PL358886A1 - Związki do leczenia upośledzonego wiotczenia dna żołądka - Google Patents

Związki do leczenia upośledzonego wiotczenia dna żołądka

Info

Publication number
PL358886A1
PL358886A1 PL01358886A PL35888601A PL358886A1 PL 358886 A1 PL358886 A1 PL 358886A1 PL 01358886 A PL01358886 A PL 01358886A PL 35888601 A PL35888601 A PL 35888601A PL 358886 A1 PL358886 A1 PL 358886A1
Authority
PL
Poland
Prior art keywords
sup
sub
alkyl
bivalent radical
alk
Prior art date
Application number
PL01358886A
Other languages
English (en)
Other versions
PL201656B1 (pl
Inventor
Emelen Kristof Van
Bruyn Marcel Frans Leopold De
Manuel Jesus Alcazar-Vaca
Jose Ignacio Andres-Gil
Francisco Javier Fernandez-Gadea
Maria Encarnacion Matesanz-Ballesteros
Jose Manuel Bartolome-Nebreda
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of PL358886A1 publication Critical patent/PL358886A1/pl
Publication of PL201656B1 publication Critical patent/PL201656B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL358886A 2000-06-22 2001-06-13 Pochodna imidazolidyny lub pirymidyny i sposób jej otrzymywania oraz kompozycja farmaceutyczna PL201656B1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00202180 2000-06-22
PCT/EP2001/006749 WO2001098306A1 (en) 2000-06-22 2001-06-13 Compounds for treating impaired fundic relaxation

Publications (2)

Publication Number Publication Date
PL358886A1 true PL358886A1 (pl) 2004-08-23
PL201656B1 PL201656B1 (pl) 2009-04-30

Family

ID=8171674

Family Applications (1)

Application Number Title Priority Date Filing Date
PL358886A PL201656B1 (pl) 2000-06-22 2001-06-13 Pochodna imidazolidyny lub pirymidyny i sposób jej otrzymywania oraz kompozycja farmaceutyczna

Country Status (33)

Country Link
US (2) US7081453B2 (pl)
EP (1) EP1296987B1 (pl)
JP (1) JP4911860B2 (pl)
KR (1) KR100821107B1 (pl)
CN (2) CN100516066C (pl)
AR (1) AR032158A1 (pl)
AT (1) ATE312104T1 (pl)
AU (1) AU783292B2 (pl)
BG (1) BG65895B1 (pl)
BR (1) BR0111859B1 (pl)
CA (1) CA2410233C (pl)
CZ (1) CZ305005B6 (pl)
DE (1) DE60115647T2 (pl)
EA (1) EA005760B1 (pl)
EE (1) EE04878B1 (pl)
EG (1) EG24462A (pl)
ES (1) ES2254467T3 (pl)
HR (1) HRP20020988B1 (pl)
HU (1) HU227398B1 (pl)
IL (2) IL153559A0 (pl)
IS (1) IS2618B (pl)
JO (1) JO2352B1 (pl)
MX (1) MXPA02012844A (pl)
MY (1) MY155267A (pl)
NO (1) NO328547B1 (pl)
NZ (1) NZ522519A (pl)
PA (1) PA8519601A1 (pl)
PL (1) PL201656B1 (pl)
SA (1) SA01220442B1 (pl)
SK (1) SK287730B6 (pl)
UA (1) UA74576C2 (pl)
WO (1) WO2001098306A1 (pl)
ZA (1) ZA200210303B (pl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2231189T3 (es) 1999-06-02 2005-05-16 Janssen Pharmaceutica N.V. Derivados de benzodioxano o benzopirano sustituidos con pirrolidinilo, piperidinilo u homopiperidinilo.
EA004645B1 (ru) 1999-06-02 2004-06-24 Янссен Фармацевтика Н.В. Аминоалкилзамещенные производные бензопирана
JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en) 2000-09-04 2012-06-17 شركة جانسين فارماسوتيكا ان. في Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en) 2000-11-21 2007-06-17 شركة جانسين فارماسوتيكا ان. في Second-phenyl carboxy amides are useful as lipid-lowering agents
NZ543102A (en) 2003-04-24 2008-12-24 Incyte Corp Aza spiro alkane derivatives as inhibitors of metalloproteases
JP4896476B2 (ja) * 2005-09-16 2012-03-14 広栄化学工業株式会社 メチルオキシメチルアミノピリジン誘導体及びその製造方法
US7999107B2 (en) 2007-01-31 2011-08-16 Merck Sharp & Dohme Corp. Substituted pyrano[2,3-B]pyridine derivatives as cannabinoid-1 receptor modulators
US9096546B2 (en) * 2007-05-10 2015-08-04 Albany Molecular Research, Inc. Aryl- and heteroaryl-substituted tetrahydrobenzo-1,4-diazepines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
MD20140044A2 (ro) 2011-11-11 2014-08-31 Pfizer Inc. 2-Tiopirimidinone şi utilizarea lor pentru tratamentul afecţiunilor cardiovasculare
AU2016257179A1 (en) 2015-05-05 2017-11-02 Pfizer Inc. 2-thiopyrimidinones
CN105481839B (zh) * 2015-11-23 2018-05-11 安徽千和新材料科技发展有限公司 一种光活性环氧啉对映体的制备方法
EP3229193A1 (en) 2016-04-07 2017-10-11 The Boeing Company A computer-implemented method and system for sharing information between passengers and air traffic management stakeholders

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910930A (en) 1973-01-04 1975-10-07 Janssen Pharmaceutica Nv 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones
DE2400049A1 (de) * 1974-01-02 1975-07-10 Spumalit Anstalt Transportkasten aus kunststoff, insbesondere fuer flaschen
GR71865B (pl) * 1978-03-20 1983-07-07 Ciba Geigy
US4329348A (en) * 1979-02-26 1982-05-11 Ciba-Geigy Corporation N-Oxacyclic-alkylpiperidines as psychostimulants
EP0144101B1 (en) * 1983-11-30 1991-02-06 Janssen Pharmaceutica N.V. Bicyclic heterocyclyl containing n-(bicyclic heterocyclyl)-4-piperidinamines
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
ZA931343B (en) 1992-03-06 1993-09-24 Akzo Nv 1,4-dioxino(2,3-b)pyridine derivatives.
US6403103B1 (en) * 1994-08-12 2002-06-11 Bio Merieux Trypanosoma cruzi antigen, gene encoding therefore, and methods of detecting and treating chagas disease
FR2744451B1 (fr) * 1996-02-01 1998-04-24 Pf Medicament Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique
US6133277A (en) * 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
ES2231189T3 (es) * 1999-06-02 2005-05-16 Janssen Pharmaceutica N.V. Derivados de benzodioxano o benzopirano sustituidos con pirrolidinilo, piperidinilo u homopiperidinilo.
EA004645B1 (ru) * 1999-06-02 2004-06-24 Янссен Фармацевтика Н.В. Аминоалкилзамещенные производные бензопирана
TWI225488B (en) * 1999-12-21 2004-12-21 Janssen Pharmaceutica Nv Derivatives of homopiperidinyl substituted benzimidazole analogues
JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus

Also Published As

Publication number Publication date
CZ2003115A3 (cs) 2003-06-18
UA74576C2 (en) 2006-01-16
CZ305005B6 (cs) 2015-03-25
HUP0301185A3 (en) 2009-03-30
JP2004501157A (ja) 2004-01-15
ZA200210303B (en) 2004-03-19
SK492003A3 (en) 2003-07-01
BG65895B1 (bg) 2010-04-30
BR0111859A (pt) 2003-05-13
MXPA02012844A (es) 2003-05-15
IS6591A (is) 2002-10-25
EE04878B1 (et) 2007-08-15
CA2410233A1 (en) 2001-12-27
AR032158A1 (es) 2003-10-29
KR20030007566A (ko) 2003-01-23
MY155267A (en) 2015-09-30
SK287730B6 (en) 2011-07-06
IL153559A (en) 2008-03-20
DE60115647T2 (de) 2006-08-24
NO20026219D0 (no) 2002-12-23
AU783292B2 (en) 2005-10-13
WO2001098306A1 (en) 2001-12-27
NO20026219L (no) 2003-02-17
HU227398B1 (hu) 2011-05-30
EP1296987A1 (en) 2003-04-02
PA8519601A1 (es) 2002-08-26
CN100516066C (zh) 2009-07-22
US20060142318A1 (en) 2006-06-29
BG107313A (bg) 2003-06-30
CN1781921A (zh) 2006-06-07
HRP20020988B1 (en) 2011-06-30
EA200300049A1 (ru) 2003-04-24
PL201656B1 (pl) 2009-04-30
JO2352B1 (en) 2006-12-12
CN1437602A (zh) 2003-08-20
US7423048B2 (en) 2008-09-09
IS2618B (is) 2010-04-15
EG24462A (en) 2009-07-16
DE60115647D1 (de) 2006-01-12
BR0111859B1 (pt) 2015-01-06
US20040019051A1 (en) 2004-01-29
NO328547B1 (no) 2010-03-15
EP1296987B1 (en) 2005-12-07
AU8386401A (en) 2002-01-02
JP4911860B2 (ja) 2012-04-04
CN1288157C (zh) 2006-12-06
HK1057896A1 (en) 2004-04-23
EE200200694A (et) 2004-06-15
ATE312104T1 (de) 2005-12-15
NZ522519A (en) 2003-09-26
HRP20020988A2 (en) 2005-02-28
KR100821107B1 (ko) 2008-04-14
SA01220442B1 (ar) 2008-05-21
US7081453B2 (en) 2006-07-25
EA005760B1 (ru) 2005-06-30
ES2254467T3 (es) 2006-06-16
CA2410233C (en) 2011-01-25
IL153559A0 (en) 2003-07-06
HUP0301185A2 (hu) 2003-08-28

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