PT2988733T - Composição farmacêutica contendo macitentano cristalino - Google Patents

Composição farmacêutica contendo macitentano cristalino

Info

Publication number
PT2988733T
PT2988733T PT14721256T PT14721256T PT2988733T PT 2988733 T PT2988733 T PT 2988733T PT 14721256 T PT14721256 T PT 14721256T PT 14721256 T PT14721256 T PT 14721256T PT 2988733 T PT2988733 T PT 2988733T
Authority
PT
Portugal
Prior art keywords
pharmaceutical composition
composition containing
containing crystalline
crystalline macitentan
macitentan
Prior art date
Application number
PT14721256T
Other languages
English (en)
Inventor
Stefinovic Marijan
Raneburger Johannes
Englmeier Ludwig
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48143162&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2988733(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of PT2988733T publication Critical patent/PT2988733T/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
    • A61J1/00—Containers specially adapted for medical or pharmaceutical purposes
    • A61J1/03—Containers specially adapted for medical or pharmaceutical purposes for pills or tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
    • B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
    • B65D65/00—Wrappers or flexible covers; Packaging materials of special type or form
    • B65D65/38—Packaging materials of special type or form
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
    • B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
    • B65D2565/00—Wrappers or flexible covers; Packaging materials of special type or form
    • B65D2565/38—Packaging materials of special type or form
    • B65D2565/381—Details of packaging materials of special type or form
    • B65D2565/388—Materials used for their gas-permeability

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Mechanical Engineering (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT14721256T 2013-04-22 2014-04-17 Composição farmacêutica contendo macitentano cristalino PT2988733T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP13164724 2013-04-22

Publications (1)

Publication Number Publication Date
PT2988733T true PT2988733T (pt) 2019-06-04

Family

ID=48143162

Family Applications (1)

Application Number Title Priority Date Filing Date
PT14721256T PT2988733T (pt) 2013-04-22 2014-04-17 Composição farmacêutica contendo macitentano cristalino

Country Status (12)

Country Link
US (2) US9730932B2 (pt)
EP (1) EP2988733B1 (pt)
AU (2) AU2014257719B2 (pt)
CA (1) CA2908410A1 (pt)
DE (1) DE14721256T1 (pt)
DK (1) DK2988733T3 (pt)
ES (1) ES2729191T3 (pt)
HU (1) HUE043804T2 (pt)
PL (1) PL2988733T3 (pt)
PT (1) PT2988733T (pt)
TR (1) TR201906685T4 (pt)
WO (1) WO2014173805A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE14721256T1 (de) 2013-04-22 2017-03-16 Sandoz Ag Pharmazeutische zusammensetzungen mit kristallinem macitentan
CN105461638A (zh) * 2015-12-10 2016-04-06 合肥久诺医药科技有限公司 一种马西替坦晶型及其制备方法
WO2018153925A1 (en) 2017-02-22 2018-08-30 Amneal Pharmaceuticals Company Gmbh Stable pharmaceutical compositions comprising macitentan
AU2020309223B2 (en) * 2019-07-05 2025-05-29 TECNIMEDE - Sociedade Técnico-Medicinal, S.A Compressed macitentan compositions, methods and uses thereof
WO2022045991A1 (en) * 2020-08-26 2022-03-03 Pharmacti̇ve İlaç Sanayi̇ Ve Ti̇caret A.Ş. Pharmaceutical compositions comprising macitentan and relevant excipients
TR2021013983A1 (tr) * 2021-09-07 2023-03-21 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Masi̇tentan i̇çeren bi̇r kapsül formülasyonu
TR2021014838A2 (tr) * 2021-09-22 2023-04-24 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Masi̇tentan i̇çeren tablet
EP4154873A1 (en) * 2021-09-22 2023-03-29 Sanovel Ilac Sanayi Ve Ticaret A.S. The tablet comprising macitentan

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4721709A (en) * 1984-07-26 1988-01-26 Pyare Seth Novel pharmaceutical compositions containing hydrophobic practically water-insoluble drugs adsorbed on pharmaceutical excipients as carrier; process for their preparation and the use of said compositions
WO2002053557A1 (en) 2000-12-18 2002-07-11 Actelion Pharmaceuticals Ltd Novel sulfamides and their use as endothelin receptor antagonists
WO2007031933A2 (en) * 2005-09-12 2007-03-22 Actelion Pharmaceuticals Ltd Stable pharmaceutical composition comprising a pyrimidine-sulfamide
CA2659558A1 (en) * 2006-08-03 2008-02-07 Merck Patent Gesellschaft Mit Beschraenkter Haftung Pack containing pharmaceutical administration forms
DE14721256T1 (de) 2013-04-22 2017-03-16 Sandoz Ag Pharmazeutische zusammensetzungen mit kristallinem macitentan

Also Published As

Publication number Publication date
TR201906685T4 (tr) 2019-05-21
ES2729191T3 (es) 2019-10-30
WO2014173805A1 (en) 2014-10-30
AU2014257719B2 (en) 2016-07-07
DK2988733T3 (da) 2019-07-01
AU2016238890A1 (en) 2016-10-27
PL2988733T3 (pl) 2019-09-30
CA2908410A1 (en) 2014-10-30
EP2988733B1 (en) 2019-03-27
EP2988733A1 (en) 2016-03-02
AU2014257719A1 (en) 2015-09-17
US20180008603A1 (en) 2018-01-11
US20160074398A1 (en) 2016-03-17
US9730932B2 (en) 2017-08-15
HUE043804T2 (hu) 2019-09-30
DE14721256T1 (de) 2017-03-16

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