PL356465A1 - Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu - Google Patents

Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu

Info

Publication number: PL356465A1
Authority: PL; Poland
Prior art keywords: 7alpha; 17alpha; 17beta; pregn; yne
Prior art date: 2002-10-04

Application number

PL02356465A

Other languages

English (en)

Inventor

Jacek Martynow

Andrzej Kutner

Wiesław Szelejewski

Wanda Wojciechowska

Hanna Fitak

Original Assignee

ANPHARM Przedsiębiorstwo Farmaceutyczne S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-10-04

Filing date

2002-10-04

Publication date

2004-04-05

2002-10-04 Application filed by ANPHARM Przedsiębiorstwo Farmaceutyczne S.A. filed Critical ANPHARM Przedsiębiorstwo Farmaceutyczne S.A.

2002-10-04 Priority to PL02356465A priority Critical patent/PL356465A1/pl

2003-10-01 Priority to AU2003278652A priority patent/AU2003278652A1/en

2003-10-01 Priority to EP03770184A priority patent/EP1556407A2/en

2003-10-01 Priority to US10/530,139 priority patent/US20060111332A1/en

2003-10-01 Priority to PCT/PL2003/000099 priority patent/WO2004031204A2/en

2004-04-05 Publication of PL356465A1 publication Critical patent/PL356465A1/pl

Links

238000004519 manufacturing process Methods 0.000 title 1
238000000034 method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J21/005—Ketals
- C07J21/006—Ketals at position 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)

PL02356465A 2002-10-04 2002-10-04 Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu PL356465A1 (pl)

Priority Applications (5)

Application Number	Priority Date	Filing Date	Title
PL02356465A PL356465A1 (pl)	2002-10-04	2002-10-04	Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu
AU2003278652A AU2003278652A1 (en)	2002-10-04	2003-10-01	Process and intermediates to prepare 17.beta.-hydroxy-7.alfa.-methyl-19-nor-17.alfa.-pregn-5(10)-en-20-yn-3-one
EP03770184A EP1556407A2 (en)	2002-10-04	2003-10-01	Process and intermediates to prepare 17.beta.-hydroxy-7.alfa.-methyl-19-nor-17.alfa.-pregn-5(10)-en-20-yn-3-one
US10/530,139 US20060111332A1 (en)	2002-10-04	2003-10-01	Process and intermediates to prepare17beta-hydroxy-7alpha-methyl-19-nor-17alpha-pregn -5(10)-en-20-yn-3-one
PCT/PL2003/000099 WO2004031204A2 (en)	2002-10-04	2003-10-01	Process and intermediates to prepare 17.beta.-hydroxy-7.alfa.-methyl-19-nor-17.alfa.-pregn-5(10)-en-20-yn-3-one

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PL02356465A PL356465A1 (pl)	2002-10-04	2002-10-04	Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu

Publications (1)

Publication Number	Publication Date
PL356465A1 true PL356465A1 (pl)	2004-04-05

Family

ID=32065086

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL02356465A PL356465A1 (pl)	2002-10-04	2002-10-04	Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu

Country Status (5)

Country	Link
US (1)	US20060111332A1 (pl)
EP (1)	EP1556407A2 (pl)
AU (1)	AU2003278652A1 (pl)
PL (1)	PL356465A1 (pl)
WO (1)	WO2004031204A2 (pl)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1861373A2 (en)	2005-03-10	2007-12-05	Mallinckrodt, Inc.	Processes for preparing morphinans and intermediates thereof
CN110981930B (zh) *	2019-12-31	2021-04-20	浙江仙居君业药业有限公司	一种替勃龙的合成方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2806030A (en) *	1954-03-20	1957-09-10	Syntex Sa	Cyclopentanophenanthrene derivatives and process for the preparation thereof
NL125069C (pl) *	1963-12-24
NL128815C (pl) *	1965-03-16
NL146838B (nl) *	1966-06-24	1975-08-15	Organon Nv	Werkwijze voor het bereiden van (delta)5(10)-3- keto-19-norsteroiden.
US3558776A (en) *	1968-06-14	1971-01-26	Upjohn Co	Pharmaceutical composition comprising 17alpha - ethynyl -17beta - hydroxy - 7alpha - methyl -5(10)-estrene-3-one
US3904611A (en) *	1972-10-16	1975-09-09	Syntex Corp	Preparation of 17' -propadienyl steroids
US4035376A (en) *	1972-10-24	1977-07-12	Janssen Pharmaceutica N.V.	Aroyl-substituted phenylacetic acid derivatives
US3928398A (en) *	1973-11-01	1975-12-23	Richardson Merrell Inc	Derivatives of 7{60 -methylestr-4-en-3{60 ,17{62 -diol
US4308265A (en) *	1979-10-05	1981-12-29	United States Of America	7α-Methylnorethindrone enanthate and its use in long term suppression of fertility in female mammals
US4252800A (en) *	1979-10-05	1981-02-24	United States Of America	7α-methylnorethindrone enanthate and its use in long term suppression of fertility in female mammals
DE3337179A1 (de) *	1983-10-10	1985-05-23	Schering AG, 1000 Berlin und 4709 Bergkamen	Estran- und androstan-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende praeparate
FR2610933B1 (fr) *	1987-02-18	1989-06-09	Roussel Uclaf	Nouveaux 19-nor steroides substitues en position 7, leur preparation, leur application comme medicaments, les compositions pharmaceutiques les renfermant
ATE239032T1 (de) *	1998-10-16	2003-05-15	Akzo Nobel Nv	(7alpha,17alpha)-17-hydroxy-7-methyl-19-nor-17- pregn-5-(10)-en-20-yn-3-on als reine verbindung

2002
- 2002-10-04 PL PL02356465A patent/PL356465A1/pl unknown
2003
- 2003-10-01 US US10/530,139 patent/US20060111332A1/en not_active Abandoned
- 2003-10-01 WO PCT/PL2003/000099 patent/WO2004031204A2/en not_active Ceased
- 2003-10-01 AU AU2003278652A patent/AU2003278652A1/en not_active Abandoned
- 2003-10-01 EP EP03770184A patent/EP1556407A2/en not_active Withdrawn

Also Published As

Publication number	Publication date
US20060111332A1 (en)	2006-05-25
AU2003278652A1 (en)	2004-04-23
WO2004031204A3 (en)	2004-07-01
AU2003278652A8 (en)	2004-04-23
WO2004031204A2 (en)	2004-04-15
EP1556407A2 (en)	2005-07-27

Legal Events

Date	Code	Title	Description
2009-10-30	DISC	Decisions on discontinuance of the proceedings (taken after the publication of the particulars of the applications)

Publication	Publication Date	Title
AU2003236991A8 (en)	2003-12-19	Representations of processes
EP1577280A4 (en)	2006-08-23	DEUTERATION PROCESS
PL355161A1 (en)	2003-01-13	Method of manufacture
GB2385602B (en)	2004-04-21	Method of photoelectrolysis
EP1488046A4 (en)	2005-11-23	CONSTRUCTION METHODS
GB0123120D0 (en)	2001-11-14	Method of attachment
IL162770A0 (en)	2005-11-20	Process for the preparation methylsteroids of 7
PL356465A1 (pl)	2004-04-05	Sposób wytwarzania 17beta-hydroksy-7alfa-metylo-19-nor-17alfa-pregn-5(10)-en-20-yn-3-onu
IL158119A0 (en)	2004-03-28	Method for the production of delta1-pyrrolines
GB0215867D0 (en)	2002-08-14	Novel method and compounds
AU2003267944A8 (en)	2003-12-22	Novel trifluoromethylepinephrine compounds and methods of making and using thereof
GB0200049D0 (en)	2002-02-20	Method of manufacture
GB0219671D0 (en)	2002-10-02	Method of manufacture
PL357986A1 (pl)	2004-06-28	Sposób wytwarzania węglikostali
GB0222015D0 (en)	2002-10-30	Means of assembly-bozz 2
PL347523A1 (en)	2001-11-05	Method of obtaining 11alpha-hydroxy-1-dehydrotestosterone
PL356317A1 (en)	2003-04-07	Method of obtaining alkanosulphonylpyridines
PL354552A1 (pl)	2003-12-29	Sposób wytwarzania 2,4-dichlorofenoluSposób wytwarzania 2,4-dichlorofenolu
GB0104109D0 (en)	2001-04-04	Method of manufacture
PL357664A1 (pl)	2004-06-14	Sposób modyfikacji cząsteczki chemicznej
PL355859A1 (pl)	2003-09-22	Sposób wykonywania ozdób
PL355451A1 (pl)	2004-02-23	Sposób wykonywania słupo-pala
PL351938A1 (en)	2003-08-11	Method of obtaining fructisiltransferase
PL355043A1 (pl)	2004-01-26	Sposób wytwarzania p-oktylofenolu
HUP0302540A3 (en)	2005-11-28	Method of producing 1-alkyl-3-aryl-5-difluoromethoxy-1h-pyrazoles