PL2024372T3 - Pochodna tieno[3,2-D]pirymidyny użyteczna jako inibitor PI3K - Google Patents

Pochodna tieno[3,2-D]pirymidyny użyteczna jako inibitor PI3K

Info

Publication number
PL2024372T3
PL2024372T3 PL07734376T PL07734376T PL2024372T3 PL 2024372 T3 PL2024372 T3 PL 2024372T3 PL 07734376 T PL07734376 T PL 07734376T PL 07734376 T PL07734376 T PL 07734376T PL 2024372 T3 PL2024372 T3 PL 2024372T3
Authority
PL
Poland
Prior art keywords
thieno
pi3k inhibitor
pyrimidine derivative
derivative useful
useful
Prior art date
Application number
PL07734376T
Other languages
English (en)
Inventor
Irina Chuckowree
Adrian FOLKES
Tim Hancox
Stephen Shuttleworth
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority claimed from PCT/IB2007/001058 external-priority patent/WO2007129161A2/en
Publication of PL2024372T3 publication Critical patent/PL2024372T3/pl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355—Non-condensed oxazines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
PL07734376T 2006-04-26 2007-04-24 Pochodna tieno[3,2-D]pirymidyny użyteczna jako inibitor PI3K PL2024372T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79496606P 2006-04-26 2006-04-26
PCT/IB2007/001058 WO2007129161A2 (en) 2006-04-26 2007-04-24 Thieno [3, 2-d] pyrimidine derivative useful as pi3k inhibitor
EP07734376A EP2024372B1 (en) 2006-04-26 2007-04-24 Thieno[3,2-d]pyrimidine derivative useful as pi3k inhibitor

Publications (1)

Publication Number Publication Date
PL2024372T3 true PL2024372T3 (pl) 2010-11-30

Family

ID=43034244

Family Applications (1)

Application Number Title Priority Date Filing Date
PL07734376T PL2024372T3 (pl) 2006-04-26 2007-04-24 Pochodna tieno[3,2-D]pirymidyny użyteczna jako inibitor PI3K

Country Status (3)

Country Link
EP (2) EP2246354A1 (pl)
PL (1) PL2024372T3 (pl)
SI (1) SI2024372T1 (pl)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3773919A (en) 1969-10-23 1973-11-20 Du Pont Polylactide-drug mixtures
AU5261001A (en) 2000-04-27 2001-11-12 Imperial Cancer Research Technology Ltd Condensed heteroaryl derivatives
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
AU2002357667A1 (en) * 2001-10-24 2003-05-06 Iconix Pharmaceuticals, Inc. Modulators of phosphoinositide 3-kinase
WO2005007083A2 (en) * 2003-06-18 2005-01-27 Smithkline Beecham Corporation Chemical compounds
EP1682123A1 (en) * 2003-11-07 2006-07-26 SmithKline Beecham (Cork) Limited Cancer treatment method
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds

Also Published As

Publication number Publication date
EP2246354A1 (en) 2010-11-03
SI2024372T1 (sl) 2010-10-29
EP2024372A2 (en) 2009-02-18
EP2024372B1 (en) 2010-06-23

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