PL2477990T3 - Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne - Google Patents

Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne

Info

Publication number: PL2477990T3
Authority: PL; Poland
Prior art keywords: phenyl; preparation; therapeutic use; pyrazolopyridine derivatives; pyrazolopyridine
Prior art date: 2009-09-18

Application number

PL10771159T

Other languages

English (en)

Inventor

Florian Auger

Peretti Danielle De

Luc Even

Original Assignee

Sanofi Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2009-09-18

Filing date

2010-09-17

Publication date

2015-02-27

2010-09-17 Application filed by Sanofi Sa filed Critical Sanofi Sa

2015-02-27 Publication of PL2477990T3 publication Critical patent/PL2477990T3/pl

Links

FXUDQKREGGIUQW-UHFFFAOYSA-N 5-phenyl-1h-pyrazolo[4,3-b]pyridine Chemical class N1=C2C=NNC2=CC=C1C1=CC=CC=C1 FXUDQKREGGIUQW-UHFFFAOYSA-N 0.000 title 1
230000001225 therapeutic effect Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Physical Education & Sports Medicine (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Addiction (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

PL10771159T 2009-09-18 2010-09-17 Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne PL2477990T3 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR0956444A FR2950344B1 (fr)	2009-09-18	2009-09-18	Derives de 5-phenyl-pyrazolopyridine, leur preparation et leur aplication en therapeutique.
EP10771159.0A EP2477990B1 (fr)	2009-09-18	2010-09-17	Dérivés de 5-phenyl-pyrazolopyridine, leur préparation et leur application en thérapeutique
PCT/FR2010/051932 WO2011033230A1 (fr)	2009-09-18	2010-09-17	Dérivés de 5-phenyl-pyrazolopyridine, leur préparation et leur application en thérapeutique

Publications (1)

Publication Number	Publication Date
PL2477990T3 true PL2477990T3 (pl)	2015-02-27

Family

ID=41572488

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL10771159T PL2477990T3 (pl)	2009-09-18	2010-09-17	Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne

Country Status (16)

Country	Link
US (1)	US8618301B2 (pl)
EP (1)	EP2477990B1 (pl)
JP (1)	JP5616453B2 (pl)
AR (1)	AR078180A1 (pl)
CY (1)	CY1116581T1 (pl)
DK (1)	DK2477990T3 (pl)
ES (1)	ES2523505T3 (pl)
FR (1)	FR2950344B1 (pl)
HR (1)	HRP20141119T1 (pl)
JO (1)	JO3017B1 (pl)
PL (1)	PL2477990T3 (pl)
PT (1)	PT2477990E (pl)
SI (1)	SI2477990T1 (pl)
TW (1)	TWI464169B (pl)
UY (1)	UY32894A (pl)
WO (1)	WO2011033230A1 (pl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2953520B1 (fr) *	2009-12-04	2011-11-25	Sanofi Aventis	Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique
EP4370518A1 (en) *	2021-07-16	2024-05-22	Sanofi	Imidazo[1,2-b][1,2,4]triazol derivatives for use in therapy
WO2023285465A1 (en) *	2021-07-16	2023-01-19	Sanofi	6h-imidazo[1,2-a]pyrrolo[2,3-e]pyridine derivatives for use in therapy

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL214231B1 (pl) *	2001-04-27	2013-07-31	Eisai R & D Man Co	Pochodne pirazolo [1,5-a] pirydyny, kompozycje je zawierajace oraz zastosowanie
CA2478715A1 (en) *	2002-03-13	2003-09-25	Pharmacia & Upjohn Company	Novel pyrazolo [1,5-a]pyridine derivatives and their use as neurotransmitter modulators
JP4890439B2 (ja) *	2005-03-07	2012-03-07	杏林製薬株式会社	ピラゾロピリジン−４−イルピリダジノン誘導体とその付加塩及びそれらを有効成分とするｐｄｅ阻害剤
FR2906250B1 (fr) *	2006-09-22	2008-10-31	Sanofi Aventis Sa	Derives de 2-aryl-6phenyl-imidazo(1,2-a) pyridines, leur preparation et leur application en therapeutique
JP5442449B2 (ja) *	2006-12-22	2014-03-12	アステックス、セラピューティックス、リミテッド	新規化合物
EP2114941B1 (en) *	2006-12-22	2015-03-25	Astex Therapeutics Limited	Bicyclic heterocyclic compounds as fgfr inhibitors
FR2925900B1 (fr) *	2008-01-02	2011-03-04	Sanofi Aventis	DERIVES DE N-PHENYL-IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2928922B1 (fr) *	2008-03-21	2010-04-23	Sanofi Aventis	Derives de 2-aryl-6-phenyl-imidazo°1,2-a!pyridines polysubstitues, leur preparation et leur application en therapeutique
FR2953520B1 (fr) *	2009-12-04	2011-11-25	Sanofi Aventis	Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique

2009
- 2009-09-18 FR FR0956444A patent/FR2950344B1/fr not_active Expired - Fee Related
2010
- 2010-09-16 JO JOP/2010/0315A patent/JO3017B1/ar active
- 2010-09-16 AR ARP100103375A patent/AR078180A1/es unknown
- 2010-09-17 PT PT107711590T patent/PT2477990E/pt unknown
- 2010-09-17 SI SI201030792T patent/SI2477990T1/sl unknown
- 2010-09-17 TW TW099131736A patent/TWI464169B/zh not_active IP Right Cessation
- 2010-09-17 PL PL10771159T patent/PL2477990T3/pl unknown
- 2010-09-17 WO PCT/FR2010/051932 patent/WO2011033230A1/fr not_active Ceased
- 2010-09-17 JP JP2012529329A patent/JP5616453B2/ja not_active Expired - Fee Related
- 2010-09-17 UY UY0001032894A patent/UY32894A/es not_active Application Discontinuation
- 2010-09-17 HR HRP20141119AT patent/HRP20141119T1/hr unknown
- 2010-09-17 ES ES10771159.0T patent/ES2523505T3/es active Active
- 2010-09-17 EP EP10771159.0A patent/EP2477990B1/fr not_active Not-in-force
- 2010-09-17 DK DK10771159.0T patent/DK2477990T3/en active
- 2010-09-17 US US13/496,118 patent/US8618301B2/en not_active Expired - Fee Related
2014
- 2014-11-20 CY CY20141100967T patent/CY1116581T1/el unknown

Also Published As

Publication number	Publication date
JP5616453B2 (ja)	2014-10-29
UY32894A (es)	2011-04-29
PT2477990E (pt)	2014-11-27
EP2477990A1 (fr)	2012-07-25
CY1116581T1 (el)	2018-03-07
JP2013505227A (ja)	2013-02-14
WO2011033230A1 (fr)	2011-03-24
DK2477990T3 (en)	2014-12-01
US20130023554A1 (en)	2013-01-24
AR078180A1 (es)	2011-10-19
FR2950344B1 (fr)	2011-11-25
JO3017B1 (ar)	2016-09-05
TWI464169B (zh)	2014-12-11
SI2477990T1 (sl)	2014-12-31
FR2950344A1 (fr)	2011-03-25
US8618301B2 (en)	2013-12-31
ES2523505T3 (es)	2014-11-26
EP2477990B1 (fr)	2014-08-20
HRP20141119T1 (hr)	2015-01-30
TW201118093A (en)	2011-06-01

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