PL199603A1 - METHOD OF MAKING NEW DERIVATIVES OF PYROLOCARBOXYLIC ACID-1 - Google Patents

METHOD OF MAKING NEW DERIVATIVES OF PYROLOCARBOXYLIC ACID-1

Info

Publication number: PL199603A1
Authority: PL; Poland
Prior art keywords: pyrolocarboxylic; acid; new derivatives; making new; making
Prior art date: 1976-07-14

Application number

PL19960377A

Other languages

Polish (pl)

Other versions

PL109390B1 (en

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1977-07-13

Publication date

1978-04-24

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL199603(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1977-02-23 Priority claimed from US05/771,286 external-priority patent/US4089969A/en

1977-07-13 Application filed by Syntex Inc filed Critical Syntex Inc

1978-04-24 Publication of PL199603A1 publication Critical patent/PL199603A1/en

1980-05-31 Publication of PL109390B1 publication Critical patent/PL109390B1/en

Links

238000004519 manufacturing process Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)

PL1977199603A 1976-07-14 1977-07-13 Method of producing new derivatives of pyrolocarboxylic-1 acid PL109390B1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70490976A	1976-07-14	1976-07-14
US05/771,286 US4089969A (en)	1976-07-14	1977-02-23	5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (2)

Publication Number	Publication Date
PL199603A1 true PL199603A1 (en)	1978-04-24
PL109390B1 PL109390B1 (en)	1980-05-31

Family

ID=27107410

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
PL1977227290A PL124444B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrrole-1-carboxylic acid
PL1977199603A PL109390B1 (en)	1976-07-14	1977-07-13	Method of producing new derivatives of pyrolocarboxylic-1 acid
PL1977227291A PL124445B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrrole-1-carboxylic acid
PL1977227289A PL124711B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrolo-1-carboxylic acid

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
PL1977227290A PL124444B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrrole-1-carboxylic acid

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
PL1977227291A PL124445B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrrole-1-carboxylic acid
PL1977227289A PL124711B1 (en)	1976-07-14	1977-07-13	Process for preparing novel derivatives of pyrolo-1-carboxylic acid

Country Status (27)

Country	Link
JP (1)	JPS539788A (en)
AR (1)	AR224997A1 (en)
CA (1)	CA1102809A (en)
CH (3)	CH641458A5 (en)
CS (1)	CS204954B2 (en)
DE (2)	DE2760330C2 (en)
DK (1)	DK151886C (en)
ES (2)	ES460706A1 (en)
FI (1)	FI63406C (en)
FR (2)	FR2358406A1 (en)
GB (1)	GB1554075A (en)
GR (1)	GR61111B (en)
HK (1)	HK15981A (en)
HU (1)	HU174224B (en)
IE (1)	IE45253B1 (en)
IL (2)	IL52493A (en)
IT (1)	IT1117313B (en)
MX (1)	MX163202B (en)
MY (1)	MY8100357A (en)
NL (2)	NL186318C (en)
NO (1)	NO147564C (en)
NZ (1)	NZ184610A (en)
PL (4)	PL124444B1 (en)
PT (1)	PT66780B (en)
SE (1)	SE434643B (en)
SU (1)	SU695558A3 (en)
YU (1)	YU40816B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) *	1979-03-19	1980-09-25	Sohachi Takeuchi	Manufacturing method of tubular vessel
US4344943A (en) *	1980-06-09	1982-08-17	Syntex (U.S.A.) Inc.	6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (en) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (en) *	1987-09-10	1995-05-01	久光製薬株式会社	Novel 3-aroyl-6,7-dihydro-5H-pyrrolo [1,2-c] imidazole-7-carboxylic acid derivative
JP2649168B2 (en) *	1988-02-25	1997-09-03	久光製薬株式会社	Novel 5,6-diphenyl-1,2-dihydro-3H-pyrrolo [1,2-a] pyrrole-1-carboxylic acid derivatives
IT1250691B (en) *	1991-07-22	1995-04-21	Giancarlo Santus	THERAPEUTIC COMPOSITIONS FOR INTRANASAL ADMINISTRATION INCLUDING KETOROLAC.
EP0612521B1 (en) *	1991-11-11	1999-06-30	Hisamitsu Pharmaceutical Co., Inc.	Fomentation containing ketorolac
DE4300697C1 (en) *	1993-01-13	1994-05-19	Roemmers Sa	New 2-pyrrolidino-ethyl ester of ketorolac - useful as analgesic, antiinflammatory and antipyretic agent with low ulcerogenicity
US5622948A (en) *	1994-12-01	1997-04-22	Syntex (U.S.A.) Inc.	Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (en) *	2007-02-27	2008-09-11	Okamura Corp	Lighting device for merchandise display shelf
CA3202461A1 (en) *	2020-12-16	2022-06-23	Robert T. Streeper	Dicarboxylic acid esters for inducing an analgesic effect

1977
- 1977-05-17 JP JP5697777A patent/JPS539788A/en active Granted
- 1977-07-07 DK DK307577A patent/DK151886C/en active
- 1977-07-07 AR AR268356A patent/AR224997A1/en active
- 1977-07-07 GR GR53907A patent/GR61111B/en unknown
- 1977-07-08 IL IL52493A patent/IL52493A/en unknown
- 1977-07-08 PT PT66780A patent/PT66780B/en unknown
- 1977-07-08 CH CH850077A patent/CH641458A5/en not_active IP Right Cessation
- 1977-07-08 NL NLAANVRAGE7707651,A patent/NL186318C/en not_active IP Right Cessation
- 1977-07-08 IE IE1423/77A patent/IE45253B1/en not_active IP Right Cessation
- 1977-07-11 GB GB28919/77A patent/GB1554075A/en not_active Expired
- 1977-07-11 YU YU1721/77A patent/YU40816B/en unknown
- 1977-07-11 FR FR7721356A patent/FR2358406A1/en active Granted
- 1977-07-11 FI FI772153A patent/FI63406C/en not_active IP Right Cessation
- 1977-07-11 NZ NZ184610A patent/NZ184610A/en unknown
- 1977-07-12 CA CA282,599A patent/CA1102809A/en not_active Expired
- 1977-07-12 CS CS774646A patent/CS204954B2/en unknown
- 1977-07-13 ES ES460706A patent/ES460706A1/en not_active Expired
- 1977-07-13 DE DE2760330A patent/DE2760330C2/de not_active Expired
- 1977-07-13 PL PL1977227290A patent/PL124444B1/en unknown
- 1977-07-13 SU SU772501050A patent/SU695558A3/en active
- 1977-07-13 DE DE19772731678 patent/DE2731678A1/en active Granted
- 1977-07-13 SE SE7708141A patent/SE434643B/en not_active IP Right Cessation
- 1977-07-13 IT IT68630/77A patent/IT1117313B/en active Protection Beyond IP Right Term
- 1977-07-13 PL PL1977199603A patent/PL109390B1/en unknown
- 1977-07-13 PL PL1977227291A patent/PL124445B1/en unknown
- 1977-07-13 PL PL1977227289A patent/PL124711B1/en unknown
- 1977-07-13 NO NO772494A patent/NO147564C/en unknown
- 1977-07-14 HU HU77SI1582A patent/HU174224B/en unknown
- 1977-12-20 FR FR7738508A patent/FR2375234A1/en active Granted
1978
- 1978-05-24 ES ES470214A patent/ES470214A1/en not_active Expired
1979
- 1979-11-22 IL IL58779A patent/IL58779A0/en unknown
1981
- 1981-04-23 HK HK159/81A patent/HK15981A/en unknown
- 1981-12-30 MY MY357/81A patent/MY8100357A/en unknown
1984
- 1984-02-22 CH CH86584A patent/CH646972A5/en not_active IP Right Cessation
- 1984-02-22 CH CH86684A patent/CH646973A5/en not_active IP Right Cessation
1991
- 1991-07-05 MX MX9100104A patent/MX163202B/en unknown
1993
- 1993-03-23 NL NL930021C patent/NL930021I2/en unknown

Also Published As

Publication number	Publication date
NL930021I2 (en)	1997-03-03
SE434643B (en)	1984-08-06
SU695558A3 (en)	1979-10-30
NL186318C (en)	1990-11-01
IT1117313B (en)	1986-02-17
CA1102809A (en)	1981-06-09
FR2358406B1 (en)	1981-04-17
FR2375234A1 (en)	1978-07-21
GB1554075A (en)	1979-10-17
FI63406B (en)	1983-02-28
NZ184610A (en)	1979-03-28
NO147564B (en)	1983-01-24
NL930021I1 (en)	1993-05-03
AU2697577A (en)	1979-01-18
FI772153A7 (en)	1978-01-15
IE45253L (en)	1978-01-14
DE2731678C2 (en)	1989-06-08
FR2358406A1 (en)	1978-02-10
FR2375234B1 (en)	1980-11-07
MX163202B (en)	1992-02-20
MY8100357A (en)	1981-12-31
NO772494L (en)	1978-01-17
DK307577A (en)	1978-01-15
JPS6254109B2 (en)	1987-11-13
ES460706A1 (en)	1978-12-01
NL186318B (en)	1990-06-01
YU172177A (en)	1983-09-30
PT66780A (en)	1977-08-01
PL124711B1 (en)	1983-02-28
NL7707651A (en)	1978-01-17
HK15981A (en)	1981-05-01
DE2760330C2 (en)	1989-06-15
CS204954B2 (en)	1981-04-30
IL58779A0 (en)	1980-02-29
PL124444B1 (en)	1983-01-31
AU513384B2 (en)	1980-11-27
DK151886C (en)	1988-06-06
YU40816B (en)	1986-06-30
NO147564C (en)	1983-05-18
DK151886B (en)	1988-01-11
DE2731678A1 (en)	1978-03-16
CH646972A5 (en)	1984-12-28
SE7708141L (en)	1978-01-15
CH641458A5 (en)	1984-02-29
IL52493A (en)	1982-02-28
HU174224B (en)	1979-11-28
ES470214A1 (en)	1979-09-16
CH646973A5 (en)	1984-12-28
PT66780B (en)	1978-12-18
PL109390B1 (en)	1980-05-31
IE45253B1 (en)	1982-07-14
FI63406C (en)	1983-06-10
IL52493A0 (en)	1977-10-31
GR61111B (en)	1978-09-12
PL124445B1 (en)	1983-01-31
AR224997A1 (en)	1982-02-15
JPS539788A (en)	1978-01-28

Publication	Publication Date	Title
PL195997A1 (en)	1978-02-27	METHOD OF MAKING NEW CARBOXYALKYLOACYLOAMINO ACID DERIVATIVES
PL201586A1 (en)	1978-09-25	METHOD OF MAKING NEW SPIRO-HYDANTION COMPOUNDS
PL196505A1 (en)	1979-06-18	METHOD OF MAKING NEW AMINO-ALKYLETERCYCLIC COMPOUNDS
PL201286A1 (en)	1978-12-04	METHOD OF MAKING NEW 1-ARYLOXY-2-HYDROXY-3-ALKYLENE-AMINOPROPANE
PL199603A1 (en)	1978-04-24	METHOD OF MAKING NEW DERIVATIVES OF PYROLOCARBOXYLIC ACID-1
PL215008A1 (en)	1979-12-17	METHOD OF MAKING PIRANONE-3 DERIVATIVES
PL197005A1 (en)	1978-10-09	METHOD OF MAKING NEW PROSTAGLANDIN DERIVATIVES
PL210045A1 (en)	1979-06-18	METHOD OF MAKING NEW FOUREPEPTIDE DERIVATIVES
PL200685A1 (en)	1978-10-09	METHOD OF MAKING NEW URACYL DERIVATIVES
PL197372A1 (en)	1979-06-18	METHOD OF MAKING CANAMYCIN DERIVATIVES
PL204134A1 (en)	1979-07-02	METHOD OF MAKING NEW AMINO-ALCOXYPHENYL DERIVATIVES
PL193183A1 (en)	1978-03-28	METHOD OF MAKING NEW DERIVATIVES OF 11-DESOXY-16-ARYL-OMEGA-TETRANOR-PROSTAGLANDINE
PL200583A1 (en)	1979-06-04	METHOD OF MAKING NEW BENZOPIRANE DERIVATIVES
PL200534A1 (en)	1978-05-22	METHOD OF MAKING NEW OXADESTIACHALOSPORINES
PL200605A1 (en)	1979-02-12	METHOD OF MAKING NEW METHIONINOENKEPHALIN DERIVATIVES
PL198878A1 (en)	1978-04-10	METHOD OF MAKING 2-CHLOROSULFINYLAZETHIDINONE DERIVATIVES
PL199364A1 (en)	1978-04-10	METHOD OF MANUFACTURING NEW DERIVATIVES OF BENZOXICINE
PL206456A1 (en)	1979-04-23	METHOD OF MAKING PYRIDAZINONE-3 DERIVATIVES
PL199602A1 (en)	1979-01-29	METHOD OF OBTAINING NEW DERIVATIVES OF PYROLOCARBOXYLIC ACID-1
PL208434A1 (en)	1979-06-04	METHOD OF MAKING NEW BENZOPIRANE DERIVATIVES
PL206833A1 (en)	1979-04-23	METHOD OF MAKING NEW DERIVATIVES OF 6-AMINOPENAM
PL197045A1 (en)	1978-02-13	METHOD OF MAKING NEW URACYL DERIVATIVES
PL202660A1 (en)	1978-08-28	METHOD OF MAKING NEW DERIVATIVES OF SPIROOXAZOLIDYNODION
PL211328A1 (en)	1979-08-13	METHOD OF MAKING NEW PHENOXYALKANOLAMINE DERIVATIVES
PL201133A1 (en)	1978-07-31	METHOD OF MAKING NEW PIRYDOBENZODWUAZEPINONOV