PL371340A1 - Sposób wytwarzania kryształów sterydów, kryształydające się otrzymać tym sposobem i ich zastosowanie w preparatach farmaceutycznych - Google Patents

Sposób wytwarzania kryształów sterydów, kryształydające się otrzymać tym sposobem i ich zastosowanie w preparatach farmaceutycznych

Info

Publication number
PL371340A1
PL371340A1 PL03371340A PL37134003A PL371340A1 PL 371340 A1 PL371340 A1 PL 371340A1 PL 03371340 A PL03371340 A PL 03371340A PL 37134003 A PL37134003 A PL 37134003A PL 371340 A1 PL371340 A1 PL 371340A1
Authority
PL
Poland
Prior art keywords
crystals
mum
pharmaceutical formulations
steroid
crystals obtained
Prior art date
Application number
PL03371340A
Other languages
English (en)
Inventor
Detlef Grawe
Hagen Gerecke
Peter Hösel
Annette Eichardt
Sabine Gliesing
Uwe Müller
Original Assignee
Schering Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Aktiengesellschaft filed Critical Schering Aktiengesellschaft
Publication of PL371340A1 publication Critical patent/PL371340A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0085—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being a saturated hydrocarbon group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
PL03371340A 2002-04-23 2003-04-22 Sposób wytwarzania kryształów sterydów, kryształydające się otrzymać tym sposobem i ich zastosowanie w preparatach farmaceutycznych PL371340A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10218107A DE10218107A1 (de) 2002-04-23 2002-04-23 Verfahren zum Herstellen von Kristallen von Steroiden, danach erhältliche Kristalle und deren Verwendung in pharmazeutischen Formulierungen

Publications (1)

Publication Number Publication Date
PL371340A1 true PL371340A1 (pl) 2005-06-13

Family

ID=29264787

Family Applications (1)

Application Number Title Priority Date Filing Date
PL03371340A PL371340A1 (pl) 2002-04-23 2003-04-22 Sposób wytwarzania kryształów sterydów, kryształydające się otrzymać tym sposobem i ich zastosowanie w preparatach farmaceutycznych

Country Status (20)

Country Link
US (1) US7148212B2 (pl)
EP (1) EP1497308B1 (pl)
JP (1) JP4490116B2 (pl)
KR (1) KR20040106380A (pl)
CN (1) CN1646555A (pl)
AT (1) ATE340186T1 (pl)
AU (1) AU2003232491A1 (pl)
BR (1) BR0309357A (pl)
CA (1) CA2480004C (pl)
DE (2) DE10218107A1 (pl)
DK (1) DK1497308T3 (pl)
ES (1) ES2274258T3 (pl)
IL (1) IL163986A0 (pl)
MX (1) MXPA04010467A (pl)
NO (1) NO20045023L (pl)
PL (1) PL371340A1 (pl)
PT (1) PT1497308E (pl)
RU (1) RU2315056C2 (pl)
WO (1) WO2003091272A1 (pl)
ZA (1) ZA200409401B (pl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10218109A1 (de) * 2002-04-23 2003-11-20 Jenapharm Gmbh Verfahren zum Herstellen von Kristallen, danach erhältliche Kristalle und deren Verwendung in pharmazeutischen Formulierungen
SI1886694T1 (sl) * 2006-08-10 2009-10-31 Bayer Schering Pharma Ag Peroralna medikamentna oblika z dienogestom in etinilestradiolom za kontracepcijo
US20080038350A1 (en) * 2006-08-10 2008-02-14 Hagen Gerecke Low-dosage peroral medication for contraception containing crystalline dienogest and ethinyl estradiol
DE102008037025C5 (de) 2008-08-08 2016-07-07 Jesalis Pharma Gmbh Verfahren zur Herstellung kristalliner Wirkstoff-Mikropartikel bzw. einer Wirkstoffpartikel-Festkörperform
DE102010003711B4 (de) 2010-04-08 2015-04-09 Jesalis Pharma Gmbh Verfahren zur Herstellung kristalliner Wirkstoffpartikel
RU2642244C2 (ru) * 2010-04-12 2018-01-24 Кларус Терапеутикс, Инк. Оральные фармацевтические композиции сложных эфиров тестостерона и способы лечения недостатка тестостерона с их использованием
US9034858B2 (en) 2010-11-30 2015-05-19 Lipocine Inc. High-strength testosterone undecanoate compositions
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
CA2947459A1 (en) 2014-05-13 2015-11-19 Akzo Nobel Chemicals International B.V. Process to crystallize chelating agents
US20160361322A1 (en) 2015-06-15 2016-12-15 Lipocine Inc. Composition and method for oral delivery of androgen prodrugs
US20180147215A1 (en) 2016-11-28 2018-05-31 Lipocine Inc. Oral testosterone undecanoate therapy
US12150945B2 (en) 2018-07-20 2024-11-26 Lipocine Inc. Liver disease
EP4151219A4 (en) 2020-05-15 2024-05-15 Shionogi & Co., Ltd DRUG COMPOSITION WITH INHIBITED IMPURITIES PRODUCTION

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3226389A (en) * 1962-01-04 1965-12-28 Du Pont 11,11,12,12-tetracyano-naphtho-2,6-quinodimethan and its anion-radical salts
AU624421B2 (en) 1988-10-05 1992-06-11 Pharmacia & Upjohn Company Finely divided solid crystalline powders via precipitation into an anti-solvent
DE3917617A1 (de) * 1989-05-31 1990-12-06 Boehringer Ingelheim Kg Mikronisierte bioabbaubare partikel, verfahren zur ihrer herstellung und ihre verwendung
FR2668945B1 (fr) * 1990-11-12 1993-02-19 Theramex Nouveau procede de cristallisation des substances organiques et les composes ainsi obtenus.
DE69227850T2 (de) 1991-07-10 1999-04-29 Chiyoda Corp., Yokohama Verfahren zur Herstellung eines Kristallinadduktes von Bisphenol A mit Phenol
NZ248813A (en) * 1992-11-25 1995-06-27 Eastman Kodak Co Polymeric grinding media used in grinding pharmaceutical substances
DE4332283A1 (de) * 1993-09-20 1995-04-13 Jenapharm Gmbh Neue 11-Benzaldoximestradien-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
KR0151363B1 (ko) * 1993-12-27 1998-10-01 시모무라 스스무 4-히드록시-4'-이소프로폭시디페닐 술폰 현상조성물, 습식분쇄방법, 및 분산액
US5718388A (en) * 1994-05-25 1998-02-17 Eastman Kodak Continuous method of grinding pharmaceutical substances
US5534270A (en) * 1995-02-09 1996-07-09 Nanosystems Llc Method of preparing stable drug nanoparticles
CN1183102C (zh) * 1998-12-25 2005-01-05 第一精密化学株式会社 泛酸钙的制备方法
EP1157996A1 (de) * 2000-05-23 2001-11-28 JENAPHARM GmbH Neue Festkörperformen des Mesoprogestins 11Beta-[4E-(Hydroxyiminomethyl)-phenyl]-17Alpha-methoxymethyl-17Beta-methoxy-estra-4,9-dien-3-on
DE10218109A1 (de) * 2002-04-23 2003-11-20 Jenapharm Gmbh Verfahren zum Herstellen von Kristallen, danach erhältliche Kristalle und deren Verwendung in pharmazeutischen Formulierungen

Also Published As

Publication number Publication date
RU2315056C2 (ru) 2008-01-20
US7148212B2 (en) 2006-12-12
DE50305122D1 (de) 2006-11-02
JP2005524698A (ja) 2005-08-18
ATE340186T1 (de) 2006-10-15
CN1646555A (zh) 2005-07-27
ZA200409401B (en) 2006-02-22
EP1497308A1 (de) 2005-01-19
ES2274258T3 (es) 2007-05-16
RU2004134324A (ru) 2006-02-10
EP1497308B1 (de) 2006-09-20
JP4490116B2 (ja) 2010-06-23
NO20045023L (no) 2004-11-18
KR20040106380A (ko) 2004-12-17
CA2480004A1 (en) 2003-11-06
DK1497308T3 (da) 2007-01-29
AU2003232491A1 (en) 2003-11-10
DE10218107A1 (de) 2003-11-20
MXPA04010467A (es) 2004-12-13
PT1497308E (pt) 2007-01-31
BR0309357A (pt) 2005-02-22
WO2003091272A1 (de) 2003-11-06
IL163986A0 (en) 2005-12-18
US20030216360A1 (en) 2003-11-20
CA2480004C (en) 2007-11-13

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Legal Events

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REFS Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)