PL4219455T3 - Sposób wytwarzania fluorowcowanego pirazolu - Google Patents

Sposób wytwarzania fluorowcowanego pirazolu

Info

Publication number: PL4219455T3
Authority: PL; Poland
Prior art keywords: preparation; methods; halogenated pyrazole; pyrazole; halogenated
Prior art date: 2019-10-18

Application number

PL23166843.5T

Other languages

English (en)

Inventor

Yanchun Cao

Xin Liu

Jianhua Mao

Zhijian Xu

Original Assignee

Fmc Corporation

Fmc Ip Technology Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2019-10-18

Filing date

2020-10-16

Publication date

2025-04-14

2020-10-16 Application filed by Fmc Corporation, Fmc Ip Technology Gmbh filed Critical Fmc Corporation

2025-04-14 Publication of PL4219455T3 publication Critical patent/PL4219455T3/pl

Links

150000003217 pyrazoles Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

PL23166843.5T 2019-10-18 2020-10-16 Sposób wytwarzania fluorowcowanego pirazolu PL4219455T3 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US201962916840P	2019-10-18	2019-10-18
US202062982248P	2020-02-27	2020-02-27

Publications (1)

Publication Number	Publication Date
PL4219455T3 true PL4219455T3 (pl)	2025-04-14

Family

ID=73198483

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
PL20804069.1T PL3976589T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2H-pirazolo-3-karboksylowego
PL20804381.0T PL3976591T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2h- pirazolo-3-karboksylowego
PL23166843.5T PL4219455T3 (pl)	2019-10-18	2020-10-16	Sposób wytwarzania fluorowcowanego pirazolu
PL22161905.9T PL4043451T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania związku pośredniego w syntezie kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2h-pirazolo-3-karboksylowego

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
PL20804069.1T PL3976589T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2H-pirazolo-3-karboksylowego
PL20804381.0T PL3976591T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2h- pirazolo-3-karboksylowego

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
PL22161905.9T PL4043451T3 (pl)	2019-10-18	2020-10-16	Sposoby wytwarzania związku pośredniego w syntezie kwasu 5-bromo-2-(3-chloropirydyn-2-ylo)-2h-pirazolo-3-karboksylowego

Country Status (17)

Country	Link
US (2)	US20220396560A1 (pl)
EP (5)	EP4043451B1 (pl)
JP (2)	JP7667144B2 (pl)
KR (2)	KR20220086612A (pl)
CN (3)	CN119039270A (pl)
AU (2)	AU2020366037A1 (pl)
BR (2)	BR112022007102A2 (pl)
HU (4)	HUE062237T2 (pl)
IL (5)	IL299818B2 (pl)
MA (2)	MA56053A (pl)
MX (2)	MX2022004631A (pl)
PL (4)	PL3976589T3 (pl)
PY (1)	PY2065468A (pl)
TW (3)	TWI884994B (pl)
UY (1)	UY38925A (pl)
WO (2)	WO2021076839A1 (pl)
ZA (2)	ZA202204277B (pl)

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EP4045487B1 (en) *	2019-10-18	2025-02-12	Fmc Corporation	Methods for the preparation of 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylic acid
AU2020366037A1 (en) *	2019-10-18	2022-04-21	Fmc Corporation	Methods for the preparation of 5-bromo-2-(3-chloro-pyridin-2-yl)-2H-pyrazole-3-carboxylic acid
CN115557931B (zh) *	2022-10-20	2024-05-14	浙江新安化工集团股份有限公司	一种3-溴-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酸的合成方法
CN117024374A (zh) *	2023-08-08	2023-11-10	安庆百谊生物科技有限公司	一种3-甲基-1，2，4-噻二唑-5-碳酰肼或其盐的合成方法

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CN111825653A (zh) *	2019-04-19	2020-10-27	安道麦马克西姆有限公司	取代吡唑类化合物的制备及其作为邻氨基苯甲酰胺前体的用途
AU2020366037A1 (en) *	2019-10-18	2022-04-21	Fmc Corporation	Methods for the preparation of 5-bromo-2-(3-chloro-pyridin-2-yl)-2H-pyrazole-3-carboxylic acid

2020
- 2020-10-16 AU AU2020366037A patent/AU2020366037A1/en active Pending
- 2020-10-16 JP JP2022521265A patent/JP7667144B2/ja active Active
- 2020-10-16 TW TW109135811A patent/TWI884994B/zh active
- 2020-10-16 EP EP22161905.9A patent/EP4043451B1/en active Active
- 2020-10-16 PL PL20804069.1T patent/PL3976589T3/pl unknown
- 2020-10-16 CN CN202411157026.7A patent/CN119039270A/zh active Pending
- 2020-10-16 PY PY202002065468A patent/PY2065468A/es unknown
- 2020-10-16 CN CN202080072845.5A patent/CN114650987B/zh active Active
- 2020-10-16 US US17/769,810 patent/US20220396560A1/en not_active Abandoned
- 2020-10-16 MA MA056053A patent/MA56053A/fr unknown
- 2020-10-16 BR BR112022007102A patent/BR112022007102A2/pt not_active Application Discontinuation
- 2020-10-16 KR KR1020227016245A patent/KR20220086612A/ko not_active Ceased
- 2020-10-16 KR KR1020227016372A patent/KR20220084347A/ko not_active Ceased
- 2020-10-16 IL IL299818A patent/IL299818B2/en unknown
- 2020-10-16 HU HUE20804381A patent/HUE062237T2/hu unknown
- 2020-10-16 BR BR112022007215A patent/BR112022007215A2/pt not_active Application Discontinuation
- 2020-10-16 PL PL20804381.0T patent/PL3976591T3/pl unknown
- 2020-10-16 MX MX2022004631A patent/MX2022004631A/es unknown
- 2020-10-16 WO PCT/US2020/055897 patent/WO2021076839A1/en not_active Ceased
- 2020-10-16 TW TW113140016A patent/TW202517625A/zh unknown
- 2020-10-16 PL PL23166843.5T patent/PL4219455T3/pl unknown
- 2020-10-16 MX MX2022004627A patent/MX2022004627A/es unknown
- 2020-10-16 MA MA056055A patent/MA56055A/fr unknown
- 2020-10-16 EP EP20804069.1A patent/EP3976589B1/en active Active
- 2020-10-16 EP EP23166843.5A patent/EP4219455B1/en active Active
- 2020-10-16 IL IL291939A patent/IL291939B2/en unknown
- 2020-10-16 HU HUE22161905A patent/HUE066520T2/hu unknown
- 2020-10-16 JP JP2022521266A patent/JP2022552273A/ja active Pending
- 2020-10-16 HU HUE23166843A patent/HUE070680T2/hu unknown
- 2020-10-16 IL IL294551A patent/IL294551B2/en unknown
- 2020-10-16 UY UY0001038925A patent/UY38925A/es unknown
- 2020-10-16 HU HUE20804069A patent/HUE062047T2/hu unknown
- 2020-10-16 CN CN202080072852.5A patent/CN114641471B/zh active Active
- 2020-10-16 AU AU2020366212A patent/AU2020366212A1/en active Pending
- 2020-10-16 EP EP23168298.0A patent/EP4253380A3/en not_active Withdrawn
- 2020-10-16 US US17/769,787 patent/US20220259178A1/en not_active Abandoned
- 2020-10-16 WO PCT/US2020/055888 patent/WO2021076835A1/en not_active Ceased
- 2020-10-16 IL IL298694A patent/IL298694B2/en unknown
- 2020-10-16 EP EP20804381.0A patent/EP3976591B1/en active Active
- 2020-10-16 TW TW109135805A patent/TWI875840B/zh active
- 2020-10-16 PL PL22161905.9T patent/PL4043451T3/pl unknown
2022
- 2022-04-10 IL IL292090A patent/IL292090B2/en unknown
- 2022-04-14 ZA ZA2022/04277A patent/ZA202204277B/en unknown
- 2022-04-14 ZA ZA2022/04278A patent/ZA202204278B/en unknown

Also Published As

Publication number	Publication date
IL298694B2 (en)	2025-05-01
IL298694B1 (en)	2025-01-01
IL292090A (en)	2022-06-01
TW202116748A (zh)	2021-05-01
CN114650987B (zh)	2024-09-06
HUE062047T2 (hu)	2023-09-28
ZA202204277B (en)	2024-08-28
MA56053A (fr)	2022-04-20
AU2020366037A1 (en)	2022-04-21
EP3976589B1 (en)	2023-04-12
EP4043451A1 (en)	2022-08-17
US20220396560A1 (en)	2022-12-15
IL294551B1 (en)	2023-01-01
EP4219455A1 (en)	2023-08-02
JP2022552273A (ja)	2022-12-15
US20220259178A1 (en)	2022-08-18
EP4253380A2 (en)	2023-10-04
IL299818B1 (en)	2024-10-01
TWI875840B (zh)	2025-03-11
AU2020366212A1 (en)	2022-04-21
EP4219455B1 (en)	2024-12-11
IL291939B (en)	2022-12-01
IL294551B2 (en)	2023-05-01
CN119039270A (zh)	2024-11-29
WO2021076835A1 (en)	2021-04-22
CN114641471B (zh)	2025-05-23
WO2021076835A8 (en)	2021-11-04
CN114641471A (zh)	2022-06-17
MX2022004627A (es)	2022-05-26
UY38925A (es)	2021-05-31
IL291939A (en)	2022-06-01
EP4043451B1 (en)	2024-02-28
EP3976589A1 (en)	2022-04-06
EP3976591B1 (en)	2023-04-19
IL299818B2 (en)	2025-02-01
EP3976591A1 (en)	2022-04-06
HUE066520T2 (hu)	2024-08-28
TWI884994B (zh)	2025-06-01
ZA202204278B (en)	2024-08-28
BR112022007102A2 (pt)	2022-07-05
MX2022004631A (es)	2022-05-24
BR112022007215A2 (pt)	2022-07-05
IL298694A (en)	2023-02-01
HUE070680T2 (hu)	2025-06-28
TW202128631A (zh)	2021-08-01
JP2022552272A (ja)	2022-12-15
PY2065468A (es)	2023-05-16
KR20220084347A (ko)	2022-06-21
PL3976589T3 (pl)	2023-07-31
TW202517625A (zh)	2025-05-01
KR20220086612A (ko)	2022-06-23
WO2021076839A1 (en)	2021-04-22
HUE062237T2 (hu)	2023-10-28
IL299818A (en)	2023-03-01
CN114650987A (zh)	2022-06-21
PL4043451T3 (pl)	2024-06-10
JP7667144B2 (ja)	2025-04-22
IL291939B2 (en)	2023-04-01
IL294551A (en)	2022-09-01
MA56055A (fr)	2022-04-06
EP4253380A3 (en)	2023-11-15
IL292090B2 (en)	2023-06-01
PL3976591T3 (pl)	2023-07-31

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