PT100234A - Novos esteres de alcoois aminados biciclicos e triciclicos, processo para a sua preparacao - Google Patents

Novos esteres de alcoois aminados biciclicos e triciclicos, processo para a sua preparacao

Info

Publication number
PT100234A
PT100234A PT100234A PT10023492A PT100234A PT 100234 A PT100234 A PT 100234A PT 100234 A PT100234 A PT 100234A PT 10023492 A PT10023492 A PT 10023492A PT 100234 A PT100234 A PT 100234A
Authority
PT
Portugal
Prior art keywords
preparation
amino acid
acid esters
new bicyclic
tricyclic amino
Prior art date
Application number
PT100234A
Other languages
English (en)
Other versions
PT100234B (pt
Inventor
Rudolf Bauer
Richard Reichl
Rolf Banholzer
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of PT100234A publication Critical patent/PT100234A/pt
Publication of PT100234B publication Critical patent/PT100234B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
PT100234A 1991-03-15 1992-03-12 Novos esteres de alcoois aminados biciclicos e triciclicos, processo para a sua preparacao PT100234B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4108393A DE4108393A1 (de) 1991-03-15 1991-03-15 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln

Publications (2)

Publication Number Publication Date
PT100234A true PT100234A (pt) 1993-07-30
PT100234B PT100234B (pt) 1999-06-30

Family

ID=6427349

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100234A PT100234B (pt) 1991-03-15 1992-03-12 Novos esteres de alcoois aminados biciclicos e triciclicos, processo para a sua preparacao

Country Status (26)

Country Link
US (1) US5654314A (pt)
EP (1) EP0579615B1 (pt)
JP (1) JP3352684B2 (pt)
KR (1) KR100307274B1 (pt)
AT (1) ATE202778T1 (pt)
AU (1) AU662128B2 (pt)
CA (1) CA2105575C (pt)
CZ (1) CZ281509B6 (pt)
DE (2) DE4108393A1 (pt)
DK (1) DK0579615T3 (pt)
ES (1) ES2160577T3 (pt)
FI (1) FI120235B (pt)
GR (1) GR3036792T3 (pt)
HU (1) HU224210B1 (pt)
IE (1) IE920815A1 (pt)
IL (1) IL101225A (pt)
MX (1) MX9201139A (pt)
NO (1) NO304266B1 (pt)
NZ (1) NZ241961A (pt)
PL (1) PL179673B1 (pt)
PT (1) PT100234B (pt)
SG (1) SG43037A1 (pt)
SK (1) SK281511B6 (pt)
UA (1) UA29406C2 (pt)
WO (1) WO1992016528A1 (pt)
ZA (1) ZA921875B (pt)

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DE10211700A1 (de) * 2002-03-16 2003-09-25 Boehringer Ingelheim Pharma Neue Difurylglykolsäureester, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel
US20030229227A1 (en) * 2002-03-16 2003-12-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg New difurylglycolic acid esters, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions
US7309707B2 (en) * 2002-03-20 2007-12-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Crystalline micronisate, process for the manufacture thereof and use thereof for the preparation of a medicament
US7311894B2 (en) * 2002-03-28 2007-12-25 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations containing an anticholinergic
US7244415B2 (en) * 2002-03-28 2007-07-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations of an anhydrate
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US7084153B2 (en) 2002-04-12 2006-08-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments comprising steroids and a novel anticholinergic
US7417051B2 (en) 2002-04-12 2008-08-26 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments comprising betamimetics and a novel anticholinergic
PT1497289E (pt) * 2002-04-12 2005-11-30 Boehringer Ingelheim Pharma Farmaco contendo betamimeticos e um novo anticolinergico
DE10256317A1 (de) * 2002-04-12 2003-10-23 Boehringer Ingelheim Pharma Arzneimittel enthaltend Betamimetika und ein neues Anticholinergikum
DE10216429A1 (de) 2002-04-12 2003-10-23 Boehringer Ingelheim Pharma Arzneimittel enthaltend Steroide und ein neues Anticholinergikum
DE10216339A1 (de) * 2002-04-13 2003-10-23 Boehringer Ingelheim Pharma Neue Ester hydroxy-substituierter Stickstoffheterocyclen, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel
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DE10224091A1 (de) * 2002-05-31 2003-12-11 Boehringer Ingelheim Pharma Technisches Verfahren zur Herstellung von Tropenol
US20040048886A1 (en) * 2002-07-09 2004-03-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on new anticholinergics and NK1 receptor antagonists
DE10255040A1 (de) * 2002-11-26 2004-06-03 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Carbaminsäureester mit anticholinerger Wirksamkeit
US7763280B2 (en) * 2002-11-28 2010-07-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Tiotropium containing powder formulation for inhalation
AU2004206846B2 (en) * 2003-01-16 2009-05-28 University Of Rochester Quaternary antimuscarinic compounds for the treatment of bladder diseases
ATE435862T1 (de) * 2003-05-28 2009-07-15 Theravance Inc Azabicycloalkanverbindungen als muscarinrezeptor antagonisten
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JPWO2006025324A1 (ja) * 2004-08-30 2008-05-08 小野薬品工業株式会社 トロパン化合物およびそれらを有効成分として含有する医薬組成物
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Also Published As

Publication number Publication date
AU662128B2 (en) 1995-08-24
JPH06505718A (ja) 1994-06-30
DE4108393A1 (de) 1992-09-17
US5654314A (en) 1997-08-05
FI934000A0 (fi) 1993-09-13
DK0579615T3 (da) 2001-09-17
ES2160577T3 (es) 2001-11-16
HU224210B1 (hu) 2005-06-28
NO304266B1 (no) 1998-11-23
NZ241961A (en) 1995-07-26
EP0579615B1 (de) 2001-07-04
FI934000L (fi) 1993-09-13
SK94993A3 (en) 1994-04-06
MX9201139A (es) 1992-10-01
UA29406C2 (uk) 2000-11-15
CZ191793A3 (en) 1994-05-18
PT100234B (pt) 1999-06-30
SK281511B6 (sk) 2001-04-09
CZ281509B6 (cs) 1996-10-16
IE920815A1 (en) 1992-09-23
PL179673B1 (pl) 2000-10-31
GR3036792T3 (en) 2002-01-31
DE59209907D1 (de) 2001-08-09
HU9302611D0 (en) 1993-12-28
FI120235B (fi) 2009-08-14
ATE202778T1 (de) 2001-07-15
AU1345792A (en) 1992-10-21
IL101225A (en) 1996-05-14
NO933274D0 (no) 1993-09-14
CA2105575A1 (en) 1992-09-16
JP3352684B2 (ja) 2002-12-03
WO1992016528A1 (de) 1992-10-01
KR100307274B1 (ko) 2001-12-05
IL101225A0 (en) 1992-11-15
ZA921875B (en) 1993-09-13
NO933274L (no) 1993-11-12
EP0579615A1 (de) 1994-01-26
SG43037A1 (en) 1997-10-17
HUT65132A (en) 1994-04-28
CA2105575C (en) 2000-04-25

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