PL2148873T3 - Pochodne 4-alkoksypirydazynowe jako szybko dysocjujący antagoniści receptora dopaminowego 2 - Google Patents

Pochodne 4-alkoksypirydazynowe jako szybko dysocjujący antagoniści receptora dopaminowego 2

Info

Publication number: PL2148873T3
Authority: PL; Poland
Prior art keywords: alkoxypyridazine; derivatives; receptor antagonists; fast dissociating; dissociating dopamine
Prior art date: 2007-04-23

Application number

PL08749604T

Other languages

English (en)

Inventor

Gregor James Macdonald

José Manuel Bartolomé-Nebreda

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-04-23

Filing date

2008-04-18

Publication date

2013-01-31

2008-04-18 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2013-01-31 Publication of PL2148873T3 publication Critical patent/PL2148873T3/pl

Links

VYFYYTLLBUKUHU-UHFFFAOYSA-N dopamine Chemical compound NCCC1=CC=C(O)C(O)=C1 VYFYYTLLBUKUHU-UHFFFAOYSA-N 0.000 title 2
229960003638 dopamine Drugs 0.000 title 1
239000002464 receptor antagonist Substances 0.000 title 1
229940044551 receptor antagonist Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Diabetes (AREA)
Addiction (AREA)
Endocrinology (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

PL08749604T 2007-04-23 2008-04-18 Pochodne 4-alkoksypirydazynowe jako szybko dysocjujący antagoniści receptora dopaminowego 2 PL2148873T3 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP07106704		2007-04-23
EP08749604A EP2148873B1 (en)	2007-04-23	2008-04-18	4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists
PCT/EP2008/054731 WO2008128995A1 (en)	2007-04-23	2008-04-18	4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists

Publications (1)

Publication Number	Publication Date
PL2148873T3 true PL2148873T3 (pl)	2013-01-31

Family

ID=38476156

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL08749604T PL2148873T3 (pl)	2007-04-23	2008-04-18	Pochodne 4-alkoksypirydazynowe jako szybko dysocjujący antagoniści receptora dopaminowego 2

Country Status (19)

Country	Link
US (1)	US8906921B2 (pl)
EP (1)	EP2148873B1 (pl)
JP (1)	JP5431305B2 (pl)
KR (1)	KR20100016620A (pl)
CN (1)	CN101663292A (pl)
AU (1)	AU2008240728B2 (pl)
CA (1)	CA2683111A1 (pl)
CY (1)	CY1113820T1 (pl)
DK (1)	DK2148873T3 (pl)
ES (1)	ES2393818T3 (pl)
HR (1)	HRP20120913T1 (pl)
IL (1)	IL201663A (pl)
MX (1)	MX2009011415A (pl)
PL (1)	PL2148873T3 (pl)
PT (1)	PT2148873E (pl)
RS (1)	RS52518B (pl)
RU (1)	RU2464268C2 (pl)
SI (1)	SI2148873T1 (pl)
WO (1)	WO2008128995A1 (pl)

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EP2310374B1 (en) *	2008-07-03	2012-10-31	Janssen Pharmaceutica N.V.	Substituted 6- (1-piperazinyl) -pyridazines as 5-ht6 receptor antagonists
EP2307374B1 (en)	2008-07-31	2017-01-25	Janssen Pharmaceutica NV	Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists

2008
- 2008-04-18 JP JP2010504647A patent/JP5431305B2/ja active Active
- 2008-04-18 CN CN200880012952A patent/CN101663292A/zh active Pending
- 2008-04-18 CA CA002683111A patent/CA2683111A1/en not_active Abandoned
- 2008-04-18 PL PL08749604T patent/PL2148873T3/pl unknown
- 2008-04-18 AU AU2008240728A patent/AU2008240728B2/en not_active Ceased
- 2008-04-18 KR KR1020097023941A patent/KR20100016620A/ko not_active Ceased
- 2008-04-18 HR HRP20120913AT patent/HRP20120913T1/hr unknown
- 2008-04-18 PT PT08749604T patent/PT2148873E/pt unknown
- 2008-04-18 US US12/597,166 patent/US8906921B2/en active Active
- 2008-04-18 WO PCT/EP2008/054731 patent/WO2008128995A1/en not_active Ceased
- 2008-04-18 RS RS20120481A patent/RS52518B/sr unknown
- 2008-04-18 DK DK08749604.8T patent/DK2148873T3/da active
- 2008-04-18 SI SI200830823T patent/SI2148873T1/sl unknown
- 2008-04-18 RU RU2009142997/04A patent/RU2464268C2/ru active
- 2008-04-18 MX MX2009011415A patent/MX2009011415A/es active IP Right Grant
- 2008-04-18 EP EP08749604A patent/EP2148873B1/en active Active
- 2008-04-18 ES ES08749604T patent/ES2393818T3/es active Active
2009
- 2009-10-21 IL IL201663A patent/IL201663A/en active IP Right Grant
2012
- 2012-11-28 CY CY20121101154T patent/CY1113820T1/el unknown

Also Published As

Publication number	Publication date
CN101663292A (zh)	2010-03-03
US8906921B2 (en)	2014-12-09
RS52518B (sr)	2013-04-30
EP2148873A1 (en)	2010-02-03
KR20100016620A (ko)	2010-02-12
US20100063058A1 (en)	2010-03-11
SI2148873T1 (sl)	2013-01-31
CA2683111A1 (en)	2008-10-30
EP2148873B1 (en)	2012-08-29
IL201663A (en)	2013-05-30
RU2464268C2 (ru)	2012-10-20
JP5431305B2 (ja)	2014-03-05
RU2009142997A (ru)	2011-05-27
CY1113820T1 (el)	2016-10-05
AU2008240728B2 (en)	2013-01-10
HRP20120913T1 (hr)	2012-12-31
PT2148873E (pt)	2012-11-20
IL201663A0 (en)	2010-05-31
JP2010525014A (ja)	2010-07-22
DK2148873T3 (da)	2012-11-26
MX2009011415A (es)	2009-11-05
ES2393818T3 (es)	2012-12-28
AU2008240728A1 (en)	2008-10-30
WO2008128995A1 (en)	2008-10-30

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