PL3178817T3 - Postać amorficzna związku tetracyklicznego - Google Patents

Postać amorficzna związku tetracyklicznego

Info

Publication number
PL3178817T3
PL3178817T3 PL15830197T PL15830197T PL3178817T3 PL 3178817 T3 PL3178817 T3 PL 3178817T3 PL 15830197 T PL15830197 T PL 15830197T PL 15830197 T PL15830197 T PL 15830197T PL 3178817 T3 PL3178817 T3 PL 3178817T3
Authority
PL
Poland
Prior art keywords
amorphous form
tetracyclic compound
tetracyclic
compound
amorphous
Prior art date
Application number
PL15830197T
Other languages
English (en)
Inventor
Koji Shiraki
Tadanobu Nakayama
Tomoaki Ota
Original Assignee
Chugai Seiyaku Kabushiki Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55263964&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL3178817(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Chugai Seiyaku Kabushiki Kaisha filed Critical Chugai Seiyaku Kabushiki Kaisha
Publication of PL3178817T3 publication Critical patent/PL3178817T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL15830197T 2014-08-08 2015-08-07 Postać amorficzna związku tetracyklicznego PL3178817T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2014162899 2014-08-08
EP15830197.8A EP3178817B1 (en) 2014-08-08 2015-08-07 Amorphous form of tetracyclic compound
PCT/JP2015/072450 WO2016021707A1 (ja) 2014-08-08 2015-08-07 ４環性化合物の非晶質体

Publications (1)

Publication Number Publication Date
PL3178817T3 true PL3178817T3 (pl) 2020-11-16

Family

ID=55263964

Family Applications (1)

Application Number Title Priority Date Filing Date
PL15830197T PL3178817T3 (pl) 2014-08-08 2015-08-07 Postać amorficzna związku tetracyklicznego

Country Status (8)

Country Link
US (5) US10344014B2 (pl)
EP (2) EP3178817B1 (pl)
JP (3) JP6906308B2 (pl)
DK (1) DK3178817T3 (pl)
ES (1) ES2803577T3 (pl)
PL (1) PL3178817T3 (pl)
TW (4) TWI831347B (pl)
WO (1) WO2016021707A1 (pl)

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ES3019912T3 (en) 2014-12-05 2025-05-21 Aragon Pharmaceuticals Inc Anticancer compositions
CA2973857C (en) 2015-01-16 2023-11-07 Chugai Seiyaku Kabushiki Kaisha Combination drug
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CN110494422A (zh) 2017-03-15 2019-11-22 太阳制药先进研究有限公司 4-甲基-3-喹啉-3-基乙炔基-苯甲酸n’-(2-氯-6-甲基-苯甲酰基)酰肼的新型无定形分散体
RU2768887C2 (ru) * 2017-03-15 2022-03-25 Сан Фарма Эдвансд Рисёч Компани Лимитед Новая аморфная дисперсия (5-{ 5-[n'-(2-хлор-6-метилбензоил)гидразинокарбонил]-2-метил-фенилэтинил} -пиридин-2-ил)амида циклопропанкарбоновой кислоты
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WO2022176017A1 (ja) * 2021-02-16 2022-08-25 大塚製薬株式会社 非晶質体及び当該非晶質体を含む組成物
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WO2015163447A1 (ja) 2014-04-25 2015-10-29 中外製薬株式会社 ４環性化合物の新規結晶
EP3157569B1 (en) 2014-06-18 2019-07-24 F.Hoffmann-La Roche Ag New pharmaceutical composition comprising non-ionic surfactants
TWI831347B (zh) 2014-08-08 2024-02-01 日商中外製藥股份有限公司 包含４環性化合物的非晶質體之固體分散體及製劑

Also Published As

Publication number Publication date
TWI718102B (zh) 2021-02-11
TWI803187B (zh) 2023-05-21
TW202115047A (zh) 2021-04-16
US20170217927A1 (en) 2017-08-03
JP7483804B2 (ja) 2024-05-15
JP2022153575A (ja) 2022-10-12
US20230339885A1 (en) 2023-10-26
JP6906308B2 (ja) 2021-07-21
US20210238160A1 (en) 2021-08-05
EP3178817B1 (en) 2020-06-10
DK3178817T3 (da) 2020-07-13
JP7116825B2 (ja) 2022-08-10
TW202222796A (zh) 2022-06-16
WO2016021707A1 (ja) 2016-02-11
EP3178817A4 (en) 2018-01-03
EP3178817A1 (en) 2017-06-14
US20190284163A1 (en) 2019-09-19
TW201613906A (en) 2016-04-16
JP2021119194A (ja) 2021-08-12
EP3660009A1 (en) 2020-06-03
US10774067B2 (en) 2020-09-15
JPWO2016021707A1 (ja) 2017-05-25
ES2803577T3 (es) 2021-01-28
TW202322823A (zh) 2023-06-16
TWI765410B (zh) 2022-05-21
TWI831347B (zh) 2024-02-01
US20250243179A1 (en) 2025-07-31
US10344014B2 (en) 2019-07-09

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