PL3209661T3 - Sposób wytwarzania polimorfu rywaroksabanu - Google Patents
Sposób wytwarzania polimorfu rywaroksabanuInfo
- Publication number
- PL3209661T3 PL3209661T3 PL15784372T PL15784372T PL3209661T3 PL 3209661 T3 PL3209661 T3 PL 3209661T3 PL 15784372 T PL15784372 T PL 15784372T PL 15784372 T PL15784372 T PL 15784372T PL 3209661 T3 PL3209661 T3 PL 3209661T3
- Authority
- PL
- Poland
- Prior art keywords
- rivaroxaban
- polymorph
- preparing
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- KGFYHTZWPPHNLQ-AWEZNQCLSA-N rivaroxaban Chemical compound S1C(Cl)=CC=C1C(=O)NC[C@@H]1OC(=O)N(C=2C=CC(=CC=2)N2C(COCC2)=O)C1 KGFYHTZWPPHNLQ-AWEZNQCLSA-N 0.000 title 1
- 229960001148 rivaroxaban Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
- C07D265/32—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14460075 | 2014-10-22 | ||
| EP15784372.3A EP3209661B1 (en) | 2014-10-22 | 2015-10-22 | Process for preparing a polymorph of rivaroxaban |
| PCT/EP2015/074538 WO2016062828A1 (en) | 2014-10-22 | 2015-10-22 | Process for preparing a polymorph of rivaroxaban |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL3209661T3 true PL3209661T3 (pl) | 2021-08-16 |
Family
ID=51904938
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL15784372T PL3209661T3 (pl) | 2014-10-22 | 2015-10-22 | Sposób wytwarzania polimorfu rywaroksabanu |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US10040786B2 (pl) |
| EP (1) | EP3209661B1 (pl) |
| EA (1) | EA034656B1 (pl) |
| PL (1) | PL3209661T3 (pl) |
| WO (1) | WO2016062828A1 (pl) |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1413218A (zh) | 1999-12-28 | 2003-04-23 | 味之素株式会社 | 天冬甜素衍生物的结晶 |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| DE102004002044A1 (de) | 2004-01-15 | 2005-08-04 | Bayer Healthcare Ag | Herstellverfahren |
| CA2823159C (en) | 2005-10-04 | 2014-10-21 | Bayer Intellectual Property Gmbh | Polymorphic form of 5-chloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophenecarboxamide |
| EA031064B2 (ru) | 2009-07-31 | 2020-07-01 | КРКА, д.д., НОВО МЕСТО | Способы кристаллизации ривароксабана |
| EP3309158B1 (en) * | 2012-12-21 | 2022-03-16 | Krka, tovarna zdravil, d.d. | Crystalline form k of rivaroxaban and process for its preparation |
| IN2014CH00290A (pl) * | 2014-01-23 | 2015-08-14 | Symed Labs Ltd |
-
2015
- 2015-10-22 EA EA201790891A patent/EA034656B1/ru not_active IP Right Cessation
- 2015-10-22 WO PCT/EP2015/074538 patent/WO2016062828A1/en not_active Ceased
- 2015-10-22 EP EP15784372.3A patent/EP3209661B1/en not_active Not-in-force
- 2015-10-22 PL PL15784372T patent/PL3209661T3/pl unknown
- 2015-10-22 US US15/520,499 patent/US10040786B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP3209661A1 (en) | 2017-08-30 |
| EP3209661B1 (en) | 2021-02-17 |
| EA034656B1 (ru) | 2020-03-03 |
| EA201790891A1 (ru) | 2017-08-31 |
| WO2016062828A1 (en) | 2016-04-28 |
| US10040786B2 (en) | 2018-08-07 |
| US20170313689A1 (en) | 2017-11-02 |
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