCESS FOR SYNTHESIZING A β-AMINOALKYLBORONIC ACID AND ESTER
US5442100A (en) * 1992-08-14 1995-08-15 The Procter & Gamble Company β-aminoalkyl and β-N-peptidylaminoalkyl boronic acids
US5354491A (en) * 1992-08-14 1994-10-11 The Procter & Gamble Company Liquid detergent compositions containing protease and certain β-aminoalkylboronic acids and esters
TR28578A (tr) * 1993-08-13 1996-11-04 Procter & Gamble Proteaz ve bazi ›-aminoalkilboronik asit ve esterlerini ihtiva eden sivi deterjan bilesimleri.
IL110898A0 (en) * 1993-09-10 1994-11-28 Narhex Australia Pty Ltd Polar-substituted hydrocarbons
US5431842A (en) * 1993-11-05 1995-07-11 The Procter & Gamble Company Liquid detergents with ortho-substituted phenylboronic acids for inhibition of proteolytic enzyme
US5965532A (en) 1996-06-28 1999-10-12 Trustees Of Tufts College Multivalent compounds for crosslinking receptors and uses thereof
US6040145A (en) 1997-05-07 2000-03-21 Tufts University Potentiation of the immune response
US6100234A (en) * 1997-05-07 2000-08-08 Tufts University Treatment of HIV
ATE357509T1 (de) 1997-09-29 2007-04-15 Point Therapeutics Inc Stimulierung von hämatopoietischen zellen im vitro
IL139247A0 (en) 1998-05-04 2001-11-25 Point Therapeutics Inc Hematopoietic stimulation
US6979697B1 (en) 1998-08-21 2005-12-27 Point Therapeutics, Inc. Regulation of substrate activity
US6890904B1 (en) 1999-05-25 2005-05-10 Point Therapeutics, Inc. Anti-tumor agents
CA2862710A1 (en) * 2012-01-09 2013-07-18 University Of Tromso Therapeutic boron-containing compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides

Also Published As

Publication number Publication date
KR900009663A (ko) 1990-07-05
DK605489A (da) 1990-06-02
DE3840452A1 (de) 1990-06-07
NO894790L (no) 1990-06-05
AU616819B2 (en) 1991-11-07
AU4566589A (en) 1990-06-07
JPH02193997A (ja) 1990-07-31
NO894790D0 (no) 1989-11-30
NZ231578A (en) 1992-02-25
PT92442A (pt) 1990-06-29
EP0371467A3 (de) 1991-04-03
EP0371467A2 (de) 1990-06-06
FI895718A0 (fi) 1989-11-29
IL92497A0 (en) 1990-08-31
DK605489D0 (da) 1989-11-30
CA2004303A1 (en) 1990-06-01
ZA899152B (en) 1990-09-26
FI895718A7 (fi) 1990-06-02

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