PL340456A1 - Novel oral dosage form of carvedilol - Google Patents

Novel oral dosage form of carvedilol

Info

Publication number: PL340456A1
Authority: PL; Poland
Prior art keywords: carvedilol; dosage form; oral dosage; novel oral; novel
Prior art date: 1997-11-12

Application number

PL98340456A

Inventor

Choon K Oh

Original Assignee

Boehringer Mannheim Pharm Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-11-12

Filing date

1998-11-12

Publication date

2001-02-12

1998-11-12 Application filed by Boehringer Mannheim Pharm Corp filed Critical Boehringer Mannheim Pharm Corp

2001-02-12 Publication of PL340456A1 publication Critical patent/PL340456A1/en

Links

NPAKNKYSJIDKMW-UHFFFAOYSA-N carvedilol Chemical compound COC1=CC=CC=C1OCCNCC(O)COC1=CC=CC2=NC3=CC=C[CH]C3=C12 NPAKNKYSJIDKMW-UHFFFAOYSA-N 0.000 title 1
229960004195 carvedilol Drugs 0.000 title 1
239000006186 oral dosage form Substances 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Heart & Thoracic Surgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Cardiology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Dispersion Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Indole Compounds (AREA)

PL98340456A 1997-11-12 1998-11-12 Novel oral dosage form of carvedilol PL340456A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US6545697P	1997-11-12	1997-11-12
PCT/US1998/024102 WO1999024017A1 (en)	1997-11-12	1998-11-12	Novel oral dosage form for carvedilol

Publications (1)

Publication Number	Publication Date
PL340456A1 true PL340456A1 (en)	2001-02-12

Family

ID=22062830

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL98340456A PL340456A1 (en)	1997-11-12	1998-11-12	Novel oral dosage form of carvedilol

Country Status (14)

Country	Link
EP (1)	EP1030651A4 (en)
JP (1)	JP2001522794A (en)
KR (1)	KR20010031952A (en)
CN (1)	CN1285738A (en)
AU (1)	AU751117B2 (en)
BR (1)	BR9814127A (en)
CA (1)	CA2309542A1 (en)
HU (1)	HUP0004345A3 (en)
IL (1)	IL136028A0 (en)
NO (1)	NO20002439L (en)
NZ (1)	NZ504418A (en)
PL (1)	PL340456A1 (en)
TR (1)	TR200001362T2 (en)
WO (1)	WO1999024017A1 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2003275953A1 (en)	2002-11-08	2004-06-07	Egalet A/S	Controlled release carvedilol compositions
WO2004056336A2 (en) *	2002-12-20	2004-07-08	Ranbaxy Laboratories Limited	Controlled release, multiple unit drug delivery systems
WO2005051322A2 (en) *	2003-11-25	2005-06-09	Sb Pharmco Puerto Rico Inc.	Controlled release pharmaceutical formulations comprising carvedilol, free based and its salts
US20050169994A1 (en) *	2003-11-25	2005-08-04	Burke Matthew D.	Carvedilol free base, salts, anhydrous forms or solvates thereof, corresponding pharmaceutical compositions, controlled release formulations, and treatment or delivery methods
EP2010162A4 (en) *	2006-04-03	2013-01-09	Isa Odidi	Drug delivery composition
TWI415604B (en) *	2009-09-29	2013-11-21	Tsh Biopharm Corp Ltd	Regulated release of caffetilol dosage form
TW201132646A (en) *	2010-02-22	2011-10-01	Daiichi Sankyo Co Ltd	Oral solid extended release dosage form
ES2706880T3 (en)	2010-02-22	2019-04-01	Daiichi Sankyo Co Ltd	Sustained-release solid preparation for oral use
TW201200165A (en) *	2010-02-22	2012-01-01	Daiichi Sankyo Co Ltd	Oral solid extended release dosage form
RU2665372C2 (en)	2012-09-03	2018-08-29	Дайити Санкио Компани, Лимитед	Hydromorphone hydrochloride-containing oral sustained-release pharmaceutical composition
KR102158339B1 (en) *	2016-02-05	2020-09-21	삼진제약주식회사	Carvedilol immediate release formulation having improved madescent
KR102492147B1 (en)	2020-12-30	2023-01-26	단국대학교 천안캠퍼스 산학협력단	Carvedilol loaded solid oral compositions using self-nanoemulsifying drug delivery system and methods for their preparation
KR102525298B1 (en)	2020-12-30	2023-04-25	단국대학교 천안캠퍼스 산학협력단	Carvedilol loaded solid dispersion with increased oral bioavailability and methods for their preparation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2815926A1 (en) *	1978-04-13	1979-10-18	Boehringer Mannheim Gmbh	NEW CARBAZOLYL- (4) -OXY-PROPANOLAMINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
JPS5598120A (en) *	1979-01-16	1980-07-25	Shin Etsu Chem Co Ltd	Preparation of drug having enteric coating
CA1146866A (en) *	1979-07-05	1983-05-24	Yamanouchi Pharmaceutical Co. Ltd.	Process for the production of sustained release pharmaceutical composition of solid medical material
US4680323A (en) *	1983-12-01	1987-07-14	Hans Lowey	Method and composition for the preparation of controlled long-acting pharmaceuticals for oral administration
EP0554306B1 (en) *	1990-10-23	1996-02-21	Davband Pty. Limited	Back support for a chair or seat
US5760069A (en) *	1995-02-08	1998-06-02	Boehringer Mannheim Pharmaceuticals Corporation-Smithkline Beecham Corporation Limited Partnership #1	Method of treatment for decreasing mortality resulting from congestive heart failure
DE19637082A1 (en) *	1996-09-12	1998-03-19	Boehringer Mannheim Gmbh	Rapidly disintegrating pellets

1998
- 1998-11-12 CN CN98813082A patent/CN1285738A/en active Pending
- 1998-11-12 BR BR9814127-9A patent/BR9814127A/en not_active IP Right Cessation
- 1998-11-12 EP EP98958546A patent/EP1030651A4/en not_active Withdrawn
- 1998-11-12 AU AU14569/99A patent/AU751117B2/en not_active Ceased
- 1998-11-12 JP JP2000520110A patent/JP2001522794A/en active Pending
- 1998-11-12 NZ NZ504418A patent/NZ504418A/en unknown
- 1998-11-12 KR KR1020007005059A patent/KR20010031952A/en not_active Ceased
- 1998-11-12 IL IL13602898A patent/IL136028A0/en not_active IP Right Cessation
- 1998-11-12 PL PL98340456A patent/PL340456A1/en unknown
- 1998-11-12 HU HU0004345A patent/HUP0004345A3/en unknown
- 1998-11-12 TR TR2000/01362T patent/TR200001362T2/en unknown
- 1998-11-12 CA CA002309542A patent/CA2309542A1/en not_active Abandoned
- 1998-11-12 WO PCT/US1998/024102 patent/WO1999024017A1/en not_active Ceased
2000
- 2000-05-11 NO NO20002439A patent/NO20002439L/en unknown

Also Published As

Publication number	Publication date
AU751117B2 (en)	2002-08-08
HUP0004345A3 (en)	2001-10-29
TR200001362T2 (en)	2000-09-21
AU1456999A (en)	1999-05-31
IL136028A0 (en)	2001-05-20
NO20002439D0 (en)	2000-05-11
EP1030651A4 (en)	2006-05-31
CA2309542A1 (en)	1999-05-20
JP2001522794A (en)	2001-11-20
NZ504418A (en)	2003-02-28
HUP0004345A2 (en)	2001-06-28
KR20010031952A (en)	2001-04-16
NO20002439L (en)	2000-05-11
BR9814127A (en)	2000-10-03
EP1030651A1 (en)	2000-08-30
WO1999024017A1 (en)	1999-05-20
CN1285738A (en)	2001-02-28

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