PL366541A1 - Granularne preparaty gaboksadolu - Google Patents

Granularne preparaty gaboksadolu

Info

Publication number: PL366541A1
Authority: PL; Poland
Prior art keywords: gaboxadol; granular preparations; granular; preparations
Prior art date: 2001-05-21

Application number

PL02366541A

Other languages

English (en)

Inventor

Michiel Onne Elema

Lene Andersen

Per Holm

Original Assignee

H.Lundbeck A/S

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-21

Filing date

2002-05-17

Publication date

2005-02-07

2002-05-17 Application filed by H.Lundbeck A/S filed Critical H.Lundbeck A/S

2005-02-07 Publication of PL366541A1 publication Critical patent/PL366541A1/pl

Links

ZXRVKCBLGJOCEE-UHFFFAOYSA-N Gaboxadol Chemical compound C1NCCC2=C1ONC2=O ZXRVKCBLGJOCEE-UHFFFAOYSA-N 0.000 title 1
229950004346 gaboxadol Drugs 0.000 title 1
238000002360 preparation method Methods 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Inorganic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Anesthesiology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

PL02366541A 2001-05-21 2002-05-17 Granularne preparaty gaboksadolu PL366541A1 (pl)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DKPA200100817		2001-05-21

Publications (1)

Publication Number	Publication Date
PL366541A1 true PL366541A1 (pl)	2005-02-07

Family

ID=8160520

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL02366541A PL366541A1 (pl)	2001-05-21	2002-05-17	Granularne preparaty gaboksadolu

Country Status (26)

Country	Link
US (1)	US20040157876A1 (pl)
EP (1)	EP1389091A1 (pl)
JP (1)	JP2004530695A (pl)
KR (1)	KR20030097890A (pl)
CN (1)	CN1511026A (pl)
AR (1)	AR033896A1 (pl)
AU (1)	AU2002338855B2 (pl)
BG (1)	BG108441A (pl)
BR (1)	BR0209834A (pl)
CA (1)	CA2447603A1 (pl)
CZ (1)	CZ20033269A3 (pl)
EA (2)	EA009731B1 (pl)
HR (1)	HRP20030950A2 (pl)
HU (1)	HUP0400051A2 (pl)
IL (1)	IL158733A0 (pl)
IS (1)	IS7020A (pl)
ME (1)	MEP6308A (pl)
MX (1)	MXPA03010596A (pl)
NO (1)	NO20035146D0 (pl)
NZ (1)	NZ547636A (pl)
PL (1)	PL366541A1 (pl)
SK (1)	SK15542003A3 (pl)
UA (1)	UA80092C2 (pl)
WO (1)	WO2002094225A1 (pl)
YU (1)	YU92103A (pl)
ZA (1)	ZA200308594B (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU7405000A (en) *	1999-09-28	2001-04-30	H. Lundbeck A/S	Melt granulated composition and modified release dosage form prepared from said composition
EP1641456B1 (en)	2003-06-25	2010-03-03	H. Lundbeck A/S	Gaboxadol for treating depression and other affective disorders
TW200528098A (en) *	2003-12-18	2005-09-01	Lundbeck & Co As H	Treatment of insomnia in human patients
GB0402118D0 (en)	2004-01-30	2004-03-03	Merck Sharp & Dohme	Polymorphic forms of a GABAA agonist
US8022084B2 (en)	2005-01-28	2011-09-20	H. Lundbeck A/S	Polymorphic forms of a GABAA agonist
EP1906953A4 (en) *	2005-04-29	2009-05-20	Lundbeck & Co As H	ACID AND BASE SALT FORMS OF GABOXADOL
AU2009255333B2 (en) *	2008-05-30	2015-07-09	Psychogenics, Inc.	Treatment for neurological and mental disorders
EP2334299A1 (en) *	2008-09-01	2011-06-22	H. Lundbeck A/S	Pharmaceutical composition comprising gaboxadol and an inhibitor of patl or oat
WO2013090452A1 (en)	2011-12-12	2013-06-20	Orbis Biosciences, Inc.	Sustained release particle formulations
IL256912B2 (en)	2015-07-17	2024-01-01	Ovid Therapeutics Inc	Methods of treating developmental disorders with gaboxadol

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4315934A (en) *	1979-09-24	1982-02-16	Sandoz Ltd.	Organic compounds
DE19525598C2 (de) *	1995-07-13	1997-09-25	Max Planck Gesellschaft	Schlafmittel
US6649186B1 (en) *	1996-09-20	2003-11-18	Ethypharm	Effervescent granules and methods for their preparation
AU7405000A (en) *	1999-09-28	2001-04-30	H. Lundbeck A/S	Melt granulated composition and modified release dosage form prepared from said composition
US6375982B1 (en) *	2000-07-05	2002-04-23	Capricorn Pharma, Inc.	Rapid-melt semi-solid compositions, methods of making same and method of using same

2002
- 2002-05-17 WO PCT/DK2002/000332 patent/WO2002094225A1/en not_active Ceased
- 2002-05-17 AR ARP020101839A patent/AR033896A1/es unknown
- 2002-05-17 PL PL02366541A patent/PL366541A1/pl not_active Application Discontinuation
- 2002-05-17 EA EA200301282A patent/EA009731B1/ru not_active IP Right Cessation
- 2002-05-17 CA CA002447603A patent/CA2447603A1/en not_active Abandoned
- 2002-05-17 HR HR20030950A patent/HRP20030950A2/hr not_active Application Discontinuation
- 2002-05-17 CZ CZ20033269A patent/CZ20033269A3/cs unknown
- 2002-05-17 BR BR0209834-2A patent/BR0209834A/pt not_active IP Right Cessation
- 2002-05-17 UA UA20031110120A patent/UA80092C2/uk unknown
- 2002-05-17 EP EP02742834A patent/EP1389091A1/en not_active Ceased
- 2002-05-17 NZ NZ547636A patent/NZ547636A/en unknown
- 2002-05-17 JP JP2002590944A patent/JP2004530695A/ja active Pending
- 2002-05-17 YU YU92103A patent/YU92103A/sh unknown
- 2002-05-17 SK SK1554-2003A patent/SK15542003A3/sk not_active Application Discontinuation
- 2002-05-17 AU AU2002338855A patent/AU2002338855B2/en not_active Ceased
- 2002-05-17 HU HU0400051A patent/HUP0400051A2/hu unknown
- 2002-05-17 US US10/478,983 patent/US20040157876A1/en not_active Abandoned
- 2002-05-17 CN CNA028104587A patent/CN1511026A/zh active Pending
- 2002-05-17 EA EA200700703A patent/EA200700703A1/ru unknown
- 2002-05-17 MX MXPA03010596A patent/MXPA03010596A/es not_active Application Discontinuation
- 2002-05-17 IL IL15873302A patent/IL158733A0/xx unknown
- 2002-05-17 ME MEP-63/08A patent/MEP6308A/xx unknown
- 2002-05-17 KR KR10-2003-7015136A patent/KR20030097890A/ko not_active Ceased
2003
- 2003-11-04 ZA ZA200308594A patent/ZA200308594B/en unknown
- 2003-11-10 IS IS7020A patent/IS7020A/is unknown
- 2003-11-19 NO NO20035146A patent/NO20035146D0/no not_active Application Discontinuation
- 2003-12-12 BG BG108441A patent/BG108441A/xx unknown

Also Published As

Publication number	Publication date
SK15542003A3 (sk)	2004-05-04
MEP6308A (xx)	2010-02-10
HUP0400051A2 (hu)	2004-04-28
WO2002094225A1 (en)	2002-11-28
NZ547636A (en)	2008-03-28
AU2002338855B2 (en)	2007-08-16
MXPA03010596A (es)	2004-03-09
AR033896A1 (es)	2004-01-07
UA80092C2 (en)	2007-08-27
EA009731B1 (ru)	2008-02-28
NO20035146L (no)	2003-11-19
JP2004530695A (ja)	2004-10-07
US20040157876A1 (en)	2004-08-12
ZA200308594B (en)	2004-11-04
NO20035146D0 (no)	2003-11-19
BG108441A (en)	2005-02-28
EA200700703A1 (ru)	2007-08-31
IS7020A (is)	2003-11-10
HRP20030950A2 (en)	2005-08-31
CZ20033269A3 (en)	2004-03-17
EA200301282A1 (ru)	2004-04-29
KR20030097890A (ko)	2003-12-31
YU92103A (sh)	2006-05-25
IL158733A0 (en)	2004-05-12
CN1511026A (zh)	2004-07-07
CA2447603A1 (en)	2002-11-28
BR0209834A (pt)	2004-06-15
EP1389091A1 (en)	2004-02-18

Legal Events

Date	Code	Title	Description
2009-10-30	REFS	Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)

Publication	Publication Date	Title
PT1438306E (pt)	2014-06-03	Derivados de uk-20
EP1578910A4 (en)	2008-06-04	NITRILASES
GB2376583B (en)	2005-01-05	Time alignment of signals
IL157426A0 (en)	2004-03-28	Peg-conjugates of hgf-nk4
EP1434772A4 (en)	2005-05-04	CONNECTIONS AND METHODS
IL158733A0 (en)	2004-05-12	Granular preparations of gaboxadol
GB0126889D0 (en)	2002-01-02	Compounds and their uses
AU2002359694A8 (en)	2003-06-30	Compounds and methods
HUP0500734A3 (en)	2005-12-28	Use of 2-alkoxyphenyl-substituted imidazotriazinones
GB0125708D0 (en)	2001-12-19	Novel compounds and processes
IL161178A0 (en)	2004-08-31	MODIFICATIONS OF SOLID 3-sn-PHOSPHOGLYCERIDES
AU2002358719A1 (en)	2003-07-15	Agaricoglycerides and analogs
EP1379240A4 (en)	2009-04-08	CONNECTIONS AND METHODS
AU2003298725A8 (en)	2004-06-23	Preparation of metallotexaphyrins
GB0100151D0 (en)	2001-02-14	Methods of sputtering
TW493722U (en)	2002-07-01	Improved structure of lampwick
IL157243A0 (en)	2004-02-19	Preparation of n-methylparoxetine and related intermediate compounds
AU2002359898A1 (en)	2003-07-24	Preparation of alpha-diimines
AU150489S (en)	2003-01-31	Set of chamfered logs
HU0104370D0 (en)	2001-12-28	Honeyed schnaps of oerseg
TW573751U (en)	2004-01-21	Structure capable of preventing jaming
IL165356A0 (en)	2006-01-15	Preparation of 4-haloalkylkylnicotinamides
AU2002300773A1 (en)	2003-06-12	Preparation of Dialkylpyridylboranes
GB0104615D0 (en)	2001-04-11	Treatment of technetium
GB0105097D0 (en)	2001-04-18	Treatment of technetium