PL424865A1 - Derivatives of colchicine, method for producing them and applications - Google Patents
Derivatives of colchicine, method for producing them and applicationsInfo
- Publication number
- PL424865A1 PL424865A1 PL424865A PL42486518A PL424865A1 PL 424865 A1 PL424865 A1 PL 424865A1 PL 424865 A PL424865 A PL 424865A PL 42486518 A PL42486518 A PL 42486518A PL 424865 A1 PL424865 A1 PL 424865A1
- Authority
- PL
- Poland
- Prior art keywords
- colchicine
- derivatives
- demethoxy
- deacetyl
- iodo
- Prior art date
Links
- IAKHMKGGTNLKSZ-INIZCTEOSA-N (S)-colchicine Chemical class C1([C@@H](NC(C)=O)CC2)=CC(=O)C(OC)=CC=C1C1=C2C=C(OC)C(OC)=C1OC IAKHMKGGTNLKSZ-INIZCTEOSA-N 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 3
- 125000002346 iodo group Chemical group I* 0.000 abstract 3
- 125000001246 bromo group Chemical group Br* 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 229940044683 chemotherapy drug Drugs 0.000 abstract 1
- 229960001338 colchicine Drugs 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Przedmiotem zgłoszenia są N-karbaminianowe pochodne N-deacetylo-4-(bromo/chloro/jodo)-10-demetoksy-10-alkilotiokolchicyny o wzorze ogólnym 1, gdzie: X oznacza Cl, Br lub I; Y oznacza grupę alkilową prostą lub rozgałęzioną, zawierającą od 1 do 4 atomów węgla. Ponadto przedmiotem zgłoszenia jest sposób otrzymywania nowych N-karbaminianów N-deacetylo-4-(bromo/chloro/jodo)-10-demetoksy-10-alkilotiokolchicyny o wzorze ogólnym 1. Przedmiotem zgłoszenia jest też sposób otrzymywania nowych N-karbaminianów N-deacetylo-4-bromo/chloro/jodo)-10-demetoksy-10-alkilotio-kolchicyny o wzorze ogólnym 1, do sporządzania leków stosowanych w chemioterapii.The subject of the application are N-deacetyl-4- (bromo / chloro / iodo) -10-demethoxy-10-alkylthiocolchicine derivatives of general formula 1, where: X is Cl, Br or I; Y is a straight or branched alkyl group containing from 1 to 4 carbon atoms. In addition, the subject of the application is a method for the preparation of new N-deacetyl-4- (bromo / chloro / iodo) -10-demethoxy-10-alkylthiocolchicine N-carbamates of the general formula 1. The subject of the application is also a method for the preparation of new N-deacetyl- N-carbamates 4-bromo / chloro / iodo) -10-demethoxy-10-alkylthio-colchicine of general formula 1, for the preparation of chemotherapy drugs.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL424865A PL231213B1 (en) | 2018-03-13 | 2018-03-13 | Colchicine derivatives, method of their preparation and application |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL424865A PL231213B1 (en) | 2018-03-13 | 2018-03-13 | Colchicine derivatives, method of their preparation and application |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL424865A1 true PL424865A1 (en) | 2018-08-13 |
| PL231213B1 PL231213B1 (en) | 2019-02-28 |
Family
ID=63112925
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL424865A PL231213B1 (en) | 2018-03-13 | 2018-03-13 | Colchicine derivatives, method of their preparation and application |
Country Status (1)
| Country | Link |
|---|---|
| PL (1) | PL231213B1 (en) |
-
2018
- 2018-03-13 PL PL424865A patent/PL231213B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PL231213B1 (en) | 2019-02-28 |
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