PL1691808T3 - Kompozycja farmaceutyczna pochodnej pirazolo-3-karboksyamidu do podawania doustnego - Google Patents

Kompozycja farmaceutyczna pochodnej pirazolo-3-karboksyamidu do podawania doustnego

Info

Publication number
PL1691808T3
PL1691808T3 PL04805418T PL04805418T PL1691808T3 PL 1691808 T3 PL1691808 T3 PL 1691808T3 PL 04805418 T PL04805418 T PL 04805418T PL 04805418 T PL04805418 T PL 04805418T PL 1691808 T3 PL1691808 T3 PL 1691808T3
Authority
PL
Poland
Prior art keywords
pyrazol
pharmaceutical composition
oral administration
carboxamide derivative
carboxamide
Prior art date
Application number
PL04805418T
Other languages
English (en)
Inventor
Thierry Breul
Jean Claude Gautier
Olivier Saslawski
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of PL1691808T3 publication Critical patent/PL1691808T3/pl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL04805418T 2003-11-10 2004-11-09 Kompozycja farmaceutyczna pochodnej pirazolo-3-karboksyamidu do podawania doustnego PL1691808T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0313259A FR2861992B1 (fr) 2003-11-10 2003-11-10 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
EP04805418A EP1691808B1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide
PCT/FR2004/002875 WO2005046690A1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3­carboxamide

Publications (1)

Publication Number Publication Date
PL1691808T3 true PL1691808T3 (pl) 2009-09-30

Family

ID=34508418

Family Applications (1)

Application Number Title Priority Date Filing Date
PL04805418T PL1691808T3 (pl) 2003-11-10 2004-11-09 Kompozycja farmaceutyczna pochodnej pirazolo-3-karboksyamidu do podawania doustnego

Country Status (27)

Country Link
US (2) US20060264469A1 (pl)
EP (1) EP1691808B1 (pl)
JP (1) JP4767171B2 (pl)
KR (1) KR20060108668A (pl)
CN (1) CN100528158C (pl)
AR (1) AR047237A1 (pl)
AT (1) ATE429227T1 (pl)
AU (1) AU2004289086A1 (pl)
BR (1) BRPI0416341A (pl)
CA (1) CA2544413A1 (pl)
CY (1) CY1110478T1 (pl)
DE (1) DE602004020797D1 (pl)
DK (1) DK1691808T3 (pl)
ES (1) ES2325373T3 (pl)
FR (1) FR2861992B1 (pl)
HR (1) HRP20090393T1 (pl)
IL (1) IL175556A (pl)
MA (1) MA28419B1 (pl)
NO (1) NO20062609L (pl)
NZ (1) NZ547763A (pl)
PL (1) PL1691808T3 (pl)
PT (1) PT1691808E (pl)
RU (1) RU2321404C1 (pl)
SI (1) SI1691808T1 (pl)
TW (1) TWI280129B (pl)
WO (1) WO2005046690A1 (pl)
ZA (1) ZA200604451B (pl)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1880715A1 (en) 2006-07-19 2008-01-23 Abbott GmbH & Co. KG Pharmaceutically acceptable solubilizing composition and pharmaceutical dosage form containing same
EP1920767A1 (en) * 2006-11-09 2008-05-14 Abbott GmbH & Co. KG Melt-processed imatinib dosage form
KR101493546B1 (ko) * 2007-08-21 2015-02-16 바실리어 파마슈티카 아게 항균 조성물
MY158809A (en) * 2010-09-22 2016-11-15 Craun Res Sdn Bhd Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same
US20130317117A1 (en) * 2010-11-24 2013-11-28 Pharmaceutics International, Inc. Self micro-emulsifying drug delivery system with increased bioavailability

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059691A (en) * 1990-01-22 1991-10-22 American Cyanamid Company N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
DK1033128T4 (da) * 1993-09-28 2012-03-19 Scherer Gmbh R P Blød gelatinekapselfremstilling
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
JPH11504028A (ja) * 1995-04-24 1999-04-06 イースム リサーチ ディベロップメント カンパニー オブ ザ ヒーブル ユニバーシティ オブ エルサレム 油/水エマルジョンを作り出す自己乳化性配合物
EP0825849A1 (en) * 1995-05-19 1998-03-04 Abbott Laboratories Self-emulsifying formulations of lipophilic drugs
US5993858A (en) * 1996-06-14 1999-11-30 Port Systems L.L.C. Method and formulation for increasing the bioavailability of poorly water-soluble drugs
BR9808845A (pt) * 1997-03-14 2000-08-01 Otsuka Pharma Co Ltd Derivado de pirimidina, agentes para a cura de uma doença alérgica, da asma e de uma dermatite atópica, agentes para inibição da produção de no de tnf-alfa, de citoquinas e da 5-lipoxigenase, processos para curar uma doença alérgica, a asma e uma dermatite atópica e para inibir a produção de no, de tnf-alfa e de citoquinas e a 5-lipoxigenase e usos de um composto
FR2761266B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
FR2761265B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
US6617426B1 (en) * 1999-06-22 2003-09-09 Merck & Co Inc Cysteinyl protease inhibitors
JP2001151669A (ja) * 1999-11-24 2001-06-05 Nippon Kayaku Co Ltd 経口用自己乳化製剤
YU43702A (sh) * 1999-12-23 2004-11-25 Pfizer Products Inc. Farmaceutske kompozicije koje obezbeđuju povećanje koncentracije leka
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
ES2283756T3 (es) * 2002-03-01 2007-11-01 Novagali Pharma Sa Sistemas autoemulsionantes de administracion de farmaco para taxoides.
GB0216700D0 (en) * 2002-07-18 2002-08-28 Astrazeneca Ab Process

Also Published As

Publication number Publication date
TW200524597A (en) 2005-08-01
ATE429227T1 (de) 2009-05-15
MA28419B1 (fr) 2007-02-01
NZ547763A (en) 2009-08-28
AR047237A1 (es) 2006-01-11
RU2006120447A (ru) 2007-12-20
US20060264469A1 (en) 2006-11-23
CA2544413A1 (fr) 2005-05-26
FR2861992B1 (fr) 2007-07-20
CN1925856A (zh) 2007-03-07
ES2325373T3 (es) 2009-09-02
IL175556A0 (en) 2008-04-13
IL175556A (en) 2010-11-30
NO20062609L (no) 2006-06-06
US20090004261A1 (en) 2009-01-01
CY1110478T1 (el) 2015-04-29
TWI280129B (en) 2007-05-01
ZA200604451B (en) 2007-10-31
JP4767171B2 (ja) 2011-09-07
AU2004289086A1 (en) 2005-05-26
SI1691808T1 (sl) 2009-10-31
RU2321404C1 (ru) 2008-04-10
HK1102021A1 (en) 2007-11-02
DE602004020797D1 (de) 2009-06-04
WO2005046690A1 (fr) 2005-05-26
FR2861992A1 (fr) 2005-05-13
JP2007516960A (ja) 2007-06-28
EP1691808A1 (fr) 2006-08-23
HRP20090393T1 (en) 2009-08-31
EP1691808B1 (fr) 2009-04-22
DK1691808T3 (da) 2009-08-03
KR20060108668A (ko) 2006-10-18
PT1691808E (pt) 2009-07-14
CN100528158C (zh) 2009-08-19
BRPI0416341A (pt) 2007-02-27

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