PL366315A1 - Antagoniści receptora IL-8 - Google Patents

Antagoniści receptora IL-8

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Publication number
PL366315A1
PL366315A1 PL01366315A PL36631501A PL366315A1 PL 366315 A1 PL366315 A1 PL 366315A1 PL 01366315 A PL01366315 A PL 01366315A PL 36631501 A PL36631501 A PL 36631501A PL 366315 A1 PL366315 A1 PL 366315A1
Authority
PL
Poland
Prior art keywords
receptor antagonists
antagonists
receptor
Prior art date
Application number
PL01366315A
Other languages
English (en)
Other versions
PL205103B1 (pl
Inventor
Michael Robert Palovich
Katherine Louisa Widdowson
Hong Nie
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of PL366315A1 publication Critical patent/PL366315A1/pl
Publication of PL205103B1 publication Critical patent/PL205103B1/pl

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    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • C07C311/64—X and Y being nitrogen atoms, e.g. N-sulfonylguanidine
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PL366315A 2000-03-24 2001-03-23 Pochodne cyjanoguanidyny, kompozycja farmaceutyczna zawierająca taki związek oraz jego zastosowanie PL205103B1 (pl)

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CO5170528A1 (es) * 1999-05-28 2002-06-27 Smithkline Beecham Corp Antagonistas de los receptores de la il-8 nistas del recpetor de la il-8
TW200418812A (en) * 2002-10-29 2004-10-01 Smithkline Beecham Corp IL-8 receptor antagonists
WO2005113534A2 (en) 2004-05-12 2005-12-01 Schering Corporation Cxcr1 and cxcr2 chemokine antagonists
WO2006043950A1 (en) * 2004-10-20 2006-04-27 Smithkline Beecham Corporation Il-8 receptor antagonists
AR060562A1 (es) * 2006-04-21 2008-06-25 Smithkline Beecham Corp Compuestos heterociclicos como antagonistas del receptor il-8. procesos de obtencion y composiciones farmaceuticas.
US8097626B2 (en) * 2006-04-21 2012-01-17 Glaxosmithkline Llc IL-8 receptor antagonists
AR061571A1 (es) * 2006-06-23 2008-09-03 Smithkline Beecham Corp Compuesto sal del acido toluenosulfonico de 4-{[6-cloro-3-({[(2- cloro-3-fluorofenil) amino]carbonil} amino)- 2- hidroxifenil]sulfonil] -1- piperazinacarbxilato de 1.1-dimetiletilo, composicion farmaceutica que lo comprende su uso para la fabricacion de un medicamento combinacion farmaceutica con un
US20090131329A1 (en) * 2007-09-14 2009-05-21 Edmund John Miller Treatment for allograft rejection
CN106243023A (zh) * 2010-09-03 2016-12-21 福马Tm有限责任公司 用于抑制nampt的胍化合物和组合物
US8648070B2 (en) 2010-12-17 2014-02-11 Boehringer Ingelheim International Gmbh Bicyclic ring system substituted sulfonamide functionalised phenols as medicaments
BR112014027700A2 (pt) * 2012-05-08 2017-06-27 Ishihara Sangyo Kaisha método para produção de um composto de ácido benzoico substituído
CA3128946A1 (en) 2019-02-07 2020-08-13 Bayer Aktiengesellschaft 3-amino-2-[2-(acylamino)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one as csnk1 inhibitors

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EP0809492A4 (en) * 1995-02-17 2007-01-24 Smithkline Beecham Corp IL-8 RECEPTOR ANTAGONISTS
AR008290A1 (es) 1996-08-15 1999-12-29 Smithkline Beecham Corp Nuevos compuestos que contienen guanidina utiles como antagonistas de los receptores de il-8, composiciones farmaceuticas que los contienenprocedimiento para la preparacion de dichos compuestos y procedimiento para la preparacion de intermediarios.
ES2194547T3 (es) * 1998-09-23 2003-11-16 Tularik Inc Arilsulfonanilida-ureas.
UY25842A1 (es) * 1998-12-16 2001-04-30 Smithkline Beecham Corp Antagonistas de receptores de il-8

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AP1548A (en) 2006-01-16
AU2001249354A1 (en) 2001-10-08
ES2344587T3 (es) 2010-09-01
WO2001072960A3 (en) 2002-02-21
ATE464893T1 (de) 2010-05-15
US20030216375A1 (en) 2003-11-20
CA2403787A1 (en) 2001-10-04
US6680317B2 (en) 2004-01-20
BG107035A (bg) 2003-04-30
MA25739A1 (fr) 2003-04-01
ZA200207576B (en) 2004-04-08
EP1272175A4 (en) 2005-08-31
SK13682002A3 (sk) 2003-06-03
EA200201019A1 (ru) 2003-12-25
MXPA02009355A (es) 2003-02-12
DE60141896D1 (de) 2010-06-02
AR031101A1 (es) 2003-09-10
WO2001072960A2 (en) 2001-10-04
BR0108867A (pt) 2005-02-09
OA12235A (en) 2003-11-06
DZ3333A1 (fr) 2001-10-04
EP1272175B1 (en) 2010-04-21
PE20020839A1 (es) 2002-12-04
PL205103B1 (pl) 2010-03-31
NO20024554D0 (no) 2002-09-23
HK1053789A1 (zh) 2003-11-07
UY26627A1 (es) 2001-09-28
EP1272175A2 (en) 2003-01-08
MY128154A (en) 2007-01-31
HUP0302614A3 (en) 2005-05-30
CZ20023192A3 (cs) 2003-02-12
JP2004508287A (ja) 2004-03-18
AP2002002599A0 (en) 2002-09-30
HUP0302614A2 (hu) 2003-11-28
IL151210A0 (en) 2003-04-10
KR20040014901A (ko) 2004-02-18
CN1452483A (zh) 2003-10-29

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