PT3700513T - Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações - Google Patents

Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações

Info

Publication number: PT3700513T
Authority: PT; Portugal
Prior art keywords: segrams; glucocorticoid receptor; receptor agonistic; selective glucocorticoid; steroidal selective
Prior art date: 2018-05-17

Application number

PT187868237T

Other languages

English (en)

Original Assignee

Association Pour La Rech A Ligbmc Ari

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2018-05-17

Filing date

2018-10-23

Publication date

2022-11-30

2018-10-23 Application filed by Association Pour La Rech A Ligbmc Ari filed Critical Association Pour La Rech A Ligbmc Ari

2022-11-30 Publication of PT3700513T publication Critical patent/PT3700513T/pt

Links

102000003676 Glucocorticoid Receptors Human genes 0.000 title 1
108090000079 Glucocorticoid Receptors Proteins 0.000 title 1
230000001270 agonistic effect Effects 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Dermatology (AREA)
Epidemiology (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Ophthalmology & Optometry (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Emergency Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Furan Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

PT187868237T 2018-05-17 2018-10-23 Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações PT3700513T (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP18305612.6A EP3569228A1 (en)	2018-05-17	2018-05-17	Non-steroidal selective glucocorticoid receptor agonistic modulators (segrams) and uses thereof

Publications (1)

Publication Number	Publication Date
PT3700513T true PT3700513T (pt)	2022-11-30

Family

ID=62386318

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT187868237T PT3700513T (pt)	2018-05-17	2018-10-23	Moduladores agonistas de recetores de glicocorticoides seletivos (segram) não esteroides e suas utilizações

Country Status (9)

Country	Link
US (1)	US11179363B2 (pt)
EP (2)	EP3569228A1 (pt)
JP (1)	JP2021509411A (pt)
KR (1)	KR20200085782A (pt)
CN (1)	CN111511359A (pt)
AU (1)	AU2018355698A1 (pt)
BR (1)	BR112020008350A2 (pt)
MA (1)	MA50443A (pt)
PT (1)	PT3700513T (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US12150922B1 (en)	2023-12-08	2024-11-26	King Faisal University	Methods of inhibiting cyclooxygenase (COX) using tolterodine

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5262165A (en)	1992-02-04	1993-11-16	Schering Corporation	Transdermal nitroglycerin patch with penetration enhancers
US6010715A (en)	1992-04-01	2000-01-04	Bertek, Inc.	Transdermal patch incorporating a polymer film incorporated with an active agent
PL181582B1 (pl)	1995-06-07	2001-08-31	Ortho Mcneil Pharm Inc	Plaster na skóre do zapobiegania owulacji u kobiety oraz plaster na skóre do przeprowadzania hormonalnej terapii substytucyjnej PL PL PL PL PL PL PL PL
US6245804B1 (en)	1997-05-30	2001-06-12	Schering Aktiengesellschaft	Nonsteroidal gestagens
DE19723722A1 (de) *	1997-05-30	1998-12-10	Schering Ag	Nichtsteroidale Gestagene
US5948433A (en)	1997-08-21	1999-09-07	Bertek, Inc.	Transdermal patch
DE19856475A1 (de) *	1998-11-27	2000-05-31	Schering Ag	Nichtsteroidale Entzündungshemmer
DE10038639A1 (de) *	2000-07-28	2002-02-21	Schering Ag	Nichtsteroidale Entzündungshemmer
WO2019081517A2 (en) *	2017-10-27	2019-05-02	Association Pour La Recherche À L`Igbmc (Ari)	NON-STEROIDIC GLUCOCORTICOIC RECEPTOR (SEGRAM) RECEPTOR AGONIST MODULATORS AND USES THEREOF

2018
- 2018-05-17 EP EP18305612.6A patent/EP3569228A1/en not_active Withdrawn
- 2018-10-23 AU AU2018355698A patent/AU2018355698A1/en not_active Abandoned
- 2018-10-23 EP EP18786823.7A patent/EP3700513B1/en active Active
- 2018-10-23 JP JP2020543706A patent/JP2021509411A/ja active Pending
- 2018-10-23 BR BR112020008350-0A patent/BR112020008350A2/pt not_active Application Discontinuation
- 2018-10-23 PT PT187868237T patent/PT3700513T/pt unknown
- 2018-10-23 CN CN201880082668.1A patent/CN111511359A/zh active Pending
- 2018-10-23 KR KR1020207014598A patent/KR20200085782A/ko not_active Ceased
- 2018-10-23 MA MA050443A patent/MA50443A/fr unknown
- 2018-10-23 US US16/759,014 patent/US11179363B2/en active Active

Also Published As

Publication number	Publication date
EP3569228A1 (en)	2019-11-20
EP3700513B1 (en)	2022-08-24
AU2018355698A1 (en)	2020-05-14
MA50443A (fr)	2020-09-02
US20210177798A1 (en)	2021-06-17
CN111511359A (zh)	2020-08-07
US11179363B2 (en)	2021-11-23
BR112020008350A2 (pt)	2020-11-03
EP3700513A2 (en)	2020-09-02
KR20200085782A (ko)	2020-07-15
JP2021509411A (ja)	2021-03-25

Publication	Publication Date	Title
IL276295A (en)	2020-09-30	Modulators of chemokine receptors and their uses
IL295598A (en)	2022-10-01	Selective estrogen receptor antagonists
IL279224A (en)	2021-01-31	1-GLP agonist receptors and their use
ZA202003325B (en)	2021-07-28	Glucocorticoid receptor agonist and immunoconjugates thereof
SG11202103325WA (en)	2021-05-28	Androgen receptor modulators and methods for their use
HUE070423T2 (hu)	2025-06-28	GLP-1 receptor agonisták és alkalmazásuk
ZA201808623B (en)	2019-08-28	Glucocorticoid receptor agonist and immunoconjugates thereof
IL276330A (en)	2020-09-30	Spiro-lactam NMDA receptor modulators and their use
ZA201805573B (en)	2020-12-23	Selective estrogen receptor degraders and uses thereof
IL276332A (en)	2020-09-30	Spiro-lactam NMDA receptor modulators and their use
IL279990A (en)	2021-03-01	Selective estrogen receptor antagonists
IL274208A (en)	2020-06-30	Nonsteroidal selective agonist agonist modulators of glucocorticoid receptors (SERAMs) and their uses
HK40034699A (en)	2021-04-30	Non-steroidal selective glucocorticoid receptoragonistic modulators (segrams) and uses thereof
MA50443A (fr)	2020-09-02	Modulateurs agonistes de récepteurs de glucocorticoïdes sélectifs (segrams) non stéroïdiens et leurs utilisations
IL272940A (en)	2020-04-30	Single-immunoglobulin interleukin-1 receptor-related variants and their uses
EP3902549A4 (en)	2022-09-14	SHORT-ACTING SELECTIVE GLUCOCORTICOID RECEPTOR MODULATORS