PT3700513T - Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações - Google Patents

Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações

Info

Publication number: PT3700513T
Authority: PT; Portugal
Prior art keywords: segrams; glucocorticoid receptor; receptor agonistic; selective glucocorticoid; steroidal selective
Prior art date: 2018-05-17

Application number

PT187868237T

Other languages

English (en)

Original Assignee

Association Pour La Rech A Ligbmc Ari

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2018-05-17

Filing date

2018-10-23

Publication date

2022-11-30

2018-10-23 Application filed by Association Pour La Rech A Ligbmc Ari filed Critical Association Pour La Rech A Ligbmc Ari

2022-11-30 Publication of PT3700513T publication Critical patent/PT3700513T/pt

Links

102000003676 Glucocorticoid Receptors Human genes 0.000 title 1
108090000079 Glucocorticoid Receptors Proteins 0.000 title 1
230000001270 agonistic effect Effects 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Dermatology (AREA)
Epidemiology (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Ophthalmology & Optometry (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Emergency Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Furan Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

PT187868237T 2018-05-17 2018-10-23 Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações PT3700513T (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP18305612.6A EP3569228A1 (en)	2018-05-17	2018-05-17	Non-steroidal selective glucocorticoid receptor agonistic modulators (segrams) and uses thereof

Publications (1)

Publication Number	Publication Date
PT3700513T true PT3700513T (pt)	2022-11-30

Family

ID=62386318

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT187868237T PT3700513T (pt)	2018-05-17	2018-10-23	Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações

Country Status (9)

Country	Link
US (1)	US11179363B2 (pt)
EP (2)	EP3569228A1 (pt)
JP (1)	JP2021509411A (pt)
KR (1)	KR20200085782A (pt)
CN (1)	CN111511359A (pt)
AU (1)	AU2018355698A1 (pt)
BR (1)	BR112020008350A2 (pt)
MA (1)	MA50443A (pt)
PT (1)	PT3700513T (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US12150922B1 (en)	2023-12-08	2024-11-26	King Faisal University	Methods of inhibiting cyclooxygenase (COX) using tolterodine

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5262165A (en)	1992-02-04	1993-11-16	Schering Corporation	Transdermal nitroglycerin patch with penetration enhancers
US6010715A (en)	1992-04-01	2000-01-04	Bertek, Inc.	Transdermal patch incorporating a polymer film incorporated with an active agent
CA2222133C (en)	1995-06-07	2002-12-24	Cygnus, Inc.	Transdermal patch and method for administering 17-deacetyl norgestimate alone or in combination with an estrogen
US6245804B1 (en)	1997-05-30	2001-06-12	Schering Aktiengesellschaft	Nonsteroidal gestagens
DE19723722A1 (de) *	1997-05-30	1998-12-10	Schering Ag	Nichtsteroidale Gestagene
US5948433A (en)	1997-08-21	1999-09-07	Bertek, Inc.	Transdermal patch
DE19856475A1 (de) *	1998-11-27	2000-05-31	Schering Ag	Nichtsteroidale Entzündungshemmer
DE10038639A1 (de) *	2000-07-28	2002-02-21	Schering Ag	Nichtsteroidale Entzündungshemmer
ES2932076T3 (es) *	2017-10-27	2023-01-11	Association Pour La Rech A Ligbmc Ari	Moduladores agonistas de los receptores de glucocorticoides selectivos (SEGRAM) no esteroideos y usos de los mismos

2018
- 2018-05-17 EP EP18305612.6A patent/EP3569228A1/en not_active Withdrawn
- 2018-10-23 CN CN201880082668.1A patent/CN111511359A/zh active Pending
- 2018-10-23 PT PT187868237T patent/PT3700513T/pt unknown
- 2018-10-23 KR KR1020207014598A patent/KR20200085782A/ko not_active Ceased
- 2018-10-23 BR BR112020008350-0A patent/BR112020008350A2/pt not_active Application Discontinuation
- 2018-10-23 US US16/759,014 patent/US11179363B2/en active Active
- 2018-10-23 EP EP18786823.7A patent/EP3700513B1/en active Active
- 2018-10-23 MA MA050443A patent/MA50443A/fr unknown
- 2018-10-23 JP JP2020543706A patent/JP2021509411A/ja active Pending
- 2018-10-23 AU AU2018355698A patent/AU2018355698A1/en not_active Abandoned

Also Published As

Publication number	Publication date
JP2021509411A (ja)	2021-03-25
BR112020008350A2 (pt)	2020-11-03
KR20200085782A (ko)	2020-07-15
EP3700513B1 (en)	2022-08-24
CN111511359A (zh)	2020-08-07
AU2018355698A1 (en)	2020-05-14
EP3569228A1 (en)	2019-11-20
EP3700513A2 (en)	2020-09-02
US20210177798A1 (en)	2021-06-17
MA50443A (fr)	2020-09-02
US11179363B2 (en)	2021-11-23

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