PL414227A1 - Dimeryczne pochodne alkaloidów drzewa chinowego, sposób ich otrzymywania oraz ich zastosowanie - Google Patents
Dimeryczne pochodne alkaloidów drzewa chinowego, sposób ich otrzymywania oraz ich zastosowanieInfo
- Publication number
- PL414227A1 PL414227A1 PL414227A PL41422715A PL414227A1 PL 414227 A1 PL414227 A1 PL 414227A1 PL 414227 A PL414227 A PL 414227A PL 41422715 A PL41422715 A PL 41422715A PL 414227 A1 PL414227 A1 PL 414227A1
- Authority
- PL
- Poland
- Prior art keywords
- application
- derivatives
- dimeric
- cinchona
- obtaining
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 229930013930 alkaloid Natural products 0.000 title 1
- KAKZBPTYRLMSJV-UHFFFAOYSA-N Butadiene Chemical compound C=CC=C KAKZBPTYRLMSJV-UHFFFAOYSA-N 0.000 abstract 2
- LOUPRKONTZGTKE-WZBLMQSHSA-N Quinine Chemical class C([C@H]([C@H](C1)C=C)C2)C[N@@]1[C@@H]2[C@H](O)C1=CC=NC2=CC=C(OC)C=C21 LOUPRKONTZGTKE-WZBLMQSHSA-N 0.000 abstract 2
- VMQMZMRVKUZKQL-UHFFFAOYSA-N Cu+ Chemical compound [Cu+] VMQMZMRVKUZKQL-UHFFFAOYSA-N 0.000 abstract 1
- 238000006736 Huisgen cycloaddition reaction Methods 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 150000003797 alkaloid derivatives Chemical class 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 239000002243 precursor Substances 0.000 abstract 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 abstract 1
- 229920002554 vinyl polymer Polymers 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Zgłoszenie dotyczy nowych dimerycznych pochodnych alkaloidów drzewa chinowego, złączonych ugrupowaniem bitriazolowym, przedstawionymi wzorem ogólnym 1, w którym R3 stanowi grupę winylową lub etylową, a R6' grupę metoksylową lub wodór. Przedmiotem zgłoszenia jest również sposób wytwarzania dimerycznych pochodnych alkaloidów, który polega na tym, że 9-azydo-9-deoksy-pochodną lub 9-epi-9-azydo-9-deoksy-pochodną alkaloidu drzewa chinowego poddaje się reakcji z prekursorem butadiynu w katalizowanej miedzią (I) reakcji podwójnej 1,3-dipolarnej cykloaddycji.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL414227A PL226006B1 (pl) | 2015-10-02 | 2015-10-02 | Dimeryczne pochodne alkaloidow drzewa chinowego, sposob ich otrzymywania oraz ich zastosowanie |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL414227A PL226006B1 (pl) | 2015-10-02 | 2015-10-02 | Dimeryczne pochodne alkaloidow drzewa chinowego, sposob ich otrzymywania oraz ich zastosowanie |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL414227A1 true PL414227A1 (pl) | 2016-07-18 |
| PL226006B1 PL226006B1 (pl) | 2017-06-30 |
Family
ID=56370120
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL414227A PL226006B1 (pl) | 2015-10-02 | 2015-10-02 | Dimeryczne pochodne alkaloidow drzewa chinowego, sposob ich otrzymywania oraz ich zastosowanie |
Country Status (1)
| Country | Link |
|---|---|
| PL (1) | PL226006B1 (pl) |
-
2015
- 2015-10-02 PL PL414227A patent/PL226006B1/pl unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PL226006B1 (pl) | 2017-06-30 |
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