PL2699581T3 - Pochodne 2-okso-1-imidazolidynyloimidazotiadiazolu - Google Patents

Pochodne 2-okso-1-imidazolidynyloimidazotiadiazolu

Info

Publication number
PL2699581T3
PL2699581T3 PL12714587T PL12714587T PL2699581T3 PL 2699581 T3 PL2699581 T3 PL 2699581T3 PL 12714587 T PL12714587 T PL 12714587T PL 12714587 T PL12714587 T PL 12714587T PL 2699581 T3 PL2699581 T3 PL 2699581T3
Authority
PL
Poland
Prior art keywords
oxo
imidazothiadiazole derivatives
imidazolidinyl
imidazolidinyl imidazothiadiazole
derivatives
Prior art date
Application number
PL12714587T
Other languages
English (en)
Inventor
Laurent Provins
Yannick Quesnel
Original Assignee
Ucb Biopharma Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Biopharma Sprl filed Critical Ucb Biopharma Sprl
Publication of PL2699581T3 publication Critical patent/PL2699581T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Lubricants (AREA)
PL12714587T 2011-04-18 2012-04-17 Pochodne 2-okso-1-imidazolidynyloimidazotiadiazolu PL2699581T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP11162853 2011-04-18
US201161480134P 2011-04-28 2011-04-28
PCT/EP2012/001658 WO2012143117A1 (en) 2011-04-18 2012-04-17 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives
EP12714587.8A EP2699581B1 (en) 2011-04-18 2012-04-17 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives

Publications (1)

Publication Number Publication Date
PL2699581T3 true PL2699581T3 (pl) 2016-05-31

Family

ID=44072751

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12714587T PL2699581T3 (pl) 2011-04-18 2012-04-17 Pochodne 2-okso-1-imidazolidynyloimidazotiadiazolu

Country Status (16)

Country Link
US (1) US8957218B2 (pl)
EP (1) EP2699581B1 (pl)
JP (1) JP5969003B2 (pl)
CA (1) CA2831830C (pl)
CY (1) CY1117210T1 (pl)
DK (1) DK2699581T3 (pl)
ES (1) ES2559288T3 (pl)
HR (1) HRP20151419T1 (pl)
HU (1) HUE026889T2 (pl)
ME (1) ME02351B (pl)
PL (1) PL2699581T3 (pl)
PT (1) PT2699581E (pl)
RS (1) RS54487B1 (pl)
SI (1) SI2699581T1 (pl)
SM (1) SMT201600024B (pl)
WO (1) WO2012143117A1 (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX386697B (es) 2014-01-21 2025-03-19 Janssen Pharmaceutica Nv Combinaciones que comprenden agonistas ortostericos o moduladores alostericos positivos del receptor glutamatergico metabotropico de subtipo 2 y su uso
ME03518B (me) 2014-01-21 2020-04-20 Janssen Pharmaceutica Nv Kombinacije koje obuhvataju pozitivne alosterične modulatore ili ortosterične agoniste metabotropnog glutamatergičnog receptora podtipa 2 i njihova primjena
CN110869375B (zh) * 2017-07-10 2022-08-30 Ucb生物制药有限责任公司 2-氧代-1-咪唑烷基咪唑并噻二唑衍生物
CN110869374B (zh) * 2017-07-10 2022-08-30 Ucb生物制药有限责任公司 2-氧代-1,3-噁唑烷基咪唑并噻二唑衍生物
EA202091403A1 (ru) 2017-12-12 2020-10-14 Юсб Байофарма Срл Производные 2-оксо-1-пирролидинилимидазотиадиазола
ES2947618T3 (es) * 2018-05-08 2023-08-14 UCB Biopharma SRL Derivados de 1-imidazotiadiazolo-2H-pirrol-5-ona
LV15614A (lv) * 2020-07-30 2022-02-20 Latvijas Organiskās Sintēzes Institūts 2-(2-okso-3-pirolin-1-il)acetamīdi kā pretkrampju līdzekļi

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1464259A (en) * 1975-10-03 1977-02-09 Pfizer Ltd Imidazo-thiazole and -thiadiazole sulphonamides and their use as therapeutic agents
GB8412357D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB8412358D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB0004297D0 (en) 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
EA010031B1 (ru) 2003-12-02 2008-06-30 Юсб, С.А. Производные имидазола, способы их получения и применения
US8178533B2 (en) * 2005-06-01 2012-05-15 Ucb Pharma, S.A. 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
US20100222326A1 (en) 2007-04-27 2010-09-02 Ucb Pharma, S.A. New Heterocyclic Derivatives Useful For The Treatment of CNS Disorders
HUE028668T2 (en) * 2009-10-23 2016-12-28 Ucb Biopharma Sprl 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives

Also Published As

Publication number Publication date
JP2014511883A (ja) 2014-05-19
HRP20151419T1 (hr) 2016-01-29
DK2699581T3 (en) 2016-01-11
HUE026889T2 (en) 2016-07-28
EP2699581A1 (en) 2014-02-26
JP5969003B2 (ja) 2016-08-10
EP2699581B1 (en) 2015-11-25
CA2831830A1 (en) 2012-10-26
ME02351B (me) 2016-06-20
RS54487B1 (sr) 2016-06-30
CA2831830C (en) 2017-12-12
CY1117210T1 (el) 2017-04-05
US20140148489A1 (en) 2014-05-29
US8957218B2 (en) 2015-02-17
WO2012143117A1 (en) 2012-10-26
ES2559288T3 (es) 2016-02-11
SMT201600024B (pl) 2016-02-25
AU2012244614A1 (en) 2013-10-31
SI2699581T1 (sl) 2016-02-29
PT2699581E (pt) 2016-03-22

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