PL3645539T3 - Pochodne pirydoimidazoryfamycyny jako środek przeciwbakteryjny - Google Patents

Pochodne pirydoimidazoryfamycyny jako środek przeciwbakteryjny

Info

Publication number
PL3645539T3
PL3645539T3 PL18755539T PL18755539T PL3645539T3 PL 3645539 T3 PL3645539 T3 PL 3645539T3 PL 18755539 T PL18755539 T PL 18755539T PL 18755539 T PL18755539 T PL 18755539T PL 3645539 T3 PL3645539 T3 PL 3645539T3
Authority
PL
Poland
Prior art keywords
pyridimidazorifamycin
derivatives
antibacterial agent
antibacterial
agent
Prior art date
Application number
PL18755539T
Other languages
English (en)
Inventor
Egidio Marchi
Alessandro Lapini Sacchetti
Claudia ORI
Lisa PRETI
Original Assignee
Biofer S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IT102017000091912A external-priority patent/IT201700091912A1/it
Application filed by Biofer S.P.A. filed Critical Biofer S.P.A.
Publication of PL3645539T3 publication Critical patent/PL3645539T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL18755539T 2017-06-26 2018-06-25 Pochodne pirydoimidazoryfamycyny jako środek przeciwbakteryjny PL3645539T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP17177894 2017-06-26
IT102017000091912A IT201700091912A1 (it) 2017-08-08 2017-08-08 Nuove pirido-imidazo rifamicine
PCT/IB2018/054645 WO2019003076A1 (en) 2017-06-26 2018-06-25 PYRIDO-IMIDAZO-RIFAMYCIN DERIVATIVES AS ANTIBACTERIAL AGENT
EP18755539.6A EP3645539B1 (en) 2017-06-26 2018-06-25 Pyrido-imidazo rifamycin derivatives as antibacterial agent

Publications (1)

Publication Number Publication Date
PL3645539T3 true PL3645539T3 (pl) 2021-10-25

Family

ID=64742822

Family Applications (1)

Application Number Title Priority Date Filing Date
PL18755539T PL3645539T3 (pl) 2017-06-26 2018-06-25 Pochodne pirydoimidazoryfamycyny jako środek przeciwbakteryjny

Country Status (10)

Country Link
US (2) US11028086B2 (pl)
EP (1) EP3645539B1 (pl)
CN (1) CN110770244A (pl)
DK (1) DK3645539T3 (pl)
ES (1) ES2868180T3 (pl)
HU (1) HUE054832T2 (pl)
MX (1) MX386622B (pl)
PL (1) PL3645539T3 (pl)
RU (1) RU2020102511A (pl)
WO (1) WO2019003076A1 (pl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1698630E (pt) 2005-03-03 2014-09-15 Alfa Wassermann Spa Novas formas polimorfas de rifaximina, processos para a sua produção e a sua utilização nas preparações medicinais
CN110770244A (zh) 2017-06-26 2020-02-07 倍尔福股份公司 吡啶并咪唑利福霉素衍生物的抗菌剂
JP2025536245A (ja) * 2022-10-05 2025-11-05 リージェンツ オブ ザ ユニバーシティ オブ ミネソタ 非結核性マイコバクテリアに対するリファマイシン

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1090759B (it) 1977-11-29 1985-06-26 Alfa Farmaceutici Spa Procedimento per la preparazione di 3 iodio e 3 bromo rifamicina s
IT1154655B (it) * 1980-05-22 1987-01-21 Alfa Farmaceutici Spa Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica
IT1199374B (it) * 1984-05-15 1988-12-30 Alfa Farmaceutici Spa Processo per la preparazione di pirido-imidazo-rifamicine
ITMI20032144A1 (it) 2003-11-07 2005-05-08 Alfa Wassermann Spa Forme polimorfe di rifaximina, processi per ottenerle e
US7250413B2 (en) * 2004-04-26 2007-07-31 Cumbre Pharmaceuticals Inc. C-25 carbamate rifamycin derivatives with activity against drug-resistant microbes
PT1698630E (pt) 2005-03-03 2014-09-15 Alfa Wassermann Spa Novas formas polimorfas de rifaximina, processos para a sua produção e a sua utilização nas preparações medicinais
CN101282981B (zh) * 2005-08-11 2012-09-26 塔甘塔治疗公司 膦酸化利福霉素及其在预防和治疗骨和关节感染中的用途
IT1397617B1 (it) * 2009-04-20 2013-01-18 Alfa Wassermann Spa Nuovi derivati della rifamicina
PL2882435T3 (pl) * 2012-08-13 2021-10-04 Adipharm Ead Preparaty farmaceutyczne zawierające 3-(4-cynamylo-L-piperazynylo)-aminopochodne 3-formyloryfamycyny S
CN110770244A (zh) 2017-06-26 2020-02-07 倍尔福股份公司 吡啶并咪唑利福霉素衍生物的抗菌剂

Also Published As

Publication number Publication date
MX386622B (es) 2025-03-19
EP3645539A1 (en) 2020-05-06
ES2868180T3 (es) 2021-10-21
EP3645539B1 (en) 2021-04-07
DK3645539T3 (da) 2021-05-10
US11028086B2 (en) 2021-06-08
RU2020102511A3 (pl) 2021-07-27
US20200157104A1 (en) 2020-05-21
RU2020102511A (ru) 2021-07-27
CN110770244A (zh) 2020-02-07
US20210363143A1 (en) 2021-11-25
MX2019015681A (es) 2020-02-26
WO2019003076A1 (en) 2019-01-03
HUE054832T2 (hu) 2021-10-28

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